| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Rattus norvegicus | Rattus norvegicus | | = 154.88 nM|= 575.44 nM|= 169.82 nM | | | | NPASS |
| Muscarinic acetylcholine receptor M5 | Homo sapiens | P08912 | 1300 nM | | | | BindingDB |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus | P08485 | | 470 nM|= 470.0 nM | | 1400 nM|= 1400.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | | | | 23 nM|1400 nM|28000 nM|= 1400.0 nM|= 23.0 nM|= 28000.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus | P08483 | 130 nM|= 130.0 nM | | | 21600 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | 1000 nM | | | | BindingDB |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus | P10980 | | 3900 nM|490 nM|= 490.0 nM|= 3900.0 nM | | 490.0 nM|75 nM|= 75.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | 12 nM | | | BindingDB |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus | P08482 | 219 nM|= 219.0 nM | 5680 nM|= 5680.0 nM | | 15000 nM|27 nM|5680 nM|12 nM|= 27.0 nM|= 12.0 nM|= 5680.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | 5300 nM | | | 56.0 nM|18197 nM|= 56.0 nM|= 18197.01 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor | Rattus norvegicus | P10980 | | = 12.0 nM | | = 14.0 nM|= 4400.0 nM|= 8.3 nM | NPASS |
| Muscarinic acetylcholine receptor | Cavia porcellus | | | | 23988 nM|1122 nM | | BindingDB |
| Cavia porcellus | Cavia porcellus | | = 58.88 nM|= 31.62 nM | | = 19952.62 nM|= 24547.09 nM|= 1122.02 nM|= 23988.33 nM | | NPASS |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | | 449 nM|3900 nM|= 449.0 nM|= 3900.0 nM | 24547 nM|19953 nM | 25 nM|72.0 nM|75 nM|490 nM|= 25.0 nM|= 72.0 nM|= 75.0 nM|= 489.78 nM | BindingDB, NPASS |