| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | = 34900.0 nM|> 30000.0 nM | > 5.0 ug.mL-1|= 35950.0 nM|= 61600.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 25700.0 nM|> 30000.0 nM | = 39389.0 nM|> 10000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 36609.0 nM|> 10000.0 nM | | | NPASS |
| MKN-45 | Homo sapiens | | | = 53690.0 nM | | | NPASS |
| NCI-H187 | Homo sapiens | | | > 5.0 ug.mL-1 | | | NPASS |
| NCI-H1975 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | > 30000.0 nM | | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | >40000 nM | | | BindingDB |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens | Q9NPD5 | | 891 nM|= 891.25 nM | | 680 nM|= 680.0 nM | BindingDB, NPASS |
| SW-1736 | Homo sapiens | | > 60000.0 nM|> 30000.0 nM | | | | NPASS |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens | Q9Y6L6 | | 3802 nM|= 3801.89 nM | | 2110 nM|= 2110.0 nM | BindingDB, NPASS |
| LoVo | Homo sapiens | | | = 1170.0 nM|= 1390.0 nM | | | NPASS |
| Tissue factor | Homo sapiens | P13726 | | 0.221000 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-321] | Homo sapiens | P18031 | | | | 3600 nM | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-405] | Homo sapiens | P18031 | | | | 2000 nM | BindingDB |
| Ubiquitin carboxyl-terminal hydrolase 7 | Homo sapiens | Q93009 | | = 33500.0 nM | | | NPASS |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens | O15296 | | >40000 nM | | | BindingDB |
| Leishmania infantum | Leishmaitum | | | = 61600.0 nM | | | NPASS |
| M14 | Homo sapiens | | | = 58000.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 28050.0 nM|= 35870.0 nM | | | NPASS |
| 8505C | Homo sapiens | | = 38000.0 nM|> 30000.0 nM | | | | NPASS |
| A-375 | Homo sapiens | | > 60000.0 nM | | | | NPASS |
| KB | Homo sapiens | | | > 5.0 ug.mL-1|= 14631.0 nM|= 54430.0 nM|> 10000.0 nM | | | NPASS |
| A549 | Homo sapiens | | = 29000.0 nM|> 30000.0 nM | = 39000.0 nM|> 200000.0 nM|= 38640.0 nM|= 10249.0 nM|> 100000.0 nM|> 10000.0 nM|> 50000.0 nM|= 26230.0 nM | | | NPASS |
| AGS | Homo sapiens | | | = 36140.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase, type II | Homo sapiens | O15296 | | > 40000.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | > 40000.0 nM | | | NPASS |
| BGC-823 | Homo sapiens | | | = 52070.0 nM | | | NPASS |
| BT-20 | Homo sapiens | | | = 11800.0 nM | | | NPASS |
| A2780 | Homo sapiens | | = 19900.0 nM|> 30000.0 nM|> 60000.0 nM | | | | NPASS |
| DLD-1 | Homo sapiens | | | > 100000.0 nM|> 200000.0 nM | | | NPASS |
| Epidermal growth factor receptor | Homo sapiens | P00533 | | >20000 nM | | | BindingDB |
| Epidermal growth factor receptor erbB1 | Homo sapiens | P00533 | | > 20000.0 nM | | | NPASS |
| FaDu | Homo sapiens | | > 60000.0 nM|> 30000.0 nM | | | | NPASS |
| HL-60 | Homo sapiens | | | = 27520.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | = 50000.0 nM|> 30000.0 nM|> 60000.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | = 42270.0 nM|= 53960.0 nM|= 17.42 ug.mL-1 | | | NPASS |
| Coagulation factor III | Homo sapiens | P13726 | | = 0.221 nM | | | NPASS |