| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Voltage-gated L-type calcium channel alpha-1C subunit | Rattus norvegicus | P22002 | | | | = 289.0 nM | NPASS |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus | P22002 | | | | 289 nM | BindingDB |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >567000 nM | | | BindingDB |
| Alpha-2c adrenergic receptor | Homo sapiens | P18825 | | | | = 5.0 nM | NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | | | 4.6 nM|3.3 nM|14 nM|13 nM|3.5 nM|5.7 nM|= 3.3 nM|= 4.6 nM|= 14.0 nM|= 5.7 nM|= 3.5 nM|= 13.0 nM | BindingDB, NPASS |
| Alpha-2a adrenergic receptor | Homo sapiens | P08913 | | | | = 8.2 nM | NPASS |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 5 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 15 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 8.2 nM | BindingDB |
| Alpha-2b adrenergic receptor | Homo sapiens | P18089 | | | | = 14.5 nM | NPASS |