IMPPAT Phytochemical information: 
Vinblastine

Vinblastine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
NCI-H2347Homo sapiens= 135.12 nMNPASS
NCI-H226Homo sapiens= 13.81 nMNPASS
NCI-H2291Homo sapiens= 232.1 nMNPASS
NCI-H23Homo sapiens= 5.706 nMNPASS
NCI-H2342Homo sapiens= 950.45 nMNPASS
NCI-H2228Homo sapiens= 41.09 nMNPASS
NCI-H2405Homo sapiens= 826.38 nMNPASS
NCI-H1648Homo sapiens= 5.519 nMNPASS
NCI-H28Homo sapiens= 34.26 nMNPASS
NCI-H292= 3.03 nMNPASS
NCI-H358Homo sapiens= 37.01 nMNPASS
NCI-H441Homo sapiens= 473.3 nMNPASS
NCI-H446Homo sapiens= 2.122 nMNPASS
NCI-H460Homo sapiens= 3.4 nM|= 46.39 nMNPASS
NCI-H510AHomo sapiens= 2.753 nMNPASS
NCI-H2170Homo sapiens= 33.41 nMNPASS
NCI-H2452Homo sapiens= 9.587 nMNPASS
NCI-H2126Homo sapiens= 25.9 nMNPASS
NCI-H1666Homo sapiens= 20.12 nMNPASS
NCI-H209Homo sapiens= 13.15 nMNPASS
NCI-H1650Homo sapiens= 126.77 nMNPASS
NCI-H1651Homo sapiens= 23.0 nMNPASS
NCI-H520= 30.13 nM|= 4.5 nMNPASS
NCI-H1693Homo sapiens= 78.21 nMNPASS
NCI-H1703Homo sapiens= 1.431 nMNPASS
NCI-H1755Homo sapiens= 19.36 nMNPASS
NCI-H1770Homo sapiens= 28.46 nMNPASS
NCI-H1792Homo sapiens= 4.391 nMNPASS
NCI-H1793Homo sapiens= 29.6 nMNPASS
NCI-H1838Homo sapiens= 191.13 nMNPASS
NCI-H1975Homo sapiens= 24.23 nMNPASS
NCI-H1993Homo sapiens= 3395.38 nMNPASS
NCI-H2009Homo sapiens= 53.45 nMNPASS
NCI-H2029Homo sapiens= 203.7 nMNPASS
NCI-H2030Homo sapiens= 27.72 nMNPASS
NCI-H2052Homo sapiens= 24.65 nMNPASS
NCI-H2087Homo sapiens= 30.53 nMNPASS
NCI-H2122Homo sapiens= 3.436 nMNPASS
NCI-H526Homo sapiens= 5.136 nMNPASS
NOMO-1Homo sapiens= 7.859 nMNPASS
NCI-H630Homo sapiens= 241.69 nMNPASS
Nuclear receptor subfamily 0 group B member 1Homo sapiensP51843>67541 nMBindingDB
OAW-28Homo sapiens= 40.72 nMNPASS
OAW-42Homo sapiens= 233.12 nMNPASS
OC-314Homo sapiens= 2.225 nMNPASS
OCI-AML2Homo sapiens= 138.49 nMNPASS
OCUB-MHomo sapiens= 7.561 nMNPASS
OE19Homo sapiens= 412.2 nMNPASS
NYHomo sapiens= 5315.23 nMNPASS
OE33Homo sapiens= 28.59 nMNPASS
ONS-76Homo sapiens= 3.742 nMNPASS
OS-RC-2Homo sapiens= 69.84 nMNPASS
OVCAR-3Homo sapiens= 46.86 nM|= 1.82 nMNPASS
OVCAR-4Homo sapiens= 27.94 nMNPASS
OVCAR-5Homo sapiens= 13.6 nMNPASS
OVCAR-8Homo sapiens= 3.9 nM|= 15.0 nM|= 6.554 nMNPASS
P-glycoprotein 1Homo sapiensP08183= 14600.0 nM|= 34000.0 nM= 2000.0 nM|> 50000.0 nM|= 34000.0 nM|= 10000.0 nM|= 10471.29 nM|= 17700.0 nM|= 19900.0 nM|= 29500.0 nM|= 29000.0 nM= 3000.0 nM= 100.0 nM|= 1300.0 nM|= 140000.0 nM|= 15000.0 nM|= 2100.0 nM|= 36500.0 nMNPASS
