| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NCI-H2347 | Homo sapiens | | | = 135.12 nM | | | NPASS |
| NCI-H226 | Homo sapiens | | | = 13.81 nM | | | NPASS |
| NCI-H2291 | Homo sapiens | | | = 232.1 nM | | | NPASS |
| NCI-H23 | Homo sapiens | | | = 5.706 nM | | | NPASS |
| NCI-H2342 | Homo sapiens | | | = 950.45 nM | | | NPASS |
| NCI-H2228 | Homo sapiens | | | = 41.09 nM | | | NPASS |
| NCI-H2405 | Homo sapiens | | | = 826.38 nM | | | NPASS |
| NCI-H1648 | Homo sapiens | | | = 5.519 nM | | | NPASS |
| NCI-H28 | Homo sapiens | | | = 34.26 nM | | | NPASS |
| NCI-H292 | | | | = 3.03 nM | | | NPASS |
| NCI-H358 | Homo sapiens | | | = 37.01 nM | | | NPASS |
| NCI-H441 | Homo sapiens | | | = 473.3 nM | | | NPASS |
| NCI-H446 | Homo sapiens | | | = 2.122 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 3.4 nM|= 46.39 nM | | | NPASS |
| NCI-H510A | Homo sapiens | | | = 2.753 nM | | | NPASS |
| NCI-H2170 | Homo sapiens | | | = 33.41 nM | | | NPASS |
| NCI-H2452 | Homo sapiens | | | = 9.587 nM | | | NPASS |
| NCI-H2126 | Homo sapiens | | | = 25.9 nM | | | NPASS |
| NCI-H1666 | Homo sapiens | | | = 20.12 nM | | | NPASS |
| NCI-H209 | Homo sapiens | | | = 13.15 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 126.77 nM | | | NPASS |
| NCI-H1651 | Homo sapiens | | | = 23.0 nM | | | NPASS |
| NCI-H520 | | | | = 30.13 nM|= 4.5 nM | | | NPASS |
| NCI-H1693 | Homo sapiens | | | = 78.21 nM | | | NPASS |
| NCI-H1703 | Homo sapiens | | | = 1.431 nM | | | NPASS |
| NCI-H1755 | Homo sapiens | | | = 19.36 nM | | | NPASS |
| NCI-H1770 | Homo sapiens | | | = 28.46 nM | | | NPASS |
| NCI-H1792 | Homo sapiens | | | = 4.391 nM | | | NPASS |
| NCI-H1793 | Homo sapiens | | | = 29.6 nM | | | NPASS |
| NCI-H1838 | Homo sapiens | | | = 191.13 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 24.23 nM | | | NPASS |
| NCI-H1993 | Homo sapiens | | | = 3395.38 nM | | | NPASS |
| NCI-H2009 | Homo sapiens | | | = 53.45 nM | | | NPASS |
| NCI-H2029 | Homo sapiens | | | = 203.7 nM | | | NPASS |
| NCI-H2030 | Homo sapiens | | | = 27.72 nM | | | NPASS |
| NCI-H2052 | Homo sapiens | | | = 24.65 nM | | | NPASS |
| NCI-H2087 | Homo sapiens | | | = 30.53 nM | | | NPASS |
| NCI-H2122 | Homo sapiens | | | = 3.436 nM | | | NPASS |
| NCI-H526 | Homo sapiens | | | = 5.136 nM | | | NPASS |
| NOMO-1 | Homo sapiens | | | = 7.859 nM | | | NPASS |
| NCI-H630 | Homo sapiens | | | = 241.69 nM | | | NPASS |
| Nuclear receptor subfamily 0 group B member 1 | Homo sapiens | P51843 | | >67541 nM | | | BindingDB |
| OAW-28 | Homo sapiens | | | = 40.72 nM | | | NPASS |
| OAW-42 | Homo sapiens | | | = 233.12 nM | | | NPASS |
| OC-314 | Homo sapiens | | | = 2.225 nM | | | NPASS |
| OCI-AML2 | Homo sapiens | | | = 138.49 nM | | | NPASS |
| OCUB-M | Homo sapiens | | | = 7.561 nM | | | NPASS |
| OE19 | Homo sapiens | | | = 412.2 nM | | | NPASS |
| NY | Homo sapiens | | | = 5315.23 nM | | | NPASS |
| OE33 | Homo sapiens | | | = 28.59 nM | | | NPASS |
| ONS-76 | Homo sapiens | | | = 3.742 nM | | | NPASS |
| OS-RC-2 | Homo sapiens | | | = 69.84 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 46.86 nM|= 1.82 nM | | | NPASS |
| OVCAR-4 | Homo sapiens | | | = 27.94 nM | | | NPASS |
| OVCAR-5 | Homo sapiens | | | = 13.6 nM | | | NPASS |
| OVCAR-8 | Homo sapiens | | | = 3.9 nM|= 15.0 nM|= 6.554 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | = 14600.0 nM|= 34000.0 nM | = 2000.0 nM|> 50000.0 nM|= 34000.0 nM|= 10000.0 nM|= 10471.29 nM|= 17700.0 nM|= 19900.0 nM|= 29500.0 nM|= 29000.0 nM | = 3000.0 nM | = 100.0 nM|= 1300.0 nM|= 140000.0 nM|= 15000.0 nM|= 2100.0 nM|= 36500.0 nM | NPASS |
| OMC-1 | Homo sapiens | | | = 144.1 nM | | | NPASS |
| NCI-H596 | | | | = 156.07 nM | | | NPASS |
| NUGC-3 | Homo sapiens | | | = 3.455 nM | | | NPASS |
| NOS-1 | Homo sapiens | | | = 40.88 nM | | | NPASS |
| NCI-H650 | Homo sapiens | | | = 27.08 nM | | | NPASS |
| NCI-H661 | Homo sapiens | | | = 8.047 nM | | | NPASS |
| NCI-H69 | Homo sapiens | | | = 1.6 nM|= 525.78 nM | | | NPASS |
| NCI-H720 | Homo sapiens | | | = 6.88 nM | | | NPASS |
| NCI-H727 | Homo sapiens | | | = 175.7 nM | | | NPASS |
| NCI-H747 | Homo sapiens | | | = 81.18 nM | | | NPASS |
| NCI-H810 | Homo sapiens | | | = 68.69 nM | | | NPASS |
| NTERA-2-cl-D1 | Homo sapiens | | | = 5.893 nM | | | NPASS |
| NCI-H82 | Homo sapiens | | | = 1642.17 nM | | | NPASS |
| NCI/ADR-RES | Homo sapiens | | | = 3900.0 ug.mL-1|= 582.0 nM|= 200.0 nM | | | NPASS |
| NEC8 | Homo sapiens | | | = 5.122 nM | | | NPASS |
| NH-12 | Homo sapiens | | | = 26.35 nM | | | NPASS |
| NKM-1 | Homo sapiens | | | = 1.273 nM | | | NPASS |
| NMC-G1 | Homo sapiens | | | = 8.484 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 12.6 nM|= 2037.0 nM|= 162.0 nM|= 8.5 nM|= 13.0 nM|= 28.0 nM | = 18.0 nM|= 246.0 nM|= 0.1 ug.mL-1|= 5.0 nM|= 540.0 nM|= 20.0 nM|= 1.6 nM|= 8.9 nM|> 375.0 nM|= 3.0 nM|= 2818.38 nM|= 0.11 nM|= 1040.0 nM|= 1.38 nM|= 90.0 nM|= 260.0 nM|= 0.4 nM|> 100.0 nM|= 0.63 nM|= 1.24 nM|= 2.28 nM|= 439.73 nM|= 0.0086 ug.mL-1|= 1.8 nM|= 0.099 nM|= 600.0 nM|= 230.0 nM|> 375000.0 nM|= 200.0 nM|= 11.0 nM|= 3.5 nM|= 15.0 nM|= 4.2 nM|= 205.0 nM|= 2.6 ug.mL-1|= 144.0 nM|= 2.0 nM|= 9.0 nM|= 211.0 nM|= 5.2 nM|= 1.0 nM|= 7.9 nM|= 19.6 nM|= 5.1 nM|= 2.9 nM|= 21.0 nM|= 193.0 nM | | | NPASS |
