IMPPAT Phytochemical information: 
Muscarine

Muscarine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Rattus norvegicusRattus norvegicus= 154.88 nM|= 575.44 nM|= 169.82 nMNPASS
Muscarinic acetylcholine receptor M5Homo sapiensP089121300 nMBindingDB
Muscarinic acetylcholine receptor M4Rattus norvegicusP08485470 nM|= 470.0 nM1400 nM|= 1400.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M4Homo sapiensP0817323 nM|1400 nM|28000 nM|= 1400.0 nM|= 23.0 nM|= 28000.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M3Rattus norvegicusP08483130 nM|= 130.0 nM21600 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M3Homo sapiensP203091000 nMBindingDB
Muscarinic acetylcholine receptor M2Rattus norvegicusP109803900 nM|490 nM|= 490.0 nM|= 3900.0 nM490.0 nM|75 nM|= 75.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5Rattus norvegicusP08482|P08483|P08485|P08911|P1098012 nMBindingDB
Muscarinic acetylcholine receptor M1Rattus norvegicusP08482219 nM|= 219.0 nM5680 nM|= 5680.0 nM15000 nM|27 nM|5680 nM|12 nM|= 27.0 nM|= 12.0 nM|= 5680.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M1Homo sapiensP112295300 nM56.0 nM|18197 nM|= 56.0 nM|= 18197.01 nMBindingDB, NPASS
Muscarinic acetylcholine receptorRattus norvegicusP10980= 12.0 nM= 14.0 nM|= 4400.0 nM|= 8.3 nMNPASS
Muscarinic acetylcholine receptorCavia porcellus23988 nM|1122 nMBindingDB
Cavia porcellusCavia porcellus= 58.88 nM|= 31.62 nM= 19952.62 nM|= 24547.09 nM|= 1122.02 nM|= 23988.33 nMNPASS
Muscarinic acetylcholine receptor M2Homo sapiensP08172449 nM|3900 nM|= 449.0 nM|= 3900.0 nM24547 nM|19953 nM25 nM|72.0 nM|75 nM|490 nM|= 25.0 nM|= 72.0 nM|= 75.0 nM|= 489.78 nMBindingDB, NPASS