OMC-1Homo sapiens= 144.1 nMNPASS
NCI-H596= 156.07 nMNPASS
NUGC-3Homo sapiens= 3.455 nMNPASS
NOS-1Homo sapiens= 40.88 nMNPASS
NCI-H650Homo sapiens= 27.08 nMNPASS
NCI-H661Homo sapiens= 8.047 nMNPASS
NCI-H69Homo sapiens= 1.6 nM|= 525.78 nMNPASS
NCI-H720Homo sapiens= 6.88 nMNPASS
NCI-H727Homo sapiens= 175.7 nMNPASS
NCI-H747Homo sapiens= 81.18 nMNPASS
NCI-H810Homo sapiens= 68.69 nMNPASS
NTERA-2-cl-D1Homo sapiens= 5.893 nMNPASS
NCI-H82Homo sapiens= 1642.17 nMNPASS
NCI/ADR-RESHomo sapiens= 3900.0 ug.mL-1|= 582.0 nM|= 200.0 nMNPASS
NEC8Homo sapiens= 5.122 nMNPASS
NH-12Homo sapiens= 26.35 nMNPASS
NKM-1Homo sapiens= 1.273 nMNPASS
NMC-G1Homo sapiens= 8.484 nMNPASS
NON-PROTEIN TARGET= 12.6 nM|= 2037.0 nM|= 162.0 nM|= 8.5 nM|= 13.0 nM|= 28.0 nM= 18.0 nM|= 246.0 nM|= 0.1 ug.mL-1|= 5.0 nM|= 540.0 nM|= 20.0 nM|= 1.6 nM|= 8.9 nM|> 375.0 nM|= 3.0 nM|= 2818.38 nM|= 0.11 nM|= 1040.0 nM|= 1.38 nM|= 90.0 nM|= 260.0 nM|= 0.4 nM|> 100.0 nM|= 0.63 nM|= 1.24 nM|= 2.28 nM|= 439.73 nM|= 0.0086 ug.mL-1|= 1.8 nM|= 0.099 nM|= 600.0 nM|= 230.0 nM|> 375000.0 nM|= 200.0 nM|= 11.0 nM|= 3.5 nM|= 15.0 nM|= 4.2 nM|= 205.0 nM|= 2.6 ug.mL-1|= 144.0 nM|= 2.0 nM|= 9.0 nM|= 211.0 nM|= 5.2 nM|= 1.0 nM|= 7.9 nM|= 19.6 nM|= 5.1 nM|= 2.9 nM|= 21.0 nM|= 193.0 nMNPASS
P-glycoprotein 1Mus musculusP06795= 8000.0 nMNPASS
NCI-N87Homo sapiens= 5.671 nMNPASS
NCI-H1623Homo sapiens= 503.24 nMNPASS
LXF-289 cell line= 10.29 nMNPASS
NCI-H1573Homo sapiens= 30.74 nMNPASS
MDA-MB-453Homo sapiens= 3.285 nMNPASS
ME-180Homo sapiens= 4.473 nMNPASS
MEG-01Homo sapiens= 14.74 nMNPASS
MEL-HOHomo sapiens= 53.86 nMNPASS
MEL-JUSOHomo sapiens= 17.51 nMNPASS
MFE-280Homo sapiens= 36.08 nMNPASS
MFH-inoHomo sapiens= 588.37 nMNPASS
MDA-MB-435Homo sapiens= 4.4 nM|= 0.34 nM|= 0.29 nM|= 0.42 nM|= 0.27 nM|= 11.0 nM|= 27.5 nM|= 0.4 nM|= 0.49 nM|= 0.5 nMNPASS
MFM-223Homo sapiens= 135.5 nMNPASS
MHH-ES-1Homo sapiens= 5.129 nMNPASS
MHH-NB-11Homo sapiens= 38.85 nMNPASS
MHH-PREB-1Homo sapiens= 1.493 nMNPASS
MIA PaCa-2Homo sapiens= 3.388 nMNPASS
MKN-1Homo sapiens= 10.1 nMNPASS
MKN-28Homo sapiens= 2.698 nMNPASS
MKN-45Homo sapiens= 48.42 nMNPASS
MG-63Homo sapiens= 14.16 nMNPASS
MKN-7Homo sapiens= 76.69 nMNPASS
MDA-MB-415Homo sapiens= 18.55 nMNPASS
MDA-MB-231Homo sapiens= 11.0 nM|= 0.12 nM|= 31.0 nM|= 44.59 nM|= 8.78 nMNPASS
LS-411NHomo sapiens= 66.35 nMNPASS
LS-513Homo sapiens= 56.27 nMNPASS