| P-glycoprotein 1 | Mus musculus | P06795 | | = 8000.0 nM | | | NPASS |
| NCI-N87 | Homo sapiens | | | = 5.671 nM | | | NPASS |
| NCI-H1623 | Homo sapiens | | | = 503.24 nM | | | NPASS |
| LXF-289 cell line | | | | = 10.29 nM | | | NPASS |
| NCI-H1573 | Homo sapiens | | | = 30.74 nM | | | NPASS |
| MDA-MB-453 | Homo sapiens | | | = 3.285 nM | | | NPASS |
| ME-180 | Homo sapiens | | | = 4.473 nM | | | NPASS |
| MEG-01 | Homo sapiens | | | = 14.74 nM | | | NPASS |
| MEL-HO | Homo sapiens | | | = 53.86 nM | | | NPASS |
| MEL-JUSO | Homo sapiens | | | = 17.51 nM | | | NPASS |
| MFE-280 | Homo sapiens | | | = 36.08 nM | | | NPASS |
| MFH-ino | Homo sapiens | | | = 588.37 nM | | | NPASS |
| MDA-MB-435 | Homo sapiens | | | = 4.4 nM|= 0.34 nM|= 0.29 nM|= 0.42 nM|= 0.27 nM|= 11.0 nM|= 27.5 nM|= 0.4 nM|= 0.49 nM|= 0.5 nM | | | NPASS |
| MFM-223 | Homo sapiens | | | = 135.5 nM | | | NPASS |
| MHH-ES-1 | Homo sapiens | | | = 5.129 nM | | | NPASS |
| MHH-NB-11 | Homo sapiens | | | = 38.85 nM | | | NPASS |
| MHH-PREB-1 | Homo sapiens | | | = 1.493 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 3.388 nM | | | NPASS |
| MKN-1 | Homo sapiens | | | = 10.1 nM | | | NPASS |
| MKN-28 | Homo sapiens | | | = 2.698 nM | | | NPASS |
| MKN-45 | Homo sapiens | | | = 48.42 nM | | | NPASS |
| MG-63 | Homo sapiens | | | = 14.16 nM | | | NPASS |
| MKN-7 | Homo sapiens | | | = 76.69 nM | | | NPASS |
| MDA-MB-415 | Homo sapiens | | | = 18.55 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 11.0 nM|= 0.12 nM|= 31.0 nM|= 44.59 nM|= 8.78 nM | | | NPASS |
| LS-411N | Homo sapiens | | | = 66.35 nM | | | NPASS |
| LS-513 | Homo sapiens | | | = 56.27 nM | | | NPASS |
| LU-134-A | Homo sapiens | | | = 8.582 nM | | | NPASS |
| LU-135 | Homo sapiens | | | = 35.58 nM | | | NPASS |
| LU-139 | Homo sapiens | | | = 14.08 nM | | | NPASS |
| LU-99A | Homo sapiens | | | = 20.83 nM | | | NPASS |
| P-glycoprotein 3 | Mus musculus | P21447 | | > 50000.0 nM | | | NPASS |
| MDA-MB-361 | Homo sapiens | | | = 1.662 nM | | | NPASS |
| LoVo | Homo sapiens | | | = 6.025 nM | | | NPASS |
| M059J | Homo sapiens | | | = 15.06 nM | | | NPASS |
| M14 | Homo sapiens | | | = 3.191 nM | | | NPASS |
| MC-IXC | Homo sapiens | | | = 2.985 nM | | | NPASS |
| MC116 | Homo sapiens | | | = 7.953 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 3.0 nM | = 0.22 ug.mL-1|= 0.02 ug.mL-1|= 2.8 nM|= 4.6 nM|= 0.79 nM|= 1.08 ug.mL-1|= 1.37 ug.mL-1|= 0.047 ug.mL-1|= 6.1 ug.mL-1|= 1900.0 nM|= 31.6 nM|= 10.9 nM|> 110.0 nM|= 0.7 nM|= 1.02 ug.mL-1|= 1.22 ug.mL-1 | | | NPASS |
| MDA-MB-157 | Homo sapiens | | | = 9.064 nM | | | NPASS |
| MDA-MB-175-VII | Homo sapiens | | | = 267.63 nM | | | NPASS |
| Lu-65 | Homo sapiens | | | = 115.72 nM | | | NPASS |
| ML-2 | Homo sapiens | | | = 8.652 nM | | | NPASS |
| MLMA | Homo sapiens | | | = 4.652 nM | | | NPASS |
| MMAC-SF | Homo sapiens | | | = 15.09 nM | | | NPASS |
| NB14 | Homo sapiens | | | = 4.953 nM | | | NPASS |
| NB17 | Homo sapiens | | | = 21.77 nM | | | NPASS |
| NB5 | Homo sapiens | | | = 15.7 nM | | | NPASS |
| NB6 | Homo sapiens | | | = 80.02 nM | | | NPASS |
| NB69 | Homo sapiens | | | = 5.73 nM | | | NPASS |
| NB7 | Homo sapiens | | | = 195.12 nM | | | NPASS |
| NBsusSR | Homo sapiens | | | = 3.232 nM | | | NPASS |
| NB13 | Homo sapiens | | | = 3.274 nM | | | NPASS |
| NCI-H1048 | Homo sapiens | | | = 10.06 nM | | | NPASS |
| NCI-H1155 | Homo sapiens | | | = 43.74 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | = 73.0 nM|= 82.0 nM | = 16.42 nM | | | NPASS |
| NCI-H1304 | Homo sapiens | | | = 133.77 nM | | | NPASS |
| NCI-H1355 | Homo sapiens | | | = 19.54 nM | | | NPASS |
| NCI-H1395 | Homo sapiens | | | = 4.277 nM | | | NPASS |
| NCI-H1437 | Homo sapiens | | | = 7.76 nM | | | NPASS |
| NCI-H1563 | Homo sapiens | | | = 21.46 nM | | | NPASS |
| NCI-H1092 | Homo sapiens | | | = 223.56 nM | | | NPASS |
| NB12 | Homo sapiens | | | = 61.41 nM | | | NPASS |
| NB10 | Homo sapiens | | | = 7.317 nM | | | NPASS |
| N592 | | | | = 4.0 nM | | | NPASS |
| MN-60 | Homo sapiens | | | = 29.44 nM | | | NPASS |
| MOLT-13 | Homo sapiens | | | = 5.603 nM | | | NPASS |
| MOLT-16 | Homo sapiens | | | = 2.429 nM | | | NPASS |
| MOLT-4 | Homo sapiens | | | = 3.847 nM | | | NPASS |
| MPP-89 | Homo sapiens | | | = 30.28 nM | | | NPASS |
| MRC5 | Homo sapiens | | | = 24.0 nM | | | NPASS |
| MS-1 | Homo sapiens | | | = 30.83 nM | | | NPASS |
| MSTO-211H | Homo sapiens | | | = 12.22 nM | | | NPASS |
| MV4-11 | Homo sapiens | | | = 2.805 nM | | | NPASS |
| MX1 | Homo sapiens | | | = 2.0 nM|= 2.9 nM|= 2.2 nM | | | NPASS |
| MZ1-PC | Homo sapiens | | | = 24.19 nM | | | NPASS |
