| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Mitochondrial import inner membrane translocase subunit TIM10 | Saccharomyces cerevisiae S288c | P87108 | | = 19700.0 nM | | | NPASS |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 5020.0 nM|= 2740.0 nM | | = 710.0 nM | NPASS |
| Monoamine oxidase B | Homo sapiens | P27338 | | = 2560.0 nM|= 2580.0 nM | | = 21500.0 nM | NPASS |
| NACHT, LRR and PYD domains-containing protein 3 | Homo sapiens | Q96P20 | | 24200 nM|= 24200.0 nM | | | BindingDB, NPASS |
| NCI-H1299 | Homo sapiens | | | = 18930.0 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 20700.0 nM|= 20500.0 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 1400.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 8500.0 nM|= 15000.0 nM|= 17110.0 nM|= 17140.0 nM|= 20300.0 nM|= 5300.0 nM|= 20340.0 nM | | | NPASS |
| NHDF | Homo sapiens | | | = 24100.0 nM | | | NPASS |
| Proteasome Macropain subunit MB1 | Homo sapiens | P28074 | | = 10000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 28100.0 nM|= 48600.0 nM|= 6200.0 nM | = 7570.0 nM|= 3840.0 nM|= 82500.0 nM|= 31390.0 nM|= 24410.0 nM|= 12520.0 nM|= 27890.0 nM|= 10300.0 nM|= 48000.0 nM|= 50000.0 nM|= 100000.0 nM|= 25430.0 nM|= 26230.0 nM|= 49850.0 nM|= 44710.0 nM|= 15060.0 nM|= 24540.0 nM|= 38300.0 nM|= 72700.0 nM|= 51700.0 nM|= 42000.0 nM|= 24600.0 nM|= 30000.0 nM|= 7500.0 nM|> 25000.0 nM | | | NPASS |
| Microtubule-associated protein tau | Homo sapiens | P10636 | | 3000 nM|3500 nM|13000 nM|= 3000.0 nM|= 3500.0 nM|= 13000.0 nM|> 200000.0 nM | | | BindingDB, NPASS |
| No relevant target | | | | = 28.0 ug.mL-1 | | | NPASS |
| Nuclear factor erythroid 2-related factor 2 | Homo sapiens | Q16236 | 21000 nM|= 21000.0 nM | | | | BindingDB, NPASS |
| PANC-1 | Homo sapiens | | | = 53000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 12220.0 nM|= 18800.0 nM|= 25430.0 nM|= 18650.0 nM|= 2000.0 nM|= 18710.0 nM|= 20900.0 nM|= 19980.0 nM|= 39000.0 nM | | | NPASS |
| PWR-1E | Homo sapiens | | | = 8140.0 nM|= 8850.0 nM | | | NPASS |
| Plasmodium falciparum 3D7 | Plasmodium falciparum 3D7 | | | = 25000.0 nM | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 30000 nM | | | BindingDB |
| Prostaglandin E synthase | Homo sapiens | O14684 | | 300 nM|220 nM|= 220.0 nM|= 200.0 nM|= 300.0 nM | | | BindingDB, NPASS |
| Prostaglandin G/H synthase 1/2 | Bos taurus | O62664|O62698 | | 2000 nM | | | BindingDB |
| NIH3T3 | Mus musculus | | | = 9510.0 nM | | | NPASS |
| MRC5 | Homo sapiens | | | = 51230.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 25670.0 nM|= 7200.0 nM|= 23870.0 nM|= 22690.0 nM|= 32330.0 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 58550.0 nM|= 42890.0 nM | | | NPASS |
| Histone deacetylase 2 | Homo sapiens | Q92769 | | | | 97670 nM|= 97670.0 nM | BindingDB, NPASS |
| Histone deacetylase 8 | Homo sapiens | Q9BY41 | | | | 64980 nM|= 64980.0 nM | BindingDB, NPASS |
| Hs-578T | Homo sapiens | | | = 55450.0 nM | | | NPASS |
| Influenza A virus | InflueA virus | | | = 6700.0 nM | | | NPASS |
| Intestinal alkaline phosphatase | Homo sapiens | P09923 | | > 100000.0 nM | | | NPASS |
