| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | = 3400.0 nM|= 700.0 nM | = 13000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 4 | Homo sapiens | Q9HBA0 | = 5100.0 nM | = 1300.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 3 | Homo sapiens | Q8NET8 | = 1000.0 nM | = 66000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 2 | Rattus norvegicus | Q9WUD2 | = 1700.0 nM | = 1500.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 2 | Homo sapiens | Q9Y5S1 | = 1700.0 nM | = 1500.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily M member 8 | Homo sapiens | Q7Z2W7 | | = 160.0 nM | | | NPASS |
| Vanilloid receptor | Homo sapiens | Q8NER1 | = 1300.0 nM | = 2600.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | = 700.0 nM | = 13000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily M member 8 | Rattus norvegicus | Q8R455 | | = 160.0 nM | | | NPASS |
| RBL-2H3 | Rattus norvegicus | | | = 11300.0 nM | | | NPASS |
| Anandamide amidohydrolase | Rattus norvegicus | P97612 | | > 100000.0 nM | | | NPASS |
| Cannabinoid CB1 receptor | Homo sapiens | P21554 | | = 3310.0 nM | | = 760.0 nM|= 897.0 nM|= 2600.0 nM | NPASS |
| Cannabinoid CB1 receptor | Rattus norvegicus | P20272 | | | | = 440.0 nM | NPASS |
| Sn1-specific diacylglycerol lipase alpha | Homo sapiens | Q9Y4D2 | | > 100000.0 nM | | | NPASS |
| Inhibin alpha chain | Homo sapiens | P05111 | | = 5200.0 nM | | | NPASS |
| N-acylsphingosine-amidohydrolase | Homo sapiens | Q02083 | | > 100000.0 nM | | | NPASS |
| Peroxisome proliferator-activated receptor gamma | Homo sapiens | P37231 | = 15700.0 nM | | | | NPASS |
| Cannabinoid CB2 receptor | Homo sapiens | P34972 | | = 3460.0 nM | | = 880.0 nM|= 153.0 nM|= 2700.0 nM|= 1220.0 nM | NPASS |