LU-134-AHomo sapiens= 8.582 nMNPASS
LU-135Homo sapiens= 35.58 nMNPASS
LU-139Homo sapiens= 14.08 nMNPASS
LU-99AHomo sapiens= 20.83 nMNPASS
P-glycoprotein 3Mus musculusP21447> 50000.0 nMNPASS
MDA-MB-361Homo sapiens= 1.662 nMNPASS
LoVoHomo sapiens= 6.025 nMNPASS
M059JHomo sapiens= 15.06 nMNPASS
M14Homo sapiens= 3.191 nMNPASS
MC-IXCHomo sapiens= 2.985 nMNPASS
MC116Homo sapiens= 7.953 nMNPASS
MCF7Homo sapiens= 3.0 nM= 0.22 ug.mL-1|= 0.02 ug.mL-1|= 2.8 nM|= 4.6 nM|= 0.79 nM|= 1.08 ug.mL-1|= 1.37 ug.mL-1|= 0.047 ug.mL-1|= 6.1 ug.mL-1|= 1900.0 nM|= 31.6 nM|= 10.9 nM|> 110.0 nM|= 0.7 nM|= 1.02 ug.mL-1|= 1.22 ug.mL-1NPASS
MDA-MB-157Homo sapiens= 9.064 nMNPASS
MDA-MB-175-VIIHomo sapiens= 267.63 nMNPASS
Lu-65Homo sapiens= 115.72 nMNPASS
ML-2Homo sapiens= 8.652 nMNPASS
MLMAHomo sapiens= 4.652 nMNPASS
MMAC-SFHomo sapiens= 15.09 nMNPASS
NB14Homo sapiens= 4.953 nMNPASS
NB17Homo sapiens= 21.77 nMNPASS
NB5Homo sapiens= 15.7 nMNPASS
NB6Homo sapiens= 80.02 nMNPASS
NB69Homo sapiens= 5.73 nMNPASS
NB7Homo sapiens= 195.12 nMNPASS
NBsusSRHomo sapiens= 3.232 nMNPASS
NB13Homo sapiens= 3.274 nMNPASS
NCI-H1048Homo sapiens= 10.06 nMNPASS
NCI-H1155Homo sapiens= 43.74 nMNPASS
NCI-H1299Homo sapiens= 73.0 nM|= 82.0 nM= 16.42 nMNPASS
NCI-H1304Homo sapiens= 133.77 nMNPASS
NCI-H1355Homo sapiens= 19.54 nMNPASS
NCI-H1395Homo sapiens= 4.277 nMNPASS
NCI-H1437Homo sapiens= 7.76 nMNPASS
NCI-H1563Homo sapiens= 21.46 nMNPASS
NCI-H1092Homo sapiens= 223.56 nMNPASS
NB12Homo sapiens= 61.41 nMNPASS
NB10Homo sapiens= 7.317 nMNPASS
N592= 4.0 nMNPASS
MN-60Homo sapiens= 29.44 nMNPASS
MOLT-13Homo sapiens= 5.603 nMNPASS
MOLT-16Homo sapiens= 2.429 nMNPASS
MOLT-4Homo sapiens= 3.847 nMNPASS
MPP-89Homo sapiens= 30.28 nMNPASS
MRC5Homo sapiens= 24.0 nMNPASS
MS-1Homo sapiens= 30.83 nMNPASS
MSTO-211HHomo sapiens= 12.22 nMNPASS
MV4-11Homo sapiens= 2.805 nMNPASS
MX1Homo sapiens= 2.0 nM|= 2.9 nM|= 2.2 nMNPASS
MZ1-PCHomo sapiens= 24.19 nMNPASS
MZ2-MELHomo sapiens= 60.31 nMNPASS
MZ7-melHomo sapiens= 11.08 nMNPASS
MeWoHomo sapiens= 9.134 nMNPASS
MoHomo sapiens= 880.24 nMNPASS
Monoamine oxidase BBos taurusP56560= 77000.0 nMNPASS
Multidrug resistance-associated protein 1Homo sapiensP3352730000 nM|= 30000.0 nMBindingDB, NPASS
NCI-H1581Homo sapiens= 4.236 nMNPASS
P12-IchikawaHomo sapiens= 1.704 nMNPASS
SNU-398Homo sapiens= 38.0 nM|= 26.0 nMNPASS
P388Mus musculus= 1.7 nM|= 8.2 nM|= 4.1 nM|= 0.7 nM|= 27.0 nM|= 0.6 nMNPASS