| MZ2-MEL | Homo sapiens | | | = 60.31 nM | | | NPASS |
| MZ7-mel | Homo sapiens | | | = 11.08 nM | | | NPASS |
| MeWo | Homo sapiens | | | = 9.134 nM | | | NPASS |
| Mo | Homo sapiens | | | = 880.24 nM | | | NPASS |
| Monoamine oxidase B | Bos taurus | P56560 | | | | = 77000.0 nM | NPASS |
| Multidrug resistance-associated protein 1 | Homo sapiens | P33527 | | 30000 nM|= 30000.0 nM | | | BindingDB, NPASS |
| NCI-H1581 | Homo sapiens | | | = 4.236 nM | | | NPASS |
| P12-Ichikawa | Homo sapiens | | | = 1.704 nM | | | NPASS |
| SNU-398 | Homo sapiens | | = 38.0 nM|= 26.0 nM | | | | NPASS |
| P388 | Mus musculus | | | = 1.7 nM|= 8.2 nM|= 4.1 nM|= 0.7 nM|= 27.0 nM|= 0.6 nM | | | NPASS |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens | Q9NPD5 | | 43500 nM|= 43500.0 nM | | 18600 nM|= 18600.0 nM | BindingDB, NPASS |
| Steroidogenic factor 1 | Homo sapiens | Q13285 | | >67541 nM | | | BindingDB |
| T-24 | Homo sapiens | | | = 5.104 nM | | | NPASS |
| T47D | Homo sapiens | | = 25.0 nM|= 43.0 nM|= 32.0 nM | = 7.711 nM|= 5.0 nM | | | NPASS |
| T84 | Homo sapiens | | | = 8147.21 nM | | | NPASS |
| T98G | Homo sapiens | | | = 11.4 nM | | | NPASS |
| TCC-SUP | Homo sapiens | | | = 23.63 nM | | | NPASS |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens | Q9Y6L6 | | 46800 nM|= 46800.0 nM | | 10200 nM|= 10200.0 nM | BindingDB, NPASS |
| TE-1 | Homo sapiens | | | = 10.85 nM | | | NPASS |
| TE-11 | Homo sapiens | | | = 5.128 nM | | | NPASS |
| TE-12 | Homo sapiens | | | = 700.72 nM | | | NPASS |
| TE-5 | Homo sapiens | | | = 6.135 nM | | | NPASS |
| TE-6 | Homo sapiens | | | = 56.47 nM | | | NPASS |
| TE-8 | Homo sapiens | | | = 6.156 nM | | | NPASS |
| TE-9 | Homo sapiens | | | = 4.27 nM | | | NPASS |
| TGBC11TKB | Homo sapiens | | | = 15.83 nM | | | NPASS |
| TE-10 | Homo sapiens | | | = 21.47 nM | | | NPASS |
| TGBC1TKB | Homo sapiens | | | = 31.21 nM | | | NPASS |
| Similar to alpha-tubulin isoform 1 | Bos taurus | | | 600 nM|700 nM | | | BindingDB |
| SW982 | Homo sapiens | | | = 8.919 nM | | | NPASS |
| SW13 | Homo sapiens | | | = 5.49 nM | | | NPASS |
| SW1417 | Homo sapiens | | | = 423.54 nM | | | NPASS |
| SW1463 | Homo sapiens | | | = 69.69 nM | | | NPASS |
| SW1573 | Homo sapiens | | | = 33.25 nM | | | NPASS |
| SW1710 | Homo sapiens | | | = 5.607 nM | | | NPASS |
| SW1783 | Homo sapiens | | | = 85.55 nM | | | NPASS |
| SW1990 | Homo sapiens | | | = 61.39 nM | | | NPASS |
| SiHa | Homo sapiens | | | = 109.77 nM | | | NPASS |
| SW48 | Homo sapiens | | | = 6.943 nM | | | NPASS |
| SW684 | Homo sapiens | | | = 101.3 nM | | | NPASS |
| SW756 | Homo sapiens | | | = 14.7 nM | | | NPASS |
| SW780 | Homo sapiens | | | = 2.329 nM | | | NPASS |
| SW837 | Homo sapiens | | | = 120.44 nM | | | NPASS |
| SW872 | Homo sapiens | | | = 255.22 nM | | | NPASS |
| SW900 | Homo sapiens | | | = 25.41 nM | | | NPASS |
| SW948 | Homo sapiens | | | = 75.99 nM | | | NPASS |
| SW626 | Homo sapiens | | | = 23.21 nM | | | NPASS |
| TGBC24TKB | Homo sapiens | | | = 32.52 nM | | | NPASS |
| TI-73 | Homo sapiens | | | = 3.212 nM | | | NPASS |
| TK-10 | Homo sapiens | | | = 42.4 nM | | | NPASS |
| UMC-11 | Homo sapiens | | | = 76.22 nM | | | NPASS |
| UMUC3 | Homo sapiens | | | = 5.107 nM | | | NPASS |
| UO-31 | Homo sapiens | | | = 13.94 nM | | | NPASS |
| VA-ES-BJ | Homo sapiens | | | = 3.273 nM | | | NPASS |
| VM-CUB-1 | Homo sapiens | | | = 4.281 nM | | | NPASS |
| VMRC-RCZ | Homo sapiens | | | = 19.27 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | < 3700.0 nM | = 27060.0 nM | | | NPASS |
| UACC-893 | Homo sapiens | | | = 98.3 nM | | | NPASS |
| WM-115 | Homo sapiens | | | = 10.16 nM | | | NPASS |
| YAPC | Homo sapiens | | | = 86.99 nM | | | NPASS |
| YH-13 | Homo sapiens | | | = 3.702 nM | | | NPASS |
| YKG-1 | Homo sapiens | | | = 5.534 nM | | | NPASS |
| ZR-75-1 | Homo sapiens | | | = 8.0 nM | | | NPASS |
| ZR-75-30 | Homo sapiens | | | = 402.55 nM | | | NPASS |
| no-10 | Homo sapiens | | | = 270.54 nM | | | NPASS |
| no-11 | Homo sapiens | | | = 38.83 nM | | | NPASS |
| WRL68 | Homo sapiens | | | = 1.45 ug.mL-1|= 2.6 ug.mL-1 | | | NPASS |
| UACC-62 | Homo sapiens | | | = 8.062 nM | | | NPASS |
| UACC-257 | Homo sapiens | | | = 90.53 nM | | | NPASS |
| U2OS | Homo sapiens | | | = 25.72 nM | | | NPASS |
| TYK-nu | Homo sapiens | | | = 11.9 nM | | | NPASS |
| Thromboxane-A synthase | Homo sapiens | P24557 | | = 1870.0 nM | | | NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | | = 410.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 94.0 nM | | | NPASS |
| Tubulin | Bos taurus | Q862F3 | | = 700.0 nM|= 600.0 nM | | | NPASS |
| Tubulin | Homo sapiens | Q9BUF5 | = 200.0 nM | = 70.0 nM|= 300.0 nM|= 2100.0 nM | | | NPASS |
| Tubulin | Sus scrofa | P02550 | | = 600.0 nM|= 1600.0 nM|= 1100.0 nM | | | NPASS |
| Tubulin alpha-1A chain | Pig | P02550 | | 200 nM | | | BindingDB |
| Tubulin beta chain | Bos taurus | Q6B856 | | | | > 100000.0 nM | NPASS |
