| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| OVCAR | Homo sapiens | | | = 77000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 78000.0 nM | | | NPASS |
| Peroxisome proliferator-activated receptor gamma | Homo sapiens | P37231 | >25000 nM|> 25000.0 nM | | | | BindingDB, NPASS |
| RBL-2H3 | Rattus norvegicus | | | = 25000.0 nM | | | NPASS |
| SH-SY5Y | Homo sapiens | | | = 97000.0 nM | | | NPASS |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus | Q9R0C9 | | | | >10000 nM | BindingDB |
| Sn1-specific diacylglycerol lipase alpha | Homo sapiens | Q9Y4D2 | | > 50000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | 180 nM|= 180.0 nM | 400 nM|210 nM|= 210.0 nM|= 400.0 nM | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | 180 nM|= 180.0 nM | | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens | Q8NER1 | 6200 nM | 82000 nM | | | BindingDB |
| Transient receptor potential cation channel subfamily V member 2 | Homo sapiens | Q9Y5S1 | 19000 nM|= 19000.0 nM | 15700 nM|= 15700.0 nM | | | BindingDB, NPASS |
| N-acylsphingosine-amidohydrolase | Homo sapiens | Q02083 | | > 50000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 3 | Homo sapiens | Q8NET8 | 5300 nM|= 5300.0 nM | 9400 nM|= 9400.0 nM | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily V member 4 | Homo sapiens | Q9HBA0 | 16100 nM|= 16100.0 nM | 5400 nM|= 5400.0 nM | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily V member 4 | Rattus norvegicus | Q9ERZ8 | 16100 nM|= 16100.0 nM | | | | BindingDB, NPASS |
| Transient receptor potential cation channel, subfamily V, member 3 | Rattus norvegicus | | 5300 nM | | | | BindingDB |
| Transient receptor potential cation channel, subfamily V, member 3 | Rattus norvegicus | E9PU00 | = 5300.0 nM | | | | NPASS |
| Vanilloid receptor | Homo sapiens | Q8NER1 | = 6200.0 nM | = 82000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily M member 8 | Rattus norvegicus | Q8R455 | | 210 nM|= 210.0 nM | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily V member 2 | Rattus norvegicus | Q9WUD2 | 19000 nM|= 19000.0 nM | | | | BindingDB, NPASS |
| N-acylethanolamine-hydrolyzing acid amidase | Homo sapiens | Q02083 | | >50000 nM | | | BindingDB |
| HepG2 | Homo sapiens | | | = 74000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 91000.0 nM | | | NPASS |
| Anandamide amidohydrolase | Rattus norvegicus | P97612 | | > 50000.0 nM | | | NPASS |
| Cannabinoid CB1 receptor | Homo sapiens | P21554 | = 75.0 nM | | | = 308.0 nM|= 13.0 nM|= 1100.0 nM|= 70.0 nM | NPASS |
| Cannabinoid CB1 receptor | Rattus norvegicus | P20272 | = 120.0 nM|= 316.23 nM | | | = 392.2 nM|= 211.2 nM | NPASS |
| MCF7 | Homo sapiens | | | = 81000.0 nM | | | NPASS |
| Cannabinoid receptor 1 | Homo sapiens | P21554 | 75 nM | | | 308 nM|310 nM|13 nM|1100 nM|70 nM | BindingDB |
| Cannabinoid receptor 1 | Rattus norvegicus | P20272 | 120 nM|316 nM | | | 308 nM|211 nM|392.2 nM | BindingDB |
| Cannabinoid receptor 2 | Homo sapiens | P34972 | 261.2 nM|73 nM|60.0 nM | | | 126 nM|96 nM|95 nM|16 nM|70 nM|300 nM | BindingDB |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | | | 541 nM|= 541.0 nM | BindingDB, NPASS |
| Cannabinoid CB2 receptor | Homo sapiens | P34972 | = 261.2 nM|= 73.0 nM | | | = 126.4 nM|= 96.0 nM|= 16.0 nM|= 70.0 nM|= 300.0 nM | NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | | | 148 nM|= 148.0 nM | BindingDB, NPASS |
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | 30400 nM|= 30400.0 nM | | 1000 nM|= 1000.0 nM | BindingDB, NPASS |
| Cytochrome P450 2B6 | Homo sapiens | P20813 | | | | 39000 nM|2550 nM|= 39000.0 nM|= 2550.0 nM | BindingDB, NPASS |
| Cytochrome P450 2J2 | Homo sapiens | P51589 | | 19000 nM|= 19000.0 nM | | | BindingDB, NPASS |
| Diacylglycerol lipase-alpha | Homo sapiens | Q9Y4D2 | | >50000 nM | | | BindingDB |
| Fatty-acid amide hydrolase 1 [30-579] | Rattus norvegicus | P97612 | | >50000 nM | | | BindingDB |
| HCT-116 | Homo sapiens | | | = 80000.0 nM | | | NPASS |
| HT-22 | Mus musculus | | = 610.0 nM | | | | NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | | | 79 nM|= 79.0 nM | BindingDB, NPASS |