Solute carrier organic anion transporter family member 1B3Homo sapiensQ9NPD543500 nM|= 43500.0 nM18600 nM|= 18600.0 nMBindingDB, NPASS
Steroidogenic factor 1Homo sapiensQ13285>67541 nMBindingDB
T-24Homo sapiens= 5.104 nMNPASS
T47DHomo sapiens= 25.0 nM|= 43.0 nM|= 32.0 nM= 7.711 nM|= 5.0 nMNPASS
T84Homo sapiens= 8147.21 nMNPASS
T98GHomo sapiens= 11.4 nMNPASS
TCC-SUPHomo sapiens= 23.63 nMNPASS
Solute carrier organic anion transporter family member 1B1Homo sapiensQ9Y6L646800 nM|= 46800.0 nM10200 nM|= 10200.0 nMBindingDB, NPASS
TE-1Homo sapiens= 10.85 nMNPASS
TE-11Homo sapiens= 5.128 nMNPASS
TE-12Homo sapiens= 700.72 nMNPASS
TE-5Homo sapiens= 6.135 nMNPASS
TE-6Homo sapiens= 56.47 nMNPASS
TE-8Homo sapiens= 6.156 nMNPASS
TE-9Homo sapiens= 4.27 nMNPASS
TGBC11TKBHomo sapiens= 15.83 nMNPASS
TE-10Homo sapiens= 21.47 nMNPASS
TGBC1TKBHomo sapiens= 31.21 nMNPASS
Similar to alpha-tubulin isoform 1Bos taurus600 nM|700 nMBindingDB
SW982Homo sapiens= 8.919 nMNPASS
SW13Homo sapiens= 5.49 nMNPASS
SW1417Homo sapiens= 423.54 nMNPASS
SW1463Homo sapiens= 69.69 nMNPASS
SW1573Homo sapiens= 33.25 nMNPASS
SW1710Homo sapiens= 5.607 nMNPASS
SW1783Homo sapiens= 85.55 nMNPASS
SW1990Homo sapiens= 61.39 nMNPASS
SiHaHomo sapiens= 109.77 nMNPASS
SW48Homo sapiens= 6.943 nMNPASS
SW684Homo sapiens= 101.3 nMNPASS
SW756Homo sapiens= 14.7 nMNPASS
SW780Homo sapiens= 2.329 nMNPASS
SW837Homo sapiens= 120.44 nMNPASS
SW872Homo sapiens= 255.22 nMNPASS
SW900Homo sapiens= 25.41 nMNPASS
SW948Homo sapiens= 75.99 nMNPASS
SW626Homo sapiens= 23.21 nMNPASS
TGBC24TKBHomo sapiens= 32.52 nMNPASS
TI-73Homo sapiens= 3.212 nMNPASS
TK-10Homo sapiens= 42.4 nMNPASS
UMC-11Homo sapiens= 76.22 nMNPASS
UMUC3Homo sapiens= 5.107 nMNPASS
UO-31Homo sapiens= 13.94 nMNPASS
VA-ES-BJHomo sapiens= 3.273 nMNPASS
VM-CUB-1Homo sapiens= 4.281 nMNPASS
VMRC-RCZHomo sapiens= 19.27 nMNPASS
VeroChlorocebus aethiops< 3700.0 nM= 27060.0 nMNPASS
UACC-893Homo sapiens= 98.3 nMNPASS
WM-115Homo sapiens= 10.16 nMNPASS
YAPCHomo sapiens= 86.99 nMNPASS
YH-13Homo sapiens= 3.702 nMNPASS
YKG-1Homo sapiens= 5.534 nMNPASS
ZR-75-1Homo sapiens= 8.0 nMNPASS
ZR-75-30Homo sapiens= 402.55 nMNPASS
no-10Homo sapiens= 270.54 nMNPASS
no-11Homo sapiens= 38.83 nMNPASS
WRL68Homo sapiens= 1.45 ug.mL-1|= 2.6 ug.mL-1NPASS
UACC-62Homo sapiens= 8.062 nMNPASS
UACC-257Homo sapiens= 90.53 nMNPASS
U2OSHomo sapiens= 25.72 nMNPASS
TYK-nuHomo sapiens= 11.9 nMNPASS
