
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Amyloid-beta A4 protein | Homo sapiens | P05067 | = 3000.0 nM | NPASS | |||
| Beta-secretase 1 | Homo sapiens | P56817 | 4500 nM|= 4500.0 nM|= 2400.0 nM | 5300 nM|= 5300.0 nM | BindingDB, NPASS | ||
| Pyruvate kinase PKM | Homo sapiens | P14618 | 850 nM | BindingDB | |||
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | = 850.0 nM | NPASS |