IMPPAT Phytochemical information: 
Bruceantin

Bruceantin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
U-266Homo sapiens= 49.0 nMNPASS
RPMI-8226Homo sapiens= 12.8 nMNPASS
REHHomo sapiens= 0.02 ug.mL-1NPASS
Plasmodium falciparum (isolate K1 / Thailand)Plasmodium falciparum K1= 0.0008 ug.mL-1NPASS
NON-PROTEIN TARGET< 0.015 ug.mL-1NPASS
NCI-H929Homo sapiens= 115.0 nMNPASS
NB-4Homo sapiens< 0.015 ug.mL-1NPASS
Kasumi 1= 0.02 ug.mL-1NPASS
HeLaHomo sapiens= 51.0 nM|= 29.0 nMNPASS
HT-29Homo sapiens= 22.0 nMNPASS
HL-60Homo sapiens= 20.0 nM= 40.0 nM|= 0.02 ug.mL-1|= 12.2 nMNPASS
DaudiHomo sapiens< 0.015 ug.mL-1NPASS
Cytochrome P450 2D6Homo sapiensP10635= 514000.0 nMNPASS
BV-173Homo sapiens< 0.015 ug.mL-1NPASS
U-937Homo sapiens< 0.015 ug.mL-1NPASS
Human immunodeficiency virus type 1 reverse transcriptaseHuman immunodeficiency virus 1Q72547> 200.0 ug.mL-1NPASS
Entamoeba histolyticaEoeba histolytica= 0.019 ug.mL-1NPASS