Thromboxane-A synthaseHomo sapiensP24557= 1870.0 nMNPASS
Trypanosoma bruceiTrypanosoma brucei= 410.0 nMNPASS
Trypanosoma brucei bruceiTrypanosoma brucei brucei= 94.0 nMNPASS
TubulinBos taurusQ862F3= 700.0 nM|= 600.0 nMNPASS
TubulinHomo sapiensQ9BUF5= 200.0 nM= 70.0 nM|= 300.0 nM|= 2100.0 nMNPASS
TubulinSus scrofaP02550= 600.0 nM|= 1600.0 nM|= 1100.0 nMNPASS
Tubulin alpha-1A chainPigP02550200 nMBindingDB
Tubulin beta chainBos taurusQ6B856> 100000.0 nMNPASS
Tubulin beta chainSus scrofaP025541100 nM|600 nM|130 nM|1600 nMBindingDB
Tubulin beta chain [1-43]LeishmadonovaniP211481000 nMBindingDB
Tubulin beta-2B chainBos taurusQ6B856>100000 nMBindingDB
U-118-MGHomo sapiens= 45.16 nMNPASS
U-251Homo sapiens= 8.1 nM|= 5.018 nMNPASS
U-266Homo sapiens= 10.8 nMNPASS
U-87 MGHomo sapiens= 29.98 nMNPASS
U-937Homo sapiens= 6880.0 nM|= 0.49 nMNPASS
SW1088Homo sapiens= 16.97 nMNPASS
SW-620Homo sapiens= 8.836 nMNPASS
SW 962Homo sapiens= 19.39 nMNPASS
SW 954Homo sapiens= 9.662 nMNPASS
RPMI-2650Homo sapiens= 26.61 nMNPASS
RPMI-7951Homo sapiens= 1.658 nMNPASS
RPMI-8226Homo sapiens= 28.0 nM|= 2.852 nMNPASS
RPMI-8866Homo sapiens= 1.966 nMNPASS
RS4-11Homo sapiens= 4.508 nMNPASS
RT-112Homo sapiens= 2.708 nMNPASS
RVH-421Homo sapiens= 7.249 nMNPASS
RO82-W-1Homo sapiens= 5.57 nMNPASS
RXF 393Homo sapiens= 1.439 nMNPASS
Reverse transcriptaseHuman immunodeficiency virus 1>246000 nMBindingDB
S-117Homo sapiens= 5.576 nMNPASS
SAOS-2Homo sapiens= 32.31 nMNPASS
SASHomo sapiens= 28.13 nMNPASS
SBC-1Homo sapiens= 8.104 nMNPASS
SBC-5Homo sapiens= 7.471 nMNPASS
SCC-15Homo sapiens= 23.15 nMNPASS
Ramos-2G6-4C10Homo sapiens= 1.546 nMNPASS
RMG-IHomo sapiens= 116.58 nMNPASS
RKOHomo sapiens= 8.239 nMNPASS
RH-18Homo sapiens= 1128.93 nMNPASS
P388/ADRMus musculus= 95.0 nM|= 4.3 nMNPASS
PA-1Homo sapiens= 0.025 ug.mL-1|= 1.15 ug.mL-1|= 0.15 ug.mL-1|= 0.03 ug.mL-1|= 8.092 nM|= 4.6 nMNPASS
PANC-03-27Homo sapiens= 5.472 nMNPASS
PANC-08-13Homo sapiens= 61.47 nMNPASS
PC-14Homo sapiens= 3.534 nMNPASS
PC-3Homo sapiens= 5.5 nM|= 5.0 nM|= 33.37 nM|= 766.0 nMNPASS
PFSK-1Homo sapiens= 4.972 nMNPASS
PSN1Homo sapiens= 1.248 nMNPASS
Panc1005Homo sapiens= 42.8 nMNPASS
Plasmodium falciparumPlasmodium falciparum= 2.0 nMNPASS
Plasmodium yoelii yoeliiPlasmodium yoelii yoelii= 7950.0 nMNPASS
QIMR-WILHomo sapiens= 8.95 nMNPASS
RCC10RGBHomo sapiens= 510.4 nMNPASS
RCM-1Homo sapiens= 1369.69 nMNPASS
RDHomo sapiens= 4.172 nM|= 52.5 nM|= 53.0 nMNPASS