| Tubulin beta chain | Sus scrofa | P02554 | | 1100 nM|600 nM|130 nM|1600 nM | | | BindingDB |
| Tubulin beta chain [1-43] | Leishmadonovani | P21148 | | 1000 nM | | | BindingDB |
| Tubulin beta-2B chain | Bos taurus | Q6B856 | | | | >100000 nM | BindingDB |
| U-118-MG | Homo sapiens | | | = 45.16 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 8.1 nM|= 5.018 nM | | | NPASS |
| U-266 | Homo sapiens | | | = 10.8 nM | | | NPASS |
| U-87 MG | Homo sapiens | | | = 29.98 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 6880.0 nM|= 0.49 nM | | | NPASS |
| SW1088 | Homo sapiens | | | = 16.97 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 8.836 nM | | | NPASS |
| SW 962 | Homo sapiens | | | = 19.39 nM | | | NPASS |
| SW 954 | Homo sapiens | | | = 9.662 nM | | | NPASS |
| RPMI-2650 | Homo sapiens | | | = 26.61 nM | | | NPASS |
| RPMI-7951 | Homo sapiens | | | = 1.658 nM | | | NPASS |
| RPMI-8226 | Homo sapiens | | | = 28.0 nM|= 2.852 nM | | | NPASS |
| RPMI-8866 | Homo sapiens | | | = 1.966 nM | | | NPASS |
| RS4-11 | Homo sapiens | | | = 4.508 nM | | | NPASS |
| RT-112 | Homo sapiens | | | = 2.708 nM | | | NPASS |
| RVH-421 | Homo sapiens | | | = 7.249 nM | | | NPASS |
| RO82-W-1 | Homo sapiens | | | = 5.57 nM | | | NPASS |
| RXF 393 | Homo sapiens | | | = 1.439 nM | | | NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >246000 nM | | | BindingDB |
| S-117 | Homo sapiens | | | = 5.576 nM | | | NPASS |
| SAOS-2 | Homo sapiens | | | = 32.31 nM | | | NPASS |
| SAS | Homo sapiens | | | = 28.13 nM | | | NPASS |
| SBC-1 | Homo sapiens | | | = 8.104 nM | | | NPASS |
| SBC-5 | Homo sapiens | | | = 7.471 nM | | | NPASS |
| SCC-15 | Homo sapiens | | | = 23.15 nM | | | NPASS |
| Ramos-2G6-4C10 | Homo sapiens | | | = 1.546 nM | | | NPASS |
| RMG-I | Homo sapiens | | | = 116.58 nM | | | NPASS |
| RKO | Homo sapiens | | | = 8.239 nM | | | NPASS |
| RH-18 | Homo sapiens | | | = 1128.93 nM | | | NPASS |
| P388/ADR | Mus musculus | | | = 95.0 nM|= 4.3 nM | | | NPASS |
| PA-1 | Homo sapiens | | | = 0.025 ug.mL-1|= 1.15 ug.mL-1|= 0.15 ug.mL-1|= 0.03 ug.mL-1|= 8.092 nM|= 4.6 nM | | | NPASS |
| PANC-03-27 | Homo sapiens | | | = 5.472 nM | | | NPASS |
| PANC-08-13 | Homo sapiens | | | = 61.47 nM | | | NPASS |
| PC-14 | Homo sapiens | | | = 3.534 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 5.5 nM|= 5.0 nM|= 33.37 nM|= 766.0 nM | | | NPASS |
| PFSK-1 | Homo sapiens | | | = 4.972 nM | | | NPASS |
| PSN1 | Homo sapiens | | | = 1.248 nM | | | NPASS |
| Panc1005 | Homo sapiens | | | = 42.8 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 2.0 nM | | | NPASS |
| Plasmodium yoelii yoelii | Plasmodium yoelii yoelii | | | = 7950.0 nM | | | NPASS |
| QIMR-WIL | Homo sapiens | | | = 8.95 nM | | | NPASS |
| RCC10RGB | Homo sapiens | | | = 510.4 nM | | | NPASS |
| RCM-1 | Homo sapiens | | | = 1369.69 nM | | | NPASS |
| RD | Homo sapiens | | | = 4.172 nM|= 52.5 nM|= 53.0 nM | | | NPASS |
| RERF-LC-MS | Homo sapiens | | | = 15.15 nM | | | NPASS |
| RH-1 | Homo sapiens | | | = 3.4 nM | | | NPASS |
| SCC-25 | Homo sapiens | | | = 15.68 nM | | | NPASS |
| P30-OHK | Homo sapiens | | | = 11.07 nM | | | NPASS |
| SCC-4 | Homo sapiens | | | = 2.395 nM | | | NPASS |
| SCH | Homo sapiens | | | = 29.72 nM | | | NPASS |
| SK-N-FI | Homo sapiens | | | = 642.78 nM | | | NPASS |
| SK-NEP-1 | Homo sapiens | | | = 1.505 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 2.7 nM|= 0.039 nM|= 8155.03 nM | | | NPASS |
| SK-PN-DW | Homo sapiens | | | = 6.138 nM | | | NPASS |
| SK-UT-1 | Homo sapiens | | | = 11.75 nM | | | NPASS |
| SKG-IIIa | Homo sapiens | | | = 17.24 nM | | | NPASS |
| SN12C | Homo sapiens | | | = 16.06 nM | | | NPASS |
| SK-N-DZ | Homo sapiens | | | = 37.37 nM | | | NPASS |
| SNB-75 | Homo sapiens | | | = 11.25 nM | | | NPASS |
| LS-123 | Homo sapiens | | | = 53.33 nM | | | NPASS |
| SNU-423 | Homo sapiens | | | = 19.47 nM | | | NPASS |
| SNU-449 | Homo sapiens | | | = 127.72 nM | | | NPASS |
| SNU-5 | Homo sapiens | | | = 132.84 nM | | | NPASS |
| SNU-C2B | Homo sapiens | | | = 24.67 nM | | | NPASS |
| SNU1 | Homo sapiens | | | = 1.622 nM | | | NPASS |
| SW 1116 | Homo sapiens | | | = 1163.6 nM | | | NPASS |
| SNU-387 | Homo sapiens | | | = 11.42 nM | | | NPASS |
| SK-N-AS | Homo sapiens | | | = 8.669 nM | | | NPASS |
| SK-MES-1 | Homo sapiens | | | = 8.645 nM | | | NPASS |
| SK-MEL3 | Homo sapiens | | | = 717.01 nM | | | NPASS |
| SF-126 | Homo sapiens | | | = 21.9 nM | | | NPASS |
| SF-268 | Homo sapiens | | | = 16.19 nM | | | NPASS |
| SF-295 | Homo sapiens | | | = 36.31 nM | | | NPASS |
| SF-539 | Homo sapiens | | | = 1.211 nM | | | NPASS |
| SH-4 | Homo sapiens | | | = 43.54 nM | | | NPASS |
| SHP77 | Homo sapiens | | | = 148.18 nM | | | NPASS |
| SJRH30 | Homo sapiens | | | = 59.36 nM | | | NPASS |
| SJSA-1 | Homo sapiens | | | = 12.06 nM | | | NPASS |
| SK-BR-3 | Homo sapiens | | | = 72.0 nM|= 0.91 nM | | | NPASS |
| SK-HEP1 | Homo sapiens | | | = 12.05 nM | | | NPASS |
| SK-LMS-1 | Homo sapiens | | | = 58.6 nM | | | NPASS |