| Intestinal alkaline phosphatase | Mus musculus | P24822 | | = 18700.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 4290.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 23120.0 nM|= 36000.0 nM|= 46760.0 nM | | | NPASS |
| KM12 | Homo sapiens | | | = 16000.0 nM | | | NPASS |
| Proteasome subunit beta type-5 | Homo sapiens | P28074 | | 10000 nM | | | BindingDB |
| MGC-803 | Homo sapiens | | | > 20000.0 nM|= 21200.0 nM | | | NPASS |
| LN-229 | Homo sapiens | | | = 15000.0 nM | | | NPASS |
| Lactoylglutathione lyase | Homo sapiens | Q04760 | | | | 5.00 nM | BindingDB |
| Leishmania amazonensis | Leishmaamazonensis | | | > 100000.0 nM | | | NPASS |
| Lymphocyte antigen 96 | Homo sapiens | Q9Y6Y9 | | | 379000 nM|= 379000.0 nM | | BindingDB, NPASS |
| Lysine-specific histone demethylase 1 | Homo sapiens | O60341 | | = 9600.0 nM | | | NPASS |
| Lysine-specific histone demethylase 1A | Homo sapiens | O60341 | | 9600 nM | | | BindingDB |
| MCF7 | Homo sapiens | | | = 32200.0 nM|= 46250.0 nM|= 42890.0 nM|= 22100.0 nM|= 9800.0 nM|= 19900.0 nM|= 9280.0 nM|= 17100.0 nM|= 68250.0 nM|= 22500.0 nM|= 83100.0 nM|= 2940.0 nM|= 2080.0 nM|= 2030.0 nM|= 29300.0 nM|= 13700.0 nM|= 61710.0 nM|= 88.0 nM|= 41900.0 nM | | | NPASS |
| MCF7R | Homo sapiens | | | = 26200.0 nM | | | NPASS |
| MDA-MB-157 | Homo sapiens | | | = 40380.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 15810.0 nM|= 16230.0 nM|= 12000.0 nM|> 10000.0 nM|= 11450.0 nM|= 26500.0 nM|= 75300.0 nM|= 31390.0 nM|= 53510.0 nM | | | NPASS |
| MDA-MB-453 | Homo sapiens | | | = 32400.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 13610.0 nM|= 2000.0 nM | | | NPASS |
| Proto-oncogene tyrosine-protein kinase Src | Mus musculus | P05480 | | 2200 nM | | | BindingDB |
| SW480 | Homo sapiens | | | = 17940.0 nM|= 15000.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 14700.0 nM|> 100000.0 nM|= 15950.0 nM|= 19100.0 nM|= 800.0 nM|= 3000.0 nM|= 3500.0 nM|= 2200.0 nM|= 11200.0 nM|= 1890.0 nM|= 12300.0 nM | | | NPASS |
| Thioredoxin reductase 3 | Homo sapiens | Q86VQ6 | | 39420 nM|41420 nM|40560 nM | | | BindingDB |
| Thiosulfate sulfurtransferase | Homo sapiens | Q16762 | | 56000 nM|= 56000.0 nM | | | BindingDB, NPASS |
| Tissue factor | Homo sapiens | P13726 | | 13 nM | | | BindingDB |
| Toll-like receptor 9 | Homo sapiens | Q9NR96 | | = 8362.0 nM | | | NPASS |
| Trichomonas vaginalis | Trichomonas vaginalis | | = 100.0 ug.mL-1 | | | | NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | = 1780.0 nM | = 3600.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 3120.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | = 15000.0 nM | = 67300.0 nM | | | NPASS |
| Tyrosinase | Homo sapiens | P14679 | | 5000 nM|= 5000.0 nM | | | BindingDB, NPASS |
| Tyrosine-protein kinase SRC | Mus musculus | P05480 | | = 2200.0 nM | | | NPASS |
| Thioredoxin reductase | Homo sapiens | Q86VQ6 | | = 39420.0 nM|= 41420.0 nM|= 40560.0 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 15260.0 nM|= 25810.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 1880.0 nM | | | NPASS |
| U2OS | Homo sapiens | | = 22800.0 nM|= 34400.0 nM | | | | NPASS |