RERF-LC-MSHomo sapiens= 15.15 nMNPASS
RH-1Homo sapiens= 3.4 nMNPASS
SCC-25Homo sapiens= 15.68 nMNPASS
P30-OHKHomo sapiens= 11.07 nMNPASS
SCC-4Homo sapiens= 2.395 nMNPASS
SCHHomo sapiens= 29.72 nMNPASS
SK-N-FIHomo sapiens= 642.78 nMNPASS
SK-NEP-1Homo sapiens= 1.505 nMNPASS
SK-OV-3Homo sapiens= 2.7 nM|= 0.039 nM|= 8155.03 nMNPASS
SK-PN-DWHomo sapiens= 6.138 nMNPASS
SK-UT-1Homo sapiens= 11.75 nMNPASS
SKG-IIIaHomo sapiens= 17.24 nMNPASS
SN12CHomo sapiens= 16.06 nMNPASS
SK-N-DZHomo sapiens= 37.37 nMNPASS
SNB-75Homo sapiens= 11.25 nMNPASS
LS-123Homo sapiens= 53.33 nMNPASS
SNU-423Homo sapiens= 19.47 nMNPASS
SNU-449Homo sapiens= 127.72 nMNPASS
SNU-5Homo sapiens= 132.84 nMNPASS
SNU-C2BHomo sapiens= 24.67 nMNPASS
SNU1Homo sapiens= 1.622 nMNPASS
SW 1116Homo sapiens= 1163.6 nMNPASS
SNU-387Homo sapiens= 11.42 nMNPASS
SK-N-ASHomo sapiens= 8.669 nMNPASS
SK-MES-1Homo sapiens= 8.645 nMNPASS
SK-MEL3Homo sapiens= 717.01 nMNPASS
SF-126Homo sapiens= 21.9 nMNPASS
SF-268Homo sapiens= 16.19 nMNPASS
SF-295Homo sapiens= 36.31 nMNPASS
SF-539Homo sapiens= 1.211 nMNPASS
SH-4Homo sapiens= 43.54 nMNPASS
SHP77Homo sapiens= 148.18 nMNPASS
SJRH30Homo sapiens= 59.36 nMNPASS
SJSA-1Homo sapiens= 12.06 nMNPASS
SK-BR-3Homo sapiens= 72.0 nM|= 0.91 nMNPASS
SK-HEP1Homo sapiens= 12.05 nMNPASS
SK-LMS-1Homo sapiens= 58.6 nMNPASS
SK-LU-1Homo sapiens= 18.71 nMNPASS
SK-MEL-1Homo sapiens= 67.32 nMNPASS
SK-MEL-2Homo sapiens= 53.3 nMNPASS
SK-MEL-24Homo sapiens= 31.55 nMNPASS
SK-MEL-28Homo sapiens= 17.04 nMNPASS
SK-MEL-30Homo sapiens= 415.46 nMNPASS
SCC-9Homo sapiens= 10.66 nMNPASS
LS-1034Homo sapiens= 2844.0 nMNPASS
MDA-MB-468Homo sapiens= 4.6 nMNPASS
LNCaP-Clone-FGCHomo sapiens= 8.279 nMNPASS
COLO-829Homo sapiens= 19.17 nMNPASS
COR-L105Homo sapiens= 65.75 nMNPASS
COR-L23Homo sapiens= 3.623 nMNPASS
COR-L88Homo sapiens= 24.32 nMNPASS
CP50-MEL-BHomo sapiens= 13.12 nMNPASS
CP66-MELHomo sapiens= 48.58 nMNPASS
CTB-1Homo sapiens= 1.636 nMNPASS
COLO-824Homo sapiens= 136.2 nMNPASS
CTV-1Homo sapiens= 1.405 nMNPASS
CWR22RHomo sapiens= 9.815 nMNPASS
Ca-SkiHomo sapiens= 4.694 nMNPASS
Ca9-22Homo sapiens= 6.391 nMNPASS
CaR-1Homo sapiens= 45.73 nMNPASS
Caco-2Homo sapiens= 2.8 ug.mL-1|= 0.46 ug.mL-1NPASS
Calu-3Homo sapiens= 551.0 nMNPASS
Calu-6Homo sapiens= 149.1 nMNPASS
CW-2Homo sapiens= 101.38 nMNPASS
Canalicular multispecific organic anion transporter 1Homo sapiensQ92887= 21000.0 nMNPASS
