
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| MCF7 | Homo sapiens | = 600.0 nM | NPASS | ||||
| Cytochrome P450 3A4 | Homo sapiens | P08684 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2D6 | Homo sapiens | P10635 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2C9 | Homo sapiens | P11712 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2C8 | Homo sapiens | P10632 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2C19 | Homo sapiens | P33261 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2E1 | Homo sapiens | P05181 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2B6 | Homo sapiens | P20813 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2A6 | Homo sapiens | P11509 | >20000 nM|> 20000.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | 1060 nM|950 nM|= 1060.0 nM|= 950.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 1A2 | Homo sapiens | P05177 | 2500 nM|= 2500.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 1A1 | Homo sapiens | P04798 | 14800 nM|= 14800.0 nM | 20 nM|71 nM|= 20.0 nM|= 71.0 nM | BindingDB, NPASS | ||
| BV-2 | Mus musculus | > 100000.0 nM | NPASS | ||||
| Cytochrome P450 2C18 | Homo sapiens | P33260 | >20000 nM|> 20000.0 nM | BindingDB, NPASS |