
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Neurogenic locus notch homolog protein 1 | Mus musculus | Q01705 | 120 nM|= 120.0 nM | BindingDB, NPASS | |||
| MCF7 | Homo sapiens | = 33.0 nM | NPASS | ||||
| HeLa | Homo sapiens | = 62.0 nM | NPASS | ||||
| BJ | Homo sapiens | = 26.0 nM | NPASS | ||||
| HEK293 | Homo sapiens | = 28.0 nM | NPASS | ||||
| CCRF-CEM | Homo sapiens | = 19.0 nM | NPASS | ||||
| HPBALL | Homo sapiens | = 14.0 nM | NPASS |