COLO-800Homo sapiens= 3.342 nMNPASS
COLO-741Homo sapiens= 2.139 nMNPASS
CEMHomo sapiens= 2.0 nM|= 1.0 nMNPASS
CFPAC-1Homo sapiens= 93.2 nMNPASS
CGTH-W-1Homo sapiens= 5.556 nMNPASS
CHL-1Homo sapiens= 12.0 nMNPASS
CHOCricetulus griseus= 17.0 nMNPASS
CHO-TAX 5-6Cricetulus griseus= 6.9 nMNPASS
CHO-VV 3-2Cricetulus griseus= 66.0 nMNPASS
COLO-792Homo sapiens= 25.63 nMNPASS
CHP-212Homo sapiens= 3.547 nMNPASS
COLO 320DMHomo sapiens= 0.52 ug.mL-1|= 1.6 ug.mL-1NPASS
COLO-320-HSRHomo sapiens= 203.92 nMNPASS
COLO-668Homo sapiens= 562.6 nMNPASS
COLO-678Homo sapiens= 2480.78 nMNPASS
COLO-679Homo sapiens= 5415.81 nMNPASS
COLO-680NHomo sapiens= 74.71 nMNPASS
COLO-684Homo sapiens= 7.666 nMNPASS
COLO 320Homo sapiens= 1.6 ug.mL-1|= 0.52 ug.mL-1NPASS
Capan-2Homo sapiens= 114.18 nMNPASS
ChaGo-K-1Homo sapiens= 1.013 nMNPASS
Cytochrome P450 3A4Homo sapiensP0868426000 nM|= 26000.0 nMBindingDB, NPASS
DU-145Homo sapiens= 0.063 nM|= 98.66 nMNPASS
DU-4475Homo sapiens= 383.01 nMNPASS
DaoyHomo sapiens= 3.102 nMNPASS
Detroit562Homo sapiens= 5.531 nMNPASS
DoTc2-4510Homo sapiens= 16.52 nMNPASS
EC-GI-10Homo sapiens= 3.531 nMNPASS
ECC10Homo sapiens= 21.16 nMNPASS
DSH1Homo sapiens= 23.21 nMNPASS
EFM-19Homo sapiens= 5.242 nMNPASS
EFO-27Homo sapiens= 7.449 nMNPASS
EGI-1Homo sapiens= 10.81 nMNPASS
EKVXHomo sapiens= 278.22 nMNPASS
EM-2Homo sapiens= 5.316 nMNPASS
EOL1Homo sapiens= 1.261 nMNPASS
EPLC-272HHomo sapiens= 10.78 nMNPASS
ES1Homo sapiens= 4.714 nMNPASS
EFO-21Homo sapiens= 44.03 nMNPASS
DOKHomo sapiens= 4.196 nMNPASS
DOHH-2Homo sapiens= 1.809 nMNPASS
DMS-79Homo sapiens= 534.65 nMNPASS
D-247MGHomo sapiens= 6.979 nMNPASS
D-263MGHomo sapiens= 9.278 nMNPASS
D-336MGHomo sapiens= 7.255 nMNPASS
D-392MGHomo sapiens= 18.86 nMNPASS
D-423MGHomo sapiens= 8.639 nMNPASS
D-502MGHomo sapiens= 23.49 nMNPASS
D-542MGHomo sapiens= 3876.68 nMNPASS
D-566MGHomo sapiens= 2.043 nMNPASS
D283 Med= 39.1 nMNPASS
DBHomo sapiens= 1.687 nMNPASS
DBTRG-05MGHomo sapiens= 225.99 nMNPASS
DELHomo sapiens= 2.16 nMNPASS
DJM-1Homo sapiens= 2816.86 nMNPASS
DK-MGHomo sapiens= 6.646 nMNPASS
DLD-1Homo sapiens= 129.0 nM|= 160.0 nMNPASS
DMS-114Homo sapiens= 20.94 nMNPASS
DMS-273Homo sapiens= 3.396 nMNPASS
CCRF-CEMHomo sapiens= 0.1 ug.mL-1|= 1.2 nM|= 0.4 nM|= 28.7 nM|= 206.6 nM|= 4.0 nM|= 0.73 nM|= 78.0 nM|= 496.0 nM|= 0.03 ug.mL-1|= 500.0 nM|= 0.7 nM|= 80.0 nM|= 0.38 nM|= 4.1 nM|= 9.4 nM|= 0.8 nM|= 2.0 nM|= 10.05 nM|= 2.9 nM|= 870.0 nM|= 1.3 nM|= 670.0 nMNPASS