| U373 MG | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | > 25000.0 nM|= 25000.0 nM|= 17870.0 nM|= 10970.0 nM | | | NPASS |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus | Q02485 | | >100000 nM | | | BindingDB |
| Voltage-gated L-type calcium channel | Rattus norvegicus | P27732 | | > 100000.0 nM | | | NPASS |
| WRL68 | Homo sapiens | | | = 27800.0 nM | | | NPASS |
| WiDr | Homo sapiens | | | = 26820.0 nM | | | NPASS |
| Y79 | Homo sapiens | | | = 30000.0 nM | | | NPASS |
| Histone deacetylase 1 | Homo sapiens | Q13547 | | | | 50790 nM|= 50790.0 nM | BindingDB, NPASS |
| U-87 MG | Homo sapiens | | | = 16000.0 nM|= 7150.0 nM | | | NPASS |
| QGY-7703 | Homo sapiens | | | = 21440.0 nM|= 23910.0 nM|= 22500.0 nM | | | NPASS |
| THP-1 | Homo sapiens | | | = 22540.0 nM | | | NPASS |
| T47D | Homo sapiens | | | = 47910.0 nM|= 19000.0 nM|= 11000.0 nM | | | NPASS |
| RWPE-1 | Homo sapiens | | | = 15620.0 nM | | | NPASS |
| Raji | Homo sapiens | | | = 97.0 molar ratio | | | NPASS |
| Rattus norvegicus | Rattus norvegicus | | | = 53.4 nM | | | NPASS |
| Replicase polyprotein 1ab | Human SARS coronavirus | P0C6X7 | >10000 nM | 23500 nM|40000 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | 5100 nM | | | BindingDB |
| Rhodesain | Trypanosoma brucei rhodesiense | Q95PM0 | | = 7750.0 nM | | | NPASS |
| SGC-7901 | Homo sapiens | | | = 26200.0 nM|> 20000.0 nM|= 22500.0 nM | | | NPASS |
| SH-SY5Y | Homo sapiens | | = 5290.0 nM | = 16100.0 nM | | | NPASS |
| SK-BR-3 | Homo sapiens | | | = 42830.0 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 36000.0 nM | | | NPASS |
| T98G | Homo sapiens | | | = 10000.0 nM|= 25000.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 43630.0 nM|= 6700.0 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 14000.0 nM|> 50000.0 nM | | | NPASS |
| Sarcoplasmic/endoplasmic reticulum calcium ATP-ase | Oryctolagus cuniculus | P04191 | | = 3000.0 nM | | = 5800.0 nM | NPASS |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus | P04191 | | 3000 nM | | 5800 nM | BindingDB |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Homo sapiens | P16615 | | 7000 nM|= 7000.0 nM | | 53000 nM|= 53000.0 nM | BindingDB, NPASS |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 | Homo sapiens | Q93084 | | 7000 nM|= 7000.0 nM | | 8600 nM|= 8600.0 nM | BindingDB, NPASS |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens | Q13153 | | 16000 nM|= 16000.0 nM | | | BindingDB, NPASS |
| Sortase | Streptococcus mutans | | | 10200 nM | | | BindingDB |
| Sortase A | Staphylococcus aureus | Q9S446 | | = 37500.0 nM | | | NPASS |
| Sortase A | Streptococcus mutans | Q8CM62 | | = 10200.0 nM | | | NPASS |
| Sortase family protein | Staphylococcus aureus | | | 37500 nM | | | BindingDB |
| SMMC-7721 | Homo sapiens | | | = 19470.0 nM|= 16680.0 nM|= 12570.0 nM|= 18800.0 nM | | | NPASS |
| Histone deacetylase | Homo sapiens | Q969S8 | | = 187000.0 nM | | | NPASS |
| Amyloid-beta A4 protein | Homo sapiens | P05067 | | = 24400.0 nM|= 8270.0 nM|= 5400.0 nM|> 20000.0 nM|= 3850.0 nM|= 900.0 nM|= 1000.0 nM|= 107.0 nM | | | NPASS |
