| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Nitric oxide synthase, inducible | Mus musculus | P29477 | | = 400.0 nM | | | NPASS |
| Nuclear factor erythroid 2-related factor 2 | Homo sapiens | Q16236 | = 19080.0 nM|= 1200.0 nM|= 580.0 nM|= 879.0 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | | = 27300.0 nM|= 11000.0 nM|= 95000.0 nM|= 6250.0 nM|= 13270.0 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 18440.0 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 22010.0 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | | = 7648.0 nM|= 11570.0 nM | | | NPASS |
| Macrophage migration inhibitory factor | Homo sapiens | P14174 | | = 2200.0 nM|= 11000.0 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 32380.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 10000.0 nM|= 22180.0 nM | | | NPASS |
| Protein-glutamine gamma-glutamyltransferase | Homo sapiens | P21980 | | | | = 366000.0 nM | NPASS |
| SGC-7901 | Homo sapiens | | | = 24950.0 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | = 7870.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 17840.0 nM | | | NPASS |
| SiHa | Homo sapiens | | | = 9953.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | > 120000.0 nM|= 15000.0 nM|= 120000.0 nM|= 102000.0 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 22470.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | = 13720.0 nM | | | NPASS |
| PC-9 | | | | = 6308.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 17660.0 nM|> 10000.0 nM|= 23130.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 21250.0 nM | | | NPASS |
| Leishmania infantum | Leishmaitum | | | = 16500.0 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 15760.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 21990.0 nM|= 11930.0 nM|> 10000.0 nM|= 20180.0 nM | | | NPASS |
| AGS | Homo sapiens | | | = 18410.0 nM | | | NPASS |
| ARPE-19 | Homo sapiens | | | = 10000.0 nM | | | NPASS |
| BACH1/MafK | Homo sapiens | | | = 15848.93 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Caco-2 | Homo sapiens | | | = 79830.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 10000.0 nM|= 13800.0 nM | | | NPASS |
| Epidermal growth factor receptor erbB1 | Homo sapiens | P00533 | | = 9000.0 nM | | | NPASS |
| HCC827 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 11590.0 nM|= 36730.0 nM | | | NPASS |
| HONE1 cell line | Homo sapiens | | | = 19260.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 66090.0 nM|> 10000.0 nM | | | NPASS |
| Hep 3B2 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| LoVo | Homo sapiens | | | = 22900.0 nM|= 18520.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | = 4000.0 nM | = 24890.0 nM|= 14050.0 nM|= 8357.0 nM|= 20990.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 3800.0 nM|= 15000.0 nM|> 10000.0 nM | | | NPASS |
| Keap1/Nrf2 | Homo sapiens | | = 870.0 nM | > 100000.0 nM | > 10000.0 nM | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 23300.0 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 24520.0 nM | | | NPASS |