| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| HepG2 | Homo sapiens | | | = 59000.0 nM | | | NPASS |
| L-lactate dehydrogenase A chain | Homo sapiens | P00338 | | | | 14000 nM|= 14000.0 nM | BindingDB, NPASS |
| Lysophosphatidylserine lipase ABHD12 | Homo sapiens | Q8N2K0 | | 11600 nM | | | BindingDB |
| MCF7 | Homo sapiens | | | = 57000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 5000.0 nM | | | NPASS |
| Monoacylglycerol lipase ABHD12 | Homo sapiens | Q8N2K0 | | = 11600.0 nM | | | NPASS |
| Monoacylglycerol lipase ABHD6 | Homo sapiens | Q9BV23 | | 48200 nM|= 48200.0 nM | | | BindingDB, NPASS |
| Monoglyceride lipase | Homo sapiens | Q99685 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| Mus musculus | Mus musculus | | | = 4.0 nM | | | NPASS |
| N-arachidonyl glycine receptor | Homo sapiens | Q14330 | 4610 nM|= 4610.0 nM|= 960.0 nM | | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily M member 8 | Homo sapiens | Q7Z2W7 | | = 160.0 nM | | | NPASS |
| OVCAR | Homo sapiens | | | = 63000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 65000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 720.0 nM|= 790.0 nM | | | NPASS |
| Pregnane X receptor | Homo sapiens | O75469 | = 31600.0 nM|= 12600.0 nM | | | | NPASS |
| SH-SY5Y | Homo sapiens | | | = 50000.0 nM | | | NPASS |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus | Q9R0C9 | | | | >100000 nM | BindingDB |
| T-24 | Homo sapiens | | | = 13.04 ug.mL-1 | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | 230 nM|= 230.0 nM | | | | BindingDB, NPASS |
| Hemozoin | Plasmodium falciparum | | | = 11300.0 nM | | | NPASS |
| Nuclear receptor subfamily 1 group I member 2 | Homo sapiens | O75469 | 31600 nM|12600 nM | | | | BindingDB |
| HCT-116 | Homo sapiens | | | = 42000.0 nM | | | NPASS |
| Glycine receptor subunit alpha-1 | Homo sapiens | P23415 | 1300 nM|= 1300.0 nM | | | | BindingDB, NPASS |
| G-protein coupled receptor 55 | Homo sapiens | Q9Y2T6 | >10000 nM|= 14200.0 nM|> 10000.0 nM | 14200 nM|= 14200.0 nM | | | BindingDB, NPASS |
| A549 | Homo sapiens | | | = 45000.0 nM | | | NPASS |
| Anandamide amidohydrolase | Homo sapiens | O00519 | | = 43600.0 nM | | | NPASS |
| Cannabinoid CB1 receptor | Homo sapiens | P21554 | = 17.0 nM|= 77.5 nM|= 43.0 nM | = 2.8 nM | | = 41.0 nM|= 28.5 nM|= 17.0 nM|= 2.9 nM|= 40.0 nM|= 10.0 nM|= 3.88 nM|= 40.7 nM|= 22.0 nM|= 18.0 nM|= 39.5 nM | NPASS |
| Cannabinoid CB1 receptor | Mus musculus | P47746 | | | | = 41.0 nM|= 40.0 nM|= 15.3 nM | NPASS |
| Cannabinoid CB1 receptor | Rattus norvegicus | P20272 | = 11.0 nM|= 199.53 nM | = 5.8 nM | | = 47.6 nM|= 66.5 nM|= 80.3 nM|= 41.0 nM|= 37.0 nM|= 39.5 nM|= 36.0 nM | NPASS |
| Cannabinoid CB2 receptor | Mus musculus | P47936 | = 7.3 nM | | | = 39.3 nM|= 9.2 nM|= 40.0 nM | NPASS |
| Cannabinoid receptor | Homo sapiens | P21554 | | | | = 41.0 nM | NPASS |
| Cannabinoid receptor | Rattus norvegicus | P20272 | | = 5.8 nM|= 218.0 nM | | = 46.0 nM|= 82.0 nM | NPASS |
| Cannabinoid receptor 1 | Homo sapiens | P21554 | 78 nM|17 nM|43 nM | 2.8 nM | | 13.7 nM|15.3 nM|5.05 nM|10.190000 nM|41 nM|10 nM|29 nM|22 nM|18 nM|17 nM|2.9 nM|40 nM | BindingDB |
| Cannabinoid receptor 1 | Mouse | P47746 | 77 nM | | | | BindingDB |
| Cannabinoid CB2 receptor | Homo sapiens | P34972 | = 1.5 nM|= 12.3 nM|= 12.0 nM | = 9.5 nM | | = 32.2 nM|= 36.0 nM|= 25.0 nM|= 3.3 nM|= 41.0 nM|= 24.0 nM|= 71.6 nM|= 36.4 nM|= 46.0 nM|= 42.0 nM|= 40.0 nM|= 47.0 nM | NPASS |
| Cannabinoid receptor 1 | Rattus norvegicus | P20272 | 11 nM|200 nM | 5.8 nM | | 80 nM|67 nM|40 nM|41 nM|36 nM|48 nM|37 nM | BindingDB |
| Cannabinoid receptor 1/2 | Homo sapiens | P21554|P34972 | | | | 41 nM | BindingDB |
| Cannabinoid receptor 1/2 | Rattus norvegicus | P20272|Q9QZN9 | | 5.8 nM|218 nM | | 46 nM|82 nM | BindingDB |
| Cannabinoid receptor 2 | Homo sapiens | P34972 | 12 nM|1.5 nM | 9.5 nM | | 25.06 nM|22.9 nM|44.9 nM|3.13 nM|16.850000 nM|32 nM|36 nM|25 nM|46 nM|42 nM|3.3 nM|41 nM|40 nM|24 nM|47 nM | BindingDB |
| Cannabinoid receptor 2 | Mus musculus | P47936 | 7.3 nM | | | 40 nM|9.2 nM|39 nM | BindingDB |
| D(3) dopamine receptor | Homo sapiens | P35462 | 10 nM | | | | BindingDB |
| Dopamine D3 receptor | Homo sapiens | P35462 | = 10.2 nM | | | | NPASS |
| Fatty acid-binding protein, liver | Mus musculus | P12710 | | | | 1.0e+3 nM | BindingDB |
| Fatty-acid amide hydrolase 1 | Homo sapiens | O00519 | | 43600 nM | | | BindingDB |
| Cannabinoid receptor 1 | Mus musculus | P47746 | | | | 15 nM|40 nM|41 nM | BindingDB |