| SK-LU-1 | Homo sapiens | | | = 18.71 nM | | | NPASS |
| SK-MEL-1 | Homo sapiens | | | = 67.32 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 53.3 nM | | | NPASS |
| SK-MEL-24 | Homo sapiens | | | = 31.55 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 17.04 nM | | | NPASS |
| SK-MEL-30 | Homo sapiens | | | = 415.46 nM | | | NPASS |
| SCC-9 | Homo sapiens | | | = 10.66 nM | | | NPASS |
| LS-1034 | Homo sapiens | | | = 2844.0 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 4.6 nM | | | NPASS |
| LNCaP-Clone-FGC | Homo sapiens | | | = 8.279 nM | | | NPASS |
| COLO-829 | Homo sapiens | | | = 19.17 nM | | | NPASS |
| COR-L105 | Homo sapiens | | | = 65.75 nM | | | NPASS |
| COR-L23 | Homo sapiens | | | = 3.623 nM | | | NPASS |
| COR-L88 | Homo sapiens | | | = 24.32 nM | | | NPASS |
| CP50-MEL-B | Homo sapiens | | | = 13.12 nM | | | NPASS |
| CP66-MEL | Homo sapiens | | | = 48.58 nM | | | NPASS |
| CTB-1 | Homo sapiens | | | = 1.636 nM | | | NPASS |
| COLO-824 | Homo sapiens | | | = 136.2 nM | | | NPASS |
| CTV-1 | Homo sapiens | | | = 1.405 nM | | | NPASS |
| CWR22R | Homo sapiens | | | = 9.815 nM | | | NPASS |
| Ca-Ski | Homo sapiens | | | = 4.694 nM | | | NPASS |
| Ca9-22 | Homo sapiens | | | = 6.391 nM | | | NPASS |
| CaR-1 | Homo sapiens | | | = 45.73 nM | | | NPASS |
| Caco-2 | Homo sapiens | | | = 2.8 ug.mL-1|= 0.46 ug.mL-1 | | | NPASS |
| Calu-3 | Homo sapiens | | | = 551.0 nM | | | NPASS |
| Calu-6 | Homo sapiens | | | = 149.1 nM | | | NPASS |
| CW-2 | Homo sapiens | | | = 101.38 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens | Q92887 | | = 21000.0 nM | | | NPASS |
| COLO-800 | Homo sapiens | | | = 3.342 nM | | | NPASS |
| COLO-741 | Homo sapiens | | | = 2.139 nM | | | NPASS |
| CEM | Homo sapiens | | | = 2.0 nM|= 1.0 nM | | | NPASS |
| CFPAC-1 | Homo sapiens | | | = 93.2 nM | | | NPASS |
| CGTH-W-1 | Homo sapiens | | | = 5.556 nM | | | NPASS |
| CHL-1 | Homo sapiens | | | = 12.0 nM | | | NPASS |
| CHO | Cricetulus griseus | | | = 17.0 nM | | | NPASS |
| CHO-TAX 5-6 | Cricetulus griseus | | | = 6.9 nM | | | NPASS |
| CHO-VV 3-2 | Cricetulus griseus | | | = 66.0 nM | | | NPASS |
| COLO-792 | Homo sapiens | | | = 25.63 nM | | | NPASS |
| CHP-212 | Homo sapiens | | | = 3.547 nM | | | NPASS |
| COLO 320DM | Homo sapiens | | | = 0.52 ug.mL-1|= 1.6 ug.mL-1 | | | NPASS |
| COLO-320-HSR | Homo sapiens | | | = 203.92 nM | | | NPASS |
| COLO-668 | Homo sapiens | | | = 562.6 nM | | | NPASS |
| COLO-678 | Homo sapiens | | | = 2480.78 nM | | | NPASS |
| COLO-679 | Homo sapiens | | | = 5415.81 nM | | | NPASS |
| COLO-680N | Homo sapiens | | | = 74.71 nM | | | NPASS |
| COLO-684 | Homo sapiens | | | = 7.666 nM | | | NPASS |
| COLO 320 | Homo sapiens | | | = 1.6 ug.mL-1|= 0.52 ug.mL-1 | | | NPASS |
| Capan-2 | Homo sapiens | | | = 114.18 nM | | | NPASS |
| ChaGo-K-1 | Homo sapiens | | | = 1.013 nM | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | 26000 nM|= 26000.0 nM | | | BindingDB, NPASS |
| DU-145 | Homo sapiens | | | = 0.063 nM|= 98.66 nM | | | NPASS |
| DU-4475 | Homo sapiens | | | = 383.01 nM | | | NPASS |
| Daoy | Homo sapiens | | | = 3.102 nM | | | NPASS |
| Detroit562 | Homo sapiens | | | = 5.531 nM | | | NPASS |
| DoTc2-4510 | Homo sapiens | | | = 16.52 nM | | | NPASS |
| EC-GI-10 | Homo sapiens | | | = 3.531 nM | | | NPASS |
| ECC10 | Homo sapiens | | | = 21.16 nM | | | NPASS |
| DSH1 | Homo sapiens | | | = 23.21 nM | | | NPASS |
| EFM-19 | Homo sapiens | | | = 5.242 nM | | | NPASS |
| EFO-27 | Homo sapiens | | | = 7.449 nM | | | NPASS |
| EGI-1 | Homo sapiens | | | = 10.81 nM | | | NPASS |
| EKVX | Homo sapiens | | | = 278.22 nM | | | NPASS |
| EM-2 | Homo sapiens | | | = 5.316 nM | | | NPASS |
| EOL1 | Homo sapiens | | | = 1.261 nM | | | NPASS |
| EPLC-272H | Homo sapiens | | | = 10.78 nM | | | NPASS |
| ES1 | Homo sapiens | | | = 4.714 nM | | | NPASS |
| EFO-21 | Homo sapiens | | | = 44.03 nM | | | NPASS |
| DOK | Homo sapiens | | | = 4.196 nM | | | NPASS |
| DOHH-2 | Homo sapiens | | | = 1.809 nM | | | NPASS |
| DMS-79 | Homo sapiens | | | = 534.65 nM | | | NPASS |
| D-247MG | Homo sapiens | | | = 6.979 nM | | | NPASS |
| D-263MG | Homo sapiens | | | = 9.278 nM | | | NPASS |
| D-336MG | Homo sapiens | | | = 7.255 nM | | | NPASS |
| D-392MG | Homo sapiens | | | = 18.86 nM | | | NPASS |
| D-423MG | Homo sapiens | | | = 8.639 nM | | | NPASS |
| D-502MG | Homo sapiens | | | = 23.49 nM | | | NPASS |
| D-542MG | Homo sapiens | | | = 3876.68 nM | | | NPASS |
| D-566MG | Homo sapiens | | | = 2.043 nM | | | NPASS |
| D283 Med | | | | = 39.1 nM | | | NPASS |
| DB | Homo sapiens | | | = 1.687 nM | | | NPASS |
| DBTRG-05MG | Homo sapiens | | | = 225.99 nM | | | NPASS |
| DEL | Homo sapiens | | | = 2.16 nM | | | NPASS |
| DJM-1 | Homo sapiens | | | = 2816.86 nM | | | NPASS |
| DK-MG | Homo sapiens | | | = 6.646 nM | | | NPASS |
| DLD-1 | Homo sapiens | | = 129.0 nM|= 160.0 nM | | | | NPASS |
