| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Sodium-dependent noradrenaline transporter | Homo sapiens | P23975 | | | | >10000 nM | BindingDB |
| D(2) dopamine receptor | Homo sapiens | P14416 | | | | 858 nM | BindingDB |
| D(3) dopamine receptor | Homo sapiens | P35462 | | | | 309 nM | BindingDB |
| D(4) dopamine receptor | Homo sapiens | P21917 | | | | 262 nM | BindingDB |
| Delta-type opioid receptor | Homo sapiens | P41143 | | | | >10000 nM | BindingDB |
| Histamine H1 receptor | Homo sapiens | P35367 | | | | >10000 nM | BindingDB |
| Histamine H2 receptor | Homo sapiens | P25021 | | | | 672 nM | BindingDB |
| Sodium-dependent serotonin transporter | Homo sapiens | P31645 | | | | 244 nM | BindingDB |
| D(1B) dopamine receptor | Homo sapiens | P21918 | | | | 2397 nM | BindingDB |
| Histamine H3 receptor | Homo sapiens | Q9Y5N1 | | | | >10000 nM | BindingDB |
| Kappa-type opioid receptor | Homo sapiens | P41145 | | | | >10000 nM | BindingDB |
| Mu-type opioid receptor | Homo sapiens | P35372 | | | | 7265 nM | BindingDB |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | | | | >10000 nM | BindingDB |
| Sodium-dependent dopamine transporter | Homo sapiens | Q01959 | | | | >10000 nM | BindingDB |
| Histamine H4 receptor | Homo sapiens | Q9H3N8 | | | | >10000 nM | BindingDB |
| D(1A) dopamine receptor | Homo sapiens | P21728 | | | | 895 nM | BindingDB |
| Alpha-1A adrenergic receptor | Homo sapiens | P35348 | | | | 430 nM|2 nM | BindingDB |
| Beta-2 adrenergic receptor | Homo sapiens | P07550 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Homo sapiens | P28222 | | | | 100 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Homo sapiens | P28221 | | | | 49 nM | BindingDB |
| 5-hydroxytryptamine receptor 1E | Homo sapiens | P28566 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Homo sapiens | P28223 | | | | 832 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Homo sapiens | P41595 | | | | 543 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Homo sapiens | P28335 | | | | 1069 nM | BindingDB |
| Beta-3 adrenergic receptor | Homo sapiens | P13945 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Homo sapiens | P47898 | | | | 2224 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Homo sapiens | P46098 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | | | | 67 nM | BindingDB |
| Alpha-1B adrenergic receptor | Homo sapiens | P35368 | | | | 1191 nM | BindingDB |
| Alpha-1D adrenergic receptor | Homo sapiens | P25100 | | | | 340 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 1288 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 252 nM | BindingDB |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 181 nM | BindingDB |
| Beta-1 adrenergic receptor | Homo sapiens | P08588 | | | | 8565 nM | BindingDB |
| 5-hydroxytryptamine receptor 6 | Homo sapiens | P50406 | | | | 257 nM | BindingDB |