IMPPAT Phytochemical information: 
Scutellarein

Scutellarein
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Pyruvate kinase PKMHomo sapiensP14618100000 nM|12500 nMBindingDB
Pyruvate kinase isozymes M1/M2Homo sapiensP14618= 100000.0 nM|= 12500.0 nMNPASS
RBL-2H3Rattus norvegicus= 67200.0 nMNPASS
Radical scavenging activity= 20020.0 nM= 24040.0 nMNPASS
Receptor-type tyrosine-protein kinase FLT3Homo sapiensP36888>10000 nMBindingDB
Receptor-type tyrosine-protein phosphatase SHomo sapiensQ13332600 nM|= 600.0 nMBindingDB, NPASS
Replicase polyprotein 1ab2019-nCoVP0DTD13020 nMBindingDB
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2P0DTD196250 nM|= 5800.0 nMBindingDB, NPASS
Salivary alpha-amylaseHomo sapiensP04745= 9640.0 nMNPASS
Sialidase 2Homo sapiensQ9Y3R4= 55000.0 nMNPASS
Solute carrier organic anion transporter family member 2B1Homo sapiensO94956= 350.0 nM|= 346.74 nMNPASS
Succinate semialdehyde dehydrogenaseHomo sapiensP51649= 7200000.0 nMNPASS
Succinate-semialdehyde dehydrogenase, mitochondrialHomo sapiensP516497200000 nMBindingDB
Tyrosine-protein kinase receptor FLT3Homo sapiensP36888> 10000.0 nMNPASS
UDP-glucuronosyltransferase 1-1Homo sapiensP22309= 41300.0 nMNPASS
UDP-glucuronosyltransferase 1A1Homo sapiensP2230941300 nMBindingDB
Xanthine dehydrogenase/oxidaseBos taurusP8045712600 nMBindingDB
Sialidase-2Homo sapiensQ9Y3R455000 nMBindingDB
Peroxisome proliferator-activated receptor gammaMus musculusP3723816400 nM|= 16400.0 nMBindingDB, NPASS
Xanthine dehydrogenaseBos taurusP80457= 12600.0 nMNPASS
NeuraminidaseInflueA virus (A/Puerto Rico/8/1934(H1N1))P03468= 14.48 ug.mL-1NPASS
AcetylcholinesteraseRattus norvegicusP37136>1.00e+5 nM|>500000 nM|> 500000.0 nMBindingDB, NPASS
Alpha-amylase 1AHomo sapiensP0DUB69640 nMBindingDB
Aurora kinase BHomo sapiensQ96GD43.85e+3 nMBindingDB
Carboxylic ester hydrolaseRattus norvegicus>1.00e+5 nMBindingDB
Cytochrome P450 1A1Homo sapiensP047981640 nM|= 1640.0 nMBindingDB, NPASS
Cytochrome P450 1B1Homo sapiensQ16678220 nM|= 220.0 nMBindingDB, NPASS
Fructose-1,6-bisphosphataseHomo sapiensP09467= 38200.0 nMNPASS
Fructose-1,6-bisphosphatase 1Homo sapiensP0946738200 nMBindingDB
G protein-coupled receptor kinase 6Homo sapiensP432506610 nM|= 6610.0 nMBindingDB, NPASS
NeuraminidaseInflueA virus (strain A/Puerto Rico/8/1934 H1N1)P0346850500 nM|48900 nMBindingDB
Histone-lysine N-methyltransferase 2AHomo sapiensQ031642920 nMBindingDB
Histone-lysine N-methyltransferase EZH1Homo sapiensQ928008770 nM|= 8770.0 nMBindingDB, NPASS
Histone-lysine N-methyltransferase MLLHomo sapiensQ03164= 2920.0 nMNPASS
Histone-lysine N-methyltransferase NSD2Homo sapiensO960282650 nM|= 2650.0 nMBindingDB, NPASS
Histone-lysine N-methyltransferase SETD7Homo sapiensQ8WTS61960 nM|= 1960.0 nMBindingDB, NPASS
Histone-lysine N-methyltransferase SMYD3Homo sapiensQ9H7B418230 nM|= 18230.0 nMBindingDB, NPASS
MV4-11Homo sapiens= 27070.0 nMNPASS
NON-PROTEIN TARGET= 500000000.0 nM|= 13370.0 nMNPASS
GABA-A receptor; anion channelHomo sapiensQ16445= 12022.64 nMNPASS