| DMS-114 | Homo sapiens | | | = 20.94 nM | | | NPASS |
| DMS-273 | Homo sapiens | | | = 3.396 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | = 0.1 ug.mL-1|= 1.2 nM|= 0.4 nM|= 28.7 nM|= 206.6 nM|= 4.0 nM|= 0.73 nM|= 78.0 nM|= 496.0 nM|= 0.03 ug.mL-1|= 500.0 nM|= 0.7 nM|= 80.0 nM|= 0.38 nM|= 4.1 nM|= 9.4 nM|= 0.8 nM|= 2.0 nM|= 10.05 nM|= 2.9 nM|= 870.0 nM|= 1.3 nM|= 670.0 nM | | | NPASS |
| CAS-1 | Homo sapiens | | | = 93.12 nM | | | NPASS |
| CAPAN-1 | Homo sapiens | | | = 52.3 nM | | | NPASS |
| CAMA-1 | Homo sapiens | | | = 32.01 nM | | | NPASS |
| A498 | Homo sapiens | | | = 5.938 nM | | | NPASS |
| A549 | Homo sapiens | | = 0.9 nM|= 0.5 nM | = 9.9 nM|= 1.1 nM|= 17.0 nM|= 20.0 nM|= 4.954 nM | | | NPASS |
| A673 | Homo sapiens | | | = 6.875 nM | | | NPASS |
| A704 | Homo sapiens | | | = 119.71 nM | | | NPASS |
| ABC-1 | Homo sapiens | | | = 15.49 nM | | | NPASS |
| ACHN | Homo sapiens | | | = 25.0 nM|= 59.04 nM | | | NPASS |
| ACN | Homo sapiens | | | = 40.29 nM | | | NPASS |
| A4-Fuk | Homo sapiens | | | = 1.867 nM | | | NPASS |
| AGS | Homo sapiens | | | = 12.3 nM | | | NPASS |
| AM-38 | Homo sapiens | | | = 36.92 nM | | | NPASS |
| AN3-CA | Homo sapiens | | | = 9.765 nM | | | NPASS |
| ASPC1 | Homo sapiens | | | = 13.21 nM | | | NPASS |
| ATN-1 | Homo sapiens | | | = 1.034 nM | | | NPASS |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | 21000 nM | | | BindingDB |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | 14600 nM|34000 nM | 34000 nM|2000 nM|>50000 nM|29000 nM|29500 nM|17700 nM|19900 nM|10471 nM|10000 nM | 3000 nM | 100 nM|1300 nM|2100 nM|140000 nM|36500 nM|15000 nM | BindingDB |
| ATP-dependent translocase ABCB1 | Mus musculus | P06795 | | 8000 nM | | | BindingDB |
| ALL-PO | Homo sapiens | | | = 5.215 nM | | | NPASS |
| A388 | Homo sapiens | | | = 6.915 nM | | | NPASS |
| A3-KAW | Homo sapiens | | | = 4.32 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 61.66 nM|= 5.0 nM|= 4.608 nM | | | NPASS |
| 23132-87 | Homo sapiens | | | = 20.64 nM | | | NPASS |
| 5637 | Homo sapiens | | | = 0.951 nM | | | NPASS |
| 639-V | Homo sapiens | | | = 5.605 nM | | | NPASS |
| 647-V | Homo sapiens | | | = 23.03 nM | | | NPASS |
| 697 | Homo sapiens | | | = 6.225 nM | | | NPASS |
| 769-P | Homo sapiens | | | = 25.55 nM | | | NPASS |
| 786-0 | Homo sapiens | | | = 4.5 nM|= 0.31 nM|= 15.58 nM | | | NPASS |
| 8-MG-BA | Homo sapiens | | | = 6.335 nM | | | NPASS |
| 8305C | Homo sapiens | | | = 3.67 nM | | | NPASS |
| 8505C | Homo sapiens | | | = 3.109 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 23.53 nM | | | NPASS |
| A-427 | Homo sapiens | | | = 12.55 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 4975.15 nM | | | NPASS |
| A101D | Homo sapiens | | | = 31.39 nM | | | NPASS |
| A172 | Homo sapiens | | | = 9.616 nM | | | NPASS |
| A204 | Homo sapiens | | | = 8.765 nM | | | NPASS |
| A2058 | Homo sapiens | | | = 4.0 nM|= 1.218 nM|= 3.7 nM | | | NPASS |
| ATP-dependent translocase ABCB1 | Mus musculus | P21447 | | >50000 nM | | | BindingDB |
| ES3 | Homo sapiens | | | = 2.766 nM | | | NPASS |
| AU565 | Homo sapiens | | | = 3.448 nM|= 4.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase | Oryctolagus cuniculus | P12530 | | = 5037.0 nM | | | NPASS |
| LOX IMVI | Homo sapiens | | | = 6.977 nM | | | NPASS |
| C2BBe1 | Homo sapiens | | | = 16.88 nM | | | NPASS |
| C32 | Homo sapiens | | | = 866.85 nM | | | NPASS |
| C3A | Homo sapiens | | | = 332.14 nM | | | NPASS |
| C8166 | Homo sapiens | | | = 27.01 nM | | | NPASS |
| CAKI-1 | Homo sapiens | | | = 24.61 nM | | | NPASS |
| CAL-120 | Homo sapiens | | | = 87.26 nM | | | NPASS |
| Bile salt export pump | Homo sapiens | O95342 | | 114700 nM|62000 nM|= 114700.0 nM|= 62000.0 nM | | | BindingDB, NPASS |
| CAL-12T | Homo sapiens | | | = 55.97 nM | | | NPASS |
| CAL-33 | Homo sapiens | | | = 6.184 nM | | | NPASS |
| CAL-39 | Homo sapiens | | | = 5.114 nM | | | NPASS |
| CAL-51 | Homo sapiens | | | = 16.39 nM | | | NPASS |
| CAL-54 | Homo sapiens | | | = 60.59 nM | | | NPASS |
| CAL-62 | Homo sapiens | | | = 10.1 nM | | | NPASS |
| CAL-72 | Homo sapiens | | | = 647.18 nM | | | NPASS |
| CAL-85-1 | Homo sapiens | | | = 6079.95 nM | | | NPASS |
| CAL-27 | Homo sapiens | | | = 2.086 nM | | | NPASS |
| Beta tubulin | Leishmadonovani | Q25270 | | = 1000.0 nM | | | NPASS |
| Becker | Homo sapiens | | | = 1.126 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 8.01 nM | | | NPASS |
| B16 | Mus musculus | | | = 3.6 ug.mL-1 | | | NPASS |
| BALL-1 | Homo sapiens | | | = 313.17 nM | | | NPASS |
| BB30-HNC | Homo sapiens | | | = 8.315 nM | | | NPASS |
| BB49-HNC | Homo sapiens | | | = 12.56 nM | | | NPASS |
| BB65-RCC | Homo sapiens | | | = 20.7 nM | | | NPASS |
| BCPAP | Homo sapiens | | | = 2.33 nM | | | NPASS |
| BE-13 | Homo sapiens | | | = 1.416 nM | | | NPASS |
| BEN | Homo sapiens | | | = 81.23 nM | | | NPASS |
| BFTC-905 | Homo sapiens | | | = 3.773 nM | | | NPASS |
| BFTC-909 | Homo sapiens | | | = 7.532 nM | | | NPASS |
