| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Sodium-dependent serotonin transporter | Rattus norvegicus | P31652 | | >10000 nM | | | BindingDB |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus | P22002 | | | | 40 nM | BindingDB |
| Cholinesterase | Homo sapiens | P06276 | | 13680 nM | | | BindingDB |
| Cholinesterase | Equus caballus | P81908 | | 8380 nM | | | BindingDB |
| Alpha-2C adrenergic receptor | Rattus norvegicus | P22086 | | | | 12 nM | BindingDB |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | 16 nM | | 1 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 4.7 nM | BindingDB |
| Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor | Rattus norvegicus | P19328|P22086|P22909 | | 165 nM | | 4.0 nM|4 nM|149 nM|7.1 nM|81 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 4.6 nM | BindingDB |
| Alpha-2A adrenergic receptor | Cavia porcellus | Q60474 | | | | 5 nM|8 nM | BindingDB |
| Alpha-2B adrenergic receptor | Canis lupus familiaris | | | | | 1 nM | BindingDB |
| Alpha-1D adrenergic receptor | Rattus norvegicus | P23944 | | | | 35 nM | BindingDB |
| Alpha-1D adrenergic receptor | Homo sapiens | P25100 | | | | 3.5 nM|1320 nM | BindingDB |
| Alpha-1B adrenergic receptor | Homo sapiens | P35368 | | | | 4.6 nM|0.6 nM|2270 nM | BindingDB |
| Adenosine receptor A2b | Rattus norvegicus | P29276 | | | 14 nM|13.8 nM | | BindingDB |
| Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor | Rattus norvegicus | P15823|P23944|P43140 | | 6300 nM | | 316 nM | BindingDB |
| Alpha-1A adrenergic receptor | Rattus norvegicus | P43140 | | | | 537 nM|50 nM | BindingDB |
| Alpha-1A adrenergic receptor | Oryctolagus cuniculus | O02824 | | | | 1800 nM|4000 nM|1300 nM | BindingDB |
| Alpha-1A adrenergic receptor | Homo sapiens | P35348 | | | | 4400 nM | BindingDB |
| Alpha-1A adrenergic receptor | Canis lupus familiaris | O77621 | | | | 234 nM | BindingDB |
| Alpha-2A adrenergic receptor | Bos taurus | Q28838 | | | | 18 nM|3.4 nM | BindingDB |
| Alpha-1A adrenergic receptor | Bos taurus | P18130 | | | | 940 nM | BindingDB |