| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Procathepsin L | Homo sapiens | P07711 | | 30340 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens | P18031 | | >50000 nM | | | BindingDB |
| T47D | Homo sapiens | | | = 12110.0 nM | | | NPASS |
| Sialidase | Clostridium perfringens | P10481 | | 29900 nM|= 8.13 ug.mL-1 | | | BindingDB, NPASS |
| SNU-638 | Homo sapiens | | | = 10410.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | > 50000.0 nM | | | NPASS |
| Tyrosyl-DNA phosphodiesterase 1 | Homo sapiens | Q9NUW8 | | 45000 nM|= 45000.0 nM | | | BindingDB, NPASS |
| Neuraminidase | InflueA virus (A/WSN/1933(H1N1)) | P03470 | | 21000 nM|21400 nM|8130 nM|9240 nM|30300 nM | | | BindingDB |
| NON-PROTEIN TARGET | | | | > 30000.0 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 68000.0 nM | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | ~ 3000.0 nM | | | NPASS |
| Cathepsin L | Homo sapiens | P07711 | | = 30340.0 nM | | | NPASS |
| Cathepsin B | Homo sapiens | P07858 | | 57680 nM|= 57680.0 nM | | | BindingDB, NPASS |
| Neuraminidase | InflueA virus | B4URF0 | | = 2.19 ug.mL-1|= 2.49 ug.mL-1|= 5.7 ug.mL-1|= 5.8 ug.mL-1|= 8.23 ug.mL-1 | | | NPASS |