| BHT-101 | Homo sapiens | | | = 31.36 nM | | | NPASS |
| BHY | Homo sapiens | | | = 15.33 nM | | | NPASS |
| BPH-1 | Homo sapiens | | | = 3.263 nM | | | NPASS |
| BT-20 | Homo sapiens | | | = 37.68 nM | | | NPASS |
| BT-474 | Homo sapiens | | | = 94.15 nM | | | NPASS |
| BT-549 | Homo sapiens | | | = 7.977 nM | | | NPASS |
| BV-173 | Homo sapiens | | | = 42.27 nM | | | NPASS |
| Amine oxidase [flavin-containing] B | Bos taurus | P56560 | | | | 77000 nM | BindingDB |
| ES4 | Homo sapiens | | | = 13.83 nM | | | NPASS |
| C-33-A | Homo sapiens | | | = 12.66 nM | | | NPASS |
| ES6 | Homo sapiens | | | = 115.12 nM | | | NPASS |
| JVM-2 | Homo sapiens | | | = 5585.18 nM | | | NPASS |
| JVM-3 | Homo sapiens | | | = 1.705 nM | | | NPASS |
| K5 | Homo sapiens | | | = 4.682 nM | | | NPASS |
| K562 | Homo sapiens | | = 1.0 nM | = 3000.0 nM|= 0.88 nM|= 170.0 nM|= 193000.0 nM|= 0.36 nM|= 1082.28 nM|= 7.0 nM|= 2.7 nM|= 10.0 nM | | | NPASS |
| KALS-1 | Homo sapiens | | | = 7.787 nM | | | NPASS |
| KARPAS-299 | Homo sapiens | | | = 1657.4 nM | | | NPASS |
| KARPAS-45 | Homo sapiens | | | = 1.793 nM | | | NPASS |
| JAR | Homo sapiens | | | = 0.608 nM | | | NPASS |
| KB | Homo sapiens | | | = 0.046 ug.mL-1|= 0.46 ug.mL-1|= 1.0 nM|= 0.8 nM | | | NPASS |
| KE-37 | Homo sapiens | | | = 3.993 nM | | | NPASS |
| KG-1 | | | | = 18.38 nM | | | NPASS |
| KGN | Homo sapiens | | | = 33.33 nM | | | NPASS |
| KINGS-1 | Homo sapiens | | | = 9.324 nM | | | NPASS |
| KLE | Homo sapiens | | | = 309.24 nM | | | NPASS |
| KM-H2 | Homo sapiens | | | = 5.339 nM | | | NPASS |
| KM12 | Homo sapiens | | | = 14.42 nM | | | NPASS |
| KB 3-1 | Homo sapiens | | | = 9271000.0 nM | | | NPASS |
| KMOE-2 | Homo sapiens | | | = 20.76 nM | | | NPASS |
| J82 | Homo sapiens | | | = 68.47 nM | | | NPASS |
| J774 | Mus musculus | | | = 2.1 nM | | | NPASS |
| HuCCT-1 | Homo sapiens | | | = 17.29 nM | | | NPASS |
| HuO-3N1 | Homo sapiens | | | = 4.827 nM | | | NPASS |
| HuO9 | Homo sapiens | | | = 12.64 nM | | | NPASS |
| HuP-T3 | Homo sapiens | | | = 17.96 nM | | | NPASS |
| HuP-T4 | Homo sapiens | | | = 43.18 nM | | | NPASS |
| HuTu80 | Homo sapiens | | | = 12.28 nM | | | NPASS |
| Huh-7 | Homo sapiens | | | = 87.74 nM | | | NPASS |
| J774.2 | | | | = 15.9 nM|= 0.8 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| IGR-1 | Homo sapiens | | | = 2.076 nM | | | NPASS |
| IGROV-1 | Homo sapiens | | | = 215.27 nM | | | NPASS |
| IMR-90 | Homo sapiens | | | > 1000.0 nM | | | NPASS |
| IST-MEL1 | Homo sapiens | | | = 4.526 nM | | | NPASS |
| IST-MES1 | Homo sapiens | | | = 67.68 nM | | | NPASS |
| IST-SL1 | Homo sapiens | | | = 1.187 nM | | | NPASS |
| J-RT3-T3-5 | Homo sapiens | | | = 0.7882 nM | | | NPASS |
| IA-LM | Homo sapiens | | | = 68.58 nM | | | NPASS |
| KNS-42 | Homo sapiens | | | = 18.69 nM | | | NPASS |
| KNS-62 | Homo sapiens | | | = 5.802 nM | | | NPASS |
| KNS-81-FD | Homo sapiens | | | = 20.16 nM | | | NPASS |
| L1210 | Mus musculus | | | = 3.15 nM|= 6.0 nM|= 0.16 nM | | | NPASS |
| L929 | Mus musculus | | | = 0.018 ug.mL-1 | | | NPASS |
| LAMA-84 | Homo sapiens | | | = 7.015 nM | | | NPASS |
| LAN-6 | Homo sapiens | | | = 47.7 nM | | | NPASS |
| LB1047-RCC | Homo sapiens | | | = 40.27 nM | | | NPASS |
| LB2241-RCC | Homo sapiens | | | = 10.12 nM | | | NPASS |
| LB2518-MEL | Homo sapiens | | | = 145.03 nM | | | NPASS |
| L-428 | Homo sapiens | | | = 309.15 nM | | | NPASS |
| LB373-MEL-D | Homo sapiens | | | = 64.11 nM | | | NPASS |
| LB831-BLC | Homo sapiens | | | = 21.23 nM | | | NPASS |
| LC-2-ad | Homo sapiens | | | = 7.896 nM | | | NPASS |
| LCLC-103H cell line | | | | = 1.502 nM | | | NPASS |
| LCLC-97TM1 | Homo sapiens | | | = 5.491 nM | | | NPASS |
| LK-2 | Homo sapiens | | | = 7.503 nM | | | NPASS |
| LN-405 | Homo sapiens | | | = 12.4 nM | | | NPASS |
| ES5 | Homo sapiens | | | = 3.882 nM | | | NPASS |
| LB771-HNC | Homo sapiens | | | = 8.574 nM | | | NPASS |
| L-363 | Homo sapiens | | | = 5.997 nM | | | NPASS |
| Kasumi 1 | | | | = 8.059 nM | | | NPASS |
| KYSE-70 cell line | | | | = 48.35 nM | | | NPASS |
| KOSC-2 | Homo sapiens | | | = 0.6975 nM | | | NPASS |
| KP-4 | Homo sapiens | | | = 2.369 nM | | | NPASS |
| KP-N-YN | Homo sapiens | | | = 46.36 nM | | | NPASS |
| KP-N-YS | Homo sapiens | | | = 22.91 nM | | | NPASS |
| KS-1 | Homo sapiens | | | = 7.987 nM | | | NPASS |
| KU-19-19 | Homo sapiens | | | = 43.72 nM | | | NPASS |
| KU812 cell line | | | | = 16.79 nM | | | NPASS |
| KURAMOCHI | Homo sapiens | | | = 233.07 nM | | | NPASS |
| KY821 | Homo sapiens | | | = 3.69 nM | | | NPASS |
| KYSE-140 | Homo sapiens | | | = 44.94 nM | | | NPASS |
| KYSE-150 cell line | | | | = 46.53 nM | | | NPASS |
| KYSE-180 | Homo sapiens | | | = 6.385 nM | | | NPASS |
| KYSE-270 | Homo sapiens | | | = 9.632 nM | | | NPASS |
| KYSE-410 | Homo sapiens | | | = 9.297 nM | | | NPASS |
| KYSE-450 | Homo sapiens | | | = 9.649 nM | | | NPASS |
| KYSE-510 | Homo sapiens | | | = 5.875 nM | | | NPASS |
