| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Matrix metalloproteinase 9 | Homo sapiens | P14780 | | | | = 4770.0 nM | NPASS |
| Matrix metalloproteinase-2 | Homo sapiens | P08253 | | | | = 10400.0 nM | NPASS |
| Mus musculus | Mus musculus | | | = 23000.0 nM | | | NPASS |
| Myosin light chain kinase, smooth muscle | Homo sapiens | Q15746 | | 12000 nM|= 12000.0 nM | | | BindingDB, NPASS |
| NCI-H522 | Homo sapiens | | = 17000.0 nM|= 23000.0 nM|= 53000.0 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | | = 1800.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 10000.0 nM|= 12589.25 nM | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 1100 nM|240 nM | | | BindingDB |
| Serine/threonine-protein kinase 33 | Homo sapiens | Q9BYT3 | 12790 nM | | | | BindingDB |
| Replicase polyprotein 1ab | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | K9N7C7 | | > 10000.0 nM | | | NPASS |
| Matrix metalloproteinase 8 | Homo sapiens | P22894 | | | | = 8710.0 nM | NPASS |
| Streptococcus mutans | Streptococcus mutans | | | = 52000.0 nM | | | NPASS |
| Transthyretin | Homo sapiens | P02766 | | | = 2100.0 nM|= 1500.0 nM | = 5400.0 nM | NPASS |
| Tyrosine-protein kinase LCK | Homo sapiens | P06239 | | = 5000.0 nM|= 66000.0 nM|= 20.0 ug.mL-1|= 82000.0 nM | | | NPASS |
| Tyrosine-protein kinase Lck | Homo sapiens | P06239 | | 66000 nM|5000 nM|81800 nM|82000 nM | | | BindingDB |
| Tyrosine-protein kinase SYK | Homo sapiens | P43405 | 25000 nM|5000 nM|= 25000.0 nM|= 5000.0 nM | 38000 nM|10000 nM|= 5.0 ug.mL-1|= 10000.0 nM|= 38000.0 nM | | | BindingDB, NPASS |
| mRNA interferase MazF | Escherichia coli K-12 | P0AE70 | > 99000.0 nM | | | | NPASS |
| Radical scavenging activity | | | | = 28000.0 nM | | | NPASS |
| Matrix metalloproteinase 12 | Homo sapiens | P39900 | | | | = 5570.0 nM | NPASS |
| Lactoylglutathione lyase | Homo sapiens | Q04760 | | 760 nM | | | BindingDB |
| BV-2 | Mus musculus | | | = 80510.0 nM | | | NPASS |
| ADAMTS4 | Homo sapiens | O75173 | | | | = 2680.0 nM | NPASS |
| ADAMTS5 | Homo sapiens | Q9UNA0 | | | | = 1180.0 nM | NPASS |
| ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 | Homo sapiens | P28907 | | >100000 nM | | | BindingDB |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 1100.0 nM|= 240.0 nM|= 390.0 nM | | | NPASS |
| Arginase-1 | Bos taurus | Q2KJ64 | | 47000 nM|= 47000.0 nM | | 136000 nM|= 136000.0 nM | BindingDB, NPASS |
| Arginase-1 | Homo sapiens | P05089 | | 69000 nM|1176000 nM|= 69000.0 nM|= 1176000.0 nM | | | BindingDB, NPASS |
| Lymphocyte differentiation antigen CD38 | Homo sapiens | P28907 | | > 100000.0 nM | | | NPASS |
| Biofilm regulatory protein A | Streptococcus mutans serotype c (strain ATCC 700610 / UA159) | Q8DVR0 | | 52000 nM | | | BindingDB |
| Calcium dependent protein kinase | Triticum aestivum | | | 19000 nM | | | BindingDB |
| Calcium dependent protein kinase | Triticum aestivum | A0T123 | | = 19000.0 nM | | | NPASS |
| Diplodia seriata | Diplodia seriata | | | = 299000.0 nM | | | NPASS |
| Endoribonuclease toxin MazF | Escherichia coli (strain K12) | P0AE70 | >99000 nM | | | | BindingDB |
| Glyoxalase I | Homo sapiens | Q04760 | | = 760.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 5000.0 nM | | | NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 894.7 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 21400.0 nM | | | | NPASS |
| J774 | Mus musculus | | | = 2600.0 nM|= 13000.0 nM|= 4000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 41000.0 nM | | | NPASS |