| Histone acetyltransferase p300 | Homo sapiens | Q09472 | | 6500 nM|25000 nM|= 6500.0 nM|= 25000.0 nM | | | BindingDB, NPASS |
| BT-549 | Homo sapiens | | | = 24930.0 nM | | | NPASS |
| BV-2 | Mus musculus | | | = 520.0 nM|= 1420.0 nM|= 4770.0 nM|= 2360.0 nM|= 4500.0 nM|= 6000.0 nM|= 4000.0 nM|= 3000.0 nM|= 8600.0 nM|= 2690.0 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 29000.0 nM|= 18250.0 nM | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 6.496 ug.mL-1 | | | NPASS |
| Beta Lactamase | Pseudomonas aeruginosa | Q932Y6 | | = 7751.0 nM | | | NPASS |
| Beta amyloid A4 protein | Homo sapiens | P05067 | | = 11300.0 nM|= 3100.0 nM|= 1500.0 nM|= 21810.0 nM | | | NPASS |
| Beta-secretase 1 | Homo sapiens | P56817 | | 343000 nM|= 343000.0 nM | | | BindingDB, NPASS |
| Bile acid transporter | Homo sapiens | Q14973 | | | = 64300.0 nM | | NPASS |
| Bone marrow cell | | | | = 7500.0 nM | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 1630 nM | | | BindingDB |
| Butyrylcholinesterase | Homo sapiens | P06276 | | > 5000.0 nM | | | NPASS |
| CCD-841CoN | Homo sapiens | | | = 105110.0 nM | | | NPASS |
| CDGSH iron-sulfur domain-containing protein 1 | Homo sapiens | Q9NZ45 | | 2360 nM|= 2360.0 nM | | 101 nM|= 101.0 nM | BindingDB, NPASS |
| CHO | Cricetulus griseus | | | = 29081.0 nM | | | NPASS |
| CHO-K1 | Cricetulus griseus | | | = 21300.0 nM | | | NPASS |
| COLO 201 | Homo sapiens | | | = 18000.0 nM | | | NPASS |
| CREB-binding protein | Homo sapiens | Q92793 | | 25000 nM|= 25000.0 nM | | | BindingDB, NPASS |
| CREB-binding protein/Histone acetyltransferase p300 | Homo sapiens | Q09472|Q92793 | | 25000 nM | | | BindingDB |
| CREB-binding protein/Histone acetyltransferase p300 | Homo sapiens | | | = 25000.0 nM | | | NPASS |
| CT26 | Mus musculus | | | = 7700.0 nM|> 20000.0 nM | | | NPASS |
| Caco-2 | Homo sapiens | | | = 28000.0 nM|= 47600.0 nM | | | NPASS |
| BT-474 | Homo sapiens | | | = 30140.0 nM|= 11000.0 nM | | | NPASS |
| BGC-823 | Homo sapiens | | | = 6.806 ug.mL-1|= 19500.0 nM|> 20000.0 nM|= 17500.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 30000.0 nM | | | NPASS |
| Amyloid-beta precursor protein | Homo sapiens | P05067 | | 11300 nM|3100 nM|1500 nM|21810 nM|22510 nM|14990 nM|18730 nM|3400 nM|9000 nM|800 nM|10000 nM|6385 nM|16250 nM|3850 nM|8270 nM | | | BindingDB |
| Histone deacetylase | Homo sapiens | O15379|P56524|Q13547|Q8WUI4|Q92769|Q969S8|Q96DB2|Q9BY41|Q9UBN7|Q9UKV0|Q9UQL6 | | 187000 nM | | | BindingDB |
| 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens | P28845 | | = 2295.0 nM | | | NPASS |
| 11-beta-hydroxysteroid dehydrogenase 1 | Rattus norvegicus | P16232 | | = 5785.0 nM | | | NPASS |
| 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens | P80365 | | = 14560.0 nM | | | NPASS |
| 17-beta-hydroxysteroid dehydrogenase type 2 | Homo sapiens | P37059 | | 1730 nM | | | BindingDB |
| 4T1 | Mus musculus | | | = 49400.0 nM | | | NPASS |
| 60 kDa chaperonin | Escherichia coli (strain K12) | P0A6F5 | | > 250000.0 nM | | | NPASS |
| A-431 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 6.52 ug.mL-1 | | | NPASS |
