| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | | = 35000.0 nM|> 20000.0 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 13760.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| NAD(+) hydrolase SARM1 | Homo sapiens | Q6SZW1 | | = 140000.0 nM|= 110000.0 nM|= 77000.0 nM | | = 130000.0 nM | NPASS |
| Nucleic Acid | | | | | | = 36400.0 nM | NPASS |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | | = 3080.0 nM | | = 742.0 nM | NPASS |
| KM12C | Homo sapiens | | | = 76340.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 20600.0 nM | | | NPASS |
| LS174T | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 71550.0 nM|> 50000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 14390.0 nM|= 31720.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 7320.0 nM|= 6030.0 nM | | | NPASS |
| MKN-28 | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | = 442.0 nM|= 218.0 nM | = 0.36 ug.mL-1|= 0.141 ug.mL-1|= 0.148 ug.mL-1 | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 16440.0 nM | | | NPASS |
| Plasmodium yoelii | Plasmodium yoelii | | | = 548.0 nM | | | NPASS |
| Prolyl endopeptidase | Homo sapiens | P48147 | | = 145000.0 nM|= 142000.0 nM | | | NPASS |
| SGC-7901 | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | = 100.0 ug.mL-1 | | | NPASS |
| SMMC-7721 | Homo sapiens | | | = 25940.0 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 126200.0 nM|= 25000.0 nM | | | NPASS |
| Serine/threonine-protein kinase NEK7 | Homo sapiens | Q8TDX7 | | = 4200.0 nM | = 15600.0 nM | | NPASS |
| Serotonin 2b (5-HT2b) receptor | Homo sapiens | P41595 | | = 3437.0 nM | | = 2187.0 nM | NPASS |
| Serotonin 4 (5-HT4) receptor | Cavia porcellus | O70528 | | = 2222.0 nM | | = 370.0 nM | NPASS |
| Sigma opioid receptor | Homo sapiens | Q99720 | | = 1289.0 nM | | = 542.0 nM | NPASS |
| Sortase | Staphylococcus aureus | Q9S446 | | = 8.7 ug.mL-1 | | | NPASS |
| Sortase A | Staphylococcus aureus | Q9S446 | | = 8.7 ug.mL-1 | | | NPASS |
| Plasmodium falciparum (isolate K1 / Thailand) | Plasmodium falciparum K1 | | | = 968.0 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 130.0 nM | | | | NPASS |
| Retinoid X receptor alpha | Homo sapiens | P19793 | | | = 24800.0 nM | | NPASS |
| Hepatocyte | Rattus norvegicus | | | = 26.5 ug.mL-1 | | | NPASS |
| A2780 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 6270.0 nM|> 50000.0 nM | | | NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | = 374.0 nM|= 2740.0 nM | | = 289.0 nM | NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | = 774.0 nM|= 40.0 nM|= 610.0 nM|= 17400.0 nM | | | NPASS |
| Alpha-2b adrenergic receptor | Homo sapiens | P18089 | | = 601.0 nM | | = 274.0 nM | NPASS |
| Alpha-2c adrenergic receptor | Homo sapiens | P18825 | | = 2837.0 nM | | = 412.0 nM | NPASS |
| BGC-823 | Homo sapiens | | | = 7040.0 nM | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 16280.0 nM | | | NPASS |
| Butyrylcholinesterase | Equus caballus | Q9N1N9 | | = 18200.0 nM | | | NPASS |
| Butyrylcholinesterase | Homo sapiens | P06276 | | = 18970.0 nM|= 47200.0 nM | | | NPASS |
| CCRF S-180 | Mus musculus | | | = 25000.0 nM | | | NPASS |
| CHO-K1 | Cricetulus griseus | | | = 336000.0 nM | | | NPASS |
| Cell division protein ftsZ | Escherichia coli K-12 | P0A9A6 | | = 10000.0 nM|= 16000.0 nM | = 23.0 nM | | NPASS |
| C6 | Rattus norvegicus | | | > 20000.0 nM | | | NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | = 4504.2 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 146200000.0 ug.mL-1|= 8320.0 nM|= 11220.0 nM|= 49010.0 nM|= 53.91 ug.mL-1|> 50000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 138400000.0 ug.mL-1 | | | NPASS |
| Cholinesterase | Equus caballus | P81908 | | = 18200.0 nM|= 18210.0 nM | | = 9200.0 nM | NPASS |
| HL-60 | Homo sapiens | | | = 5830.0 nM|= 27420.0 nM | | | NPASS |
| HERG | Homo sapiens | Q12809 | | = 3100.0 nM | | | NPASS |
| HCT-8 | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 8450.0 nM|> 20000.0 nM|> 10000.0 nM|> 50000.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 39950.0 nM|> 10000.0 nM|= 83090.0 nM|= 25000.0 nM | | | NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 111000.0 nM | | | NPASS |
| ECa-109 cell line | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 16590.0 nM | | | NPASS |
| Human herpesvirus 5 | Human herpesvirus 5 | | | = 680.0 nM | | | NPASS |