| KYSE-520 cell line | | | | = 47.62 nM | | | NPASS |
| Hs-578T | Homo sapiens | | | = 17.31 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 0.07 nM|= 440.0 nM|= 5946000.0 nM|= 0.26 nM|= 4.6 ug.mL-1|= 80.7 nM|= 81.0 nM | | | NPASS |
| JEG-3 | Homo sapiens | | | = 12.48 nM | | | NPASS |
| HUVEC | Homo sapiens | | | = 49.0 nM|= 0.8 nM | | | NPASS |
| GCT | Homo sapiens | | | = 4.728 nM | | | NPASS |
| GI-1 | Homo sapiens | | | = 4.362 nM | | | NPASS |
| GI-ME-N | Homo sapiens | | | = 6.076 nM | | | NPASS |
| GMS-10 | Homo sapiens | | | = 11.28 nM | | | NPASS |
| GOTO | Homo sapiens | | | = 8.207 nM | | | NPASS |
| GP5d | Homo sapiens | | | = 4.674 nM | | | NPASS |
| GR-ST | Homo sapiens | | | = 7.631 nM | | | NPASS |
| GCIY | Homo sapiens | | | = 49.73 nM | | | NPASS |
| GT3TKB | Homo sapiens | | | = 1.92 nM | | | NPASS |
| H4 | Homo sapiens | | | = 5.837 nM | | | NPASS |
| H9 | Homo sapiens | | | = 2.248 nM | | | NPASS |
| HAL-01 | Homo sapiens | | | = 233.41 nM | | | NPASS |
| HC-1 | Homo sapiens | | | = 4.211 nM | | | NPASS |
| HCC 2998 | Homo sapiens | | | = 19.83 nM | | | NPASS |
| HCC1143 | Homo sapiens | | | = 3.8 nM | | | NPASS |
| HCC1187 | Homo sapiens | | | = 2.754 nM | | | NPASS |
| H-EMC-SS | Homo sapiens | | | = 255.94 nM | | | NPASS |
| GB-1 | Homo sapiens | | | = 39.85 nM | | | NPASS |
| GAMG | Homo sapiens | | | = 19.38 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 10.0 nM | | | NPASS |
| ES7 | Homo sapiens | | | = 5.753 nM | | | NPASS |
| ES8 | Homo sapiens | | | = 3.24 nM | | | NPASS |
| ESS-1 | Homo sapiens | | | = 4.876 nM | | | NPASS |
| ETK-1 | Homo sapiens | | | = 5.788 nM | | | NPASS |
| EW-1 | Homo sapiens | | | = 3.148 nM | | | NPASS |
| EW-11 | Homo sapiens | | | = 7.151 nM | | | NPASS |
| EW-13 | Homo sapiens | | | = 36.52 nM | | | NPASS |
| EW-16 | Homo sapiens | | | = 7.832 nM | | | NPASS |
| EW-18 | Homo sapiens | | | = 510.36 nM | | | NPASS |
| EW-22 | Homo sapiens | | | = 29.35 nM | | | NPASS |
| EW-24 | Homo sapiens | | | = 18.01 nM | | | NPASS |
| EW-3 | Homo sapiens | | | = 37.21 nM | | | NPASS |
| FTC-133 | Homo sapiens | | | = 8.444 nM | | | NPASS |
| FaDu | Homo sapiens | | | = 20.02 nM | | | NPASS |
| G-361 | Homo sapiens | | | = 4123.67 nM | | | NPASS |
| G-401 | Homo sapiens | | | = 8.671 nM | | | NPASS |
| G-402 | Homo sapiens | | | = 17.58 nM | | | NPASS |
| HCC1395 | Homo sapiens | | | = 29.25 nM | | | NPASS |
| HCC1419 | Homo sapiens | | | = 57.16 nM | | | NPASS |
| GAK | Homo sapiens | | | = 219.86 nM | | | NPASS |
| HCC1806 | Homo sapiens | | | = 0.6303 nM | | | NPASS |
| HO-1-N-1 | Homo sapiens | | | = 1.756 nM | | | NPASS |
| HOP-62 | Homo sapiens | | | = 1406.87 nM | | | NPASS |
| HOP-92 | Homo sapiens | | | = 25.92 nM | | | NPASS |
| HOS | Homo sapiens | | | = 6.25 nM | | | NPASS |
| HPAF-II | Homo sapiens | | | = 40.05 nM | | | NPASS |
| HSC-2 | Homo sapiens | | | = 20.2 nM | | | NPASS |
| HSC-3 | Homo sapiens | | | = 4.389 nM | | | NPASS |
| HSC-4 | Homo sapiens | | | = 2.355 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | = 0.099 nM|= 4.228 nM | | | NPASS |
| HT-1376 | Homo sapiens | | | = 60.4 nM | | | NPASS |
| HT-144 | Homo sapiens | | | = 3.319 nM | | | NPASS |
| HT-29 | Homo sapiens | | = 2.0 nM | = 0.53 nM|= 4.0 nM|= 30.0 nM|= 45.85 nM|= 4.5 nM | | | NPASS |
| HT-3 | Homo sapiens | | | = 37.07 nM | | | NPASS |
| HT1197 | Homo sapiens | | | = 99.76 nM | | | NPASS |
| HT55 | Homo sapiens | | | = 391.6 nM | | | NPASS |
| HCC1569 | Homo sapiens | | | = 92.26 nM | | | NPASS |
| HTC-C3 | Homo sapiens | | | = 10.38 nM | | | NPASS |
| HN | Homo sapiens | | | = 4.15 nM | | | NPASS |
| HMV-2 cell line | | | | = 3.905 nM | | | NPASS |
| HT | Homo sapiens | | | = 15.64 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 1.0 nM|= 1.6 nM|= 1.11 nM|= 4.371 nM | | | NPASS |
| HCC1954 | Homo sapiens | | | = 121.72 nM | | | NPASS |
| HLE | Homo sapiens | | | = 4.235 nM | | | NPASS |
| HCC1937 | Homo sapiens | | | = 2049.18 nM | | | NPASS |
| HCC2218 | Homo sapiens | | | = 79.26 nM | | | NPASS |
| HCC38 | Homo sapiens | | | = 58.38 nM | | | NPASS |
| HCC70 | Homo sapiens | | | = 20.8 nM|= 3.5 nM | | | NPASS |
| HCE-T | Homo sapiens | | | = 20.01 nM | | | NPASS |
| HCT-116 | Homo sapiens | | = 44.0 nM|= 36.0 nM | = 8.7 nM|= 4.0 nM|= 0.7 nM|= 3.0 nM|= 135.0 nM|= 1.8 nM|= 1.1 nM|= 1.3 nM|= 6.8 nM|= 600.0 nM|= 27.0 nM|= 1.42 nM|= 3.626 nM|= 3.5 nM | | | NPASS |
| HCT-116/VM46 | Homo sapiens | | | = 600.0 nM|> 110.0 nM | | | NPASS |
| HCE-4 | Homo sapiens | | | = 18.09 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 43.0 nM|= 79.4 nM|= 10.0 nM|= 28.5 nM|= 24.0 nM|= 78.58 nM | | | NPASS |
| HD-MY-Z | Homo sapiens | | | = 3.33 nM | | | NPASS |
| HDLM-2 | Homo sapiens | | | = 642.79 nM | | | NPASS |
| HEC-1 | Homo sapiens | | | = 11.35 nM | | | NPASS |
| HEL | Homo sapiens | | | = 32.84 nM | | | NPASS |
| HGC-27 | Homo sapiens | | | = 1.012 nM | | | NPASS |
| HH | Homo sapiens | | | = 6.367 nM | | | NPASS |