| A549 | Homo sapiens | | | = 17300.0 nM|= 60200.0 nM|= 23540.0 nM|= 27800.0 nM|= 6.521 ug.mL-1|= 6800.0 nM|= 18000.0 nM|> 10000.0 nM|= 43900.0 nM|= 23000.0 nM|= 17900.0 nM|= 28000.0 nM|= 25330.0 nM|= 52300.0 nM|= 38120.0 nM|= 24180.0 nM|= 44750.0 nM|= 32500.0 nM | | | NPASS |
| Casein kinase I epsilon | Homo sapiens | P49674 | | > 10000.0 nM | | | NPASS |
| A549/CDDP | Homo sapiens | | | = 32390.0 nM | | | NPASS |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 1630.0 nM | | | NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | 132130 nM|= 132130.0 nM | | | BindingDB, NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | >5000 nM|> 5000.0 nM | | | BindingDB, NPASS |
| Alkaline phosphatase placental-like | Homo sapiens | P10696 | | > 100000.0 nM | | | NPASS |
| Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | P05186 | | > 100000.0 nM | | | NPASS |
| Alpha-glucosidase | Saccharomyces cerevisiae S288c | P53341|P38158|P07265 | | = 44800.0 nM | | | NPASS |
| Alpha-synuclein | Homo sapiens | P37840 | | 220 nM|161800 nM|= 220.0 nM|= 161800.0 nM|= 3300.0 nM | 500 nM|2000 nM|5000 nM|6500 nM|= 500.0 nM|= 2000.0 nM|= 5000.0 nM|= 6500.0 nM | | BindingDB, NPASS |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | 5020 nM | | 710 nM | BindingDB |
| Amine oxidase [flavin-containing] B | Homo sapiens | P27338 | | 2560 nM | | 21500 nM | BindingDB |
| Aminopeptidase N | Homo sapiens | P15144 | | 15500 nM|= 15500.0 nM | | | BindingDB, NPASS |
| AGS | Homo sapiens | | | = 9770.0 nM|= 20760.0 nM | | | NPASS |
| Chaperonin GroEL | Escherichia coli | | | >250000 nM | | | BindingDB |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens | P10809 | | 8300 nM | | | BindingDB |
| Cholinesterase | Homo sapiens | P06276 | | >5000 nM | | | BindingDB |
| HepG2 | Homo sapiens | | | = 50000.0 nM|= 4430.0 nM|= 52300.0 nM|= 10000.0 nM|= 13780.0 nM|= 16010.0 nM|= 17370.0 nM|= 20300.0 nM|= 9440.0 nM|= 36770.0 nM|= 22750.0 nM|= 17300.0 nM|= 27230.0 nM | | | NPASS |
| Glycogen synthase kinase-3 beta | Homo sapiens | P49841 | | 17950 nM|= 17950.0 nM|> 10000.0 nM | > 10000.0 nM | | BindingDB, NPASS |
| Glycogen synthase kinase-3 beta | Rattus norvegicus | P18266 | | 66 nM|= 66.0 nM | | | BindingDB, NPASS |
| Glyoxalase I | Homo sapiens | Q04760 | | | | = 5.0 nM | NPASS |
| GroEL/GroES | Escherichia coli | | | = 2900.0 nM|= 3100.0 nM | | | NPASS |
| H9c2 | Rattus norvegicus | | | > 79000.0 nM | | | NPASS |
| Cholinesterase | Equus caballus | P81908 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| HCT-8 | Homo sapiens | | | = 6.278 ug.mL-1 | | | NPASS |
| HEK-293T | Homo sapiens | | | > 400000.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | > 400000.0 nM|= 94100.0 nM | | | NPASS |
| Glutathione-S-transferase | Schistosoma japonicum | Q26513 | | > 20000.0 nM | | | NPASS |
| HEp-2 | Homo sapiens | | | = 21370.0 nM | | | NPASS |
| HSC-2 | Homo sapiens | | | = 7800.0 nM|= 3100.0 nM | | | NPASS |
| HSC-3 | Homo sapiens | | | = 11000.0 nM | | | NPASS |
| HSC-4 | Homo sapiens | | | = 7100.0 nM | | | NPASS |
