
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Adenosine receptor A3 | Homo sapiens | P0DMS8 | >100000 nM | 103000 nM | BindingDB | ||
| Platelet-derived growth factor receptor alpha/beta | Mus musculus | P05622|P26618 | >100000 nM | >100000 nM | BindingDB | ||
| Adenosine receptor A2a/A2b | Rattus norvegicus | P29276|P30543 | >250000 nM|250000 nM | BindingDB | |||
| Adenosine receptor A2b | Homo sapiens | P29275 | 130000 nM | BindingDB | |||
| Adenosine receptor A1 | Rattus norvegicus | P25099 | >10000 nM|105000 nM | BindingDB | |||
| Adenosine receptor A1 | Homo sapiens | P30542 | 105000 nM | 105000 nM | BindingDB | ||
| Adenosine receptor A1 | Bos taurus | P28190 | >10000 nM | BindingDB | |||
| Adenosine receptor A2a | Homo sapiens | P29274 | >250000 nM | >10000 nM|>250000 nM | BindingDB |