
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Neurogenic locus notch homolog protein 1 | Homo sapiens | P46531 | 2000 nM|= 2000.0 nM | BindingDB, NPASS | |||
| NON-PROTEIN TARGET | = 4.0 nM | NPASS | |||||
| U373 MG | Homo sapiens | = 32.0 nM | NPASS | ||||
| HCT-15 | Homo sapiens | = 27.0 nM | NPASS | ||||
| A549 | Homo sapiens | = 5.0 nM | NPASS | ||||
| LoVo | Homo sapiens | = 17.0 nM | NPASS |