| HSP60/HSP10 | Homo sapiens | | | = 8300.0 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | = 13100.0 nM|= 10000.0 nM|= 21920.0 nM | | | NPASS |
| HT-22 | Mus musculus | | | = 52400.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 14000.0 nM|= 20730.0 nM|= 132370.0 nM|= 23400.0 nM|= 18740.0 nM | | | NPASS |
| HaCaT | Homo sapiens | | | = 13000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 21800.0 nM|= 12110.0 nM|= 51870.0 nM|= 25410.0 nM|= 31890.0 nM|= 8200.0 nM|= 4330.0 nM|= 14030.0 nM|= 5390.0 nM|= 3570.0 nM|= 3560.0 nM|= 32400.0 nM | | | NPASS |
| Hep 3B2 | Homo sapiens | | | = 10000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 6300.0 nM | | | NPASS |
| Glutathione S-transferase P | Human | P09211 | | 6.9e+4 nM | | | BindingDB |
| HCT-116 | Homo sapiens | | | = 13770.0 nM|= 10910.0 nM|= 50000.0 nM|>= 5510.0 nM|= 10500.0 nM|= 3830.0 nM|= 2670.0 nM|= 2400.0 nM|= 10000.0 nM|= 34700.0 nM | | | NPASS |
| GES1 | Homo sapiens | | | = 29100.0 nM | | | NPASS |
| Co-chaperonin GroES | Escherichia coli | | | 2900 nM|3100 nM | | | BindingDB |
| Coagulation factor III | Homo sapiens | P13726 | | = 13.16 nM | | | NPASS |
| Colon 26 | Mus musculus | | | = 30340.0 nM | | | NPASS |
| Glutathione S-transferase Mu 2 | Homo sapiens | P28161 | | = 1810.0 nM | | | NPASS |
| Cyclooxygenase | Bos taurus | O62698 | | = 2000.0 nM | | | NPASS |
| Cysteine protease | Trypanosoma brucei rhodesiense | | | 7750 nM | | | BindingDB |
| D-amino-acid oxidase | Sus scrofa | P00371 | | = 1070.0 nM | | | NPASS |
| DLD-1 | Homo sapiens | | | > 40000.0 nM|= 145500.0 nM|= 10000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 28410.0 nM|= 26230.0 nM|= 33150.0 nM|= 2000.0 nM|= 33120.0 nM|= 31700.0 nM|= 41000.0 nM | | | NPASS |
| Dengue virus 2 | Dengue virus 2 | | | = 11510.0 nM | | | NPASS |
| Dual specificity protein kinase CLK1 | Homo sapiens | P49759 | | = 4921.0 nM|> 10000.0 nM | > 1000.0 nM | | NPASS |
| Cyclin-dependent kinase 5/CDK5 activator 1 | Homo sapiens | Q00535|Q15078 | | > 10000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK3 | Homo sapiens | P49761 | | > 10000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK4 | Homo sapiens | Q9HAZ1 | | = 9749.0 nM | | | NPASS |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens | Q9Y463 | | > 10000.0 nM|= 147.7 nM | | | NPASS |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 | Homo sapiens | Q9NR20 | | > 10000.0 nM | | | NPASS |
| Dual-specificity tyrosine-phosphorylation regulated kinase 1A | Homo sapiens | Q13627 | | > 10000.0 nM|= 300.0 nM | > 1000.0 nM | | NPASS |
| Dual-specificity tyrosine-phosphorylation regulated kinase 2 | Homo sapiens | Q92630 | | = 1058.0 nM|= 2.5 nM|= 5.0 nM | | | NPASS |
| Dual-specificity tyrosine-phosphorylation regulated kinase 3 | Homo sapiens | O43781 | | = 4264.0 nM | | | NPASS |
| EA.hy 926 | Homo sapiens | | | = 20000.0 nM | | | NPASS |
| Epidermal growth factor receptor | Homo sapiens | P00533 | | 8650 nM | | | BindingDB |
| Estradiol 17-beta-dehydrogenase 2 | Homo sapiens | P37059 | | = 1730.0 nM | | | NPASS |
| Dual specificity protein kinase CLK2 | Homo sapiens | P49760 | | > 10000.0 nM | | | NPASS |