CAS-1Homo sapiens= 93.12 nMNPASS
CAPAN-1Homo sapiens= 52.3 nMNPASS
CAMA-1Homo sapiens= 32.01 nMNPASS
A498Homo sapiens= 5.938 nMNPASS
A549Homo sapiens= 0.9 nM|= 0.5 nM= 9.9 nM|= 1.1 nM|= 17.0 nM|= 20.0 nM|= 4.954 nMNPASS
A673Homo sapiens= 6.875 nMNPASS
A704Homo sapiens= 119.71 nMNPASS
ABC-1Homo sapiens= 15.49 nMNPASS
ACHNHomo sapiens= 25.0 nM|= 59.04 nMNPASS
ACNHomo sapiens= 40.29 nMNPASS
A4-FukHomo sapiens= 1.867 nMNPASS
AGSHomo sapiens= 12.3 nMNPASS
AM-38Homo sapiens= 36.92 nMNPASS
AN3-CAHomo sapiens= 9.765 nMNPASS
ASPC1Homo sapiens= 13.21 nMNPASS
ATN-1Homo sapiens= 1.034 nMNPASS
ATP-binding cassette sub-family C member 2Homo sapiensQ9288721000 nMBindingDB
ATP-dependent translocase ABCB1Homo sapiensP0818314600 nM|34000 nM34000 nM|2000 nM|>50000 nM|29000 nM|29500 nM|17700 nM|19900 nM|10471 nM|10000 nM3000 nM100 nM|1300 nM|2100 nM|140000 nM|36500 nM|15000 nMBindingDB
ATP-dependent translocase ABCB1Mus musculusP067958000 nMBindingDB
ALL-POHomo sapiens= 5.215 nMNPASS
A388Homo sapiens= 6.915 nMNPASS
A3-KAWHomo sapiens= 4.32 nMNPASS
A2780Homo sapiens= 61.66 nM|= 5.0 nM|= 4.608 nMNPASS
23132-87Homo sapiens= 20.64 nMNPASS
5637Homo sapiens= 0.951 nMNPASS
639-VHomo sapiens= 5.605 nMNPASS
647-VHomo sapiens= 23.03 nMNPASS
697Homo sapiens= 6.225 nMNPASS
769-PHomo sapiens= 25.55 nMNPASS
786-0Homo sapiens= 4.5 nM|= 0.31 nM|= 15.58 nMNPASS
8-MG-BAHomo sapiens= 6.335 nMNPASS
8305CHomo sapiens= 3.67 nMNPASS
8505CHomo sapiens= 3.109 nMNPASS
A-375Homo sapiens= 23.53 nMNPASS
A-427Homo sapiens= 12.55 nMNPASS
A-431Homo sapiens= 4975.15 nMNPASS
A101DHomo sapiens= 31.39 nMNPASS
A172Homo sapiens= 9.616 nMNPASS
A204Homo sapiens= 8.765 nMNPASS
A2058Homo sapiens= 4.0 nM|= 1.218 nM|= 3.7 nMNPASS
ATP-dependent translocase ABCB1Mus musculusP21447>50000 nMBindingDB
ES3Homo sapiens= 2.766 nMNPASS
AU565Homo sapiens= 3.448 nM|= 4.0 nMNPASS
Arachidonate 15-lipoxygenaseOryctolagus cuniculusP12530= 5037.0 nMNPASS
LOX IMVIHomo sapiens= 6.977 nMNPASS
C2BBe1Homo sapiens= 16.88 nMNPASS
C32Homo sapiens= 866.85 nMNPASS
C3AHomo sapiens= 332.14 nMNPASS
C8166Homo sapiens= 27.01 nMNPASS
CAKI-1Homo sapiens= 24.61 nMNPASS
CAL-120Homo sapiens= 87.26 nMNPASS
Bile salt export pumpHomo sapiensO95342114700 nM|62000 nM|= 114700.0 nM|= 62000.0 nMBindingDB, NPASS
CAL-12THomo sapiens= 55.97 nMNPASS
CAL-33Homo sapiens= 6.184 nMNPASS
CAL-39Homo sapiens= 5.114 nMNPASS
CAL-51Homo sapiens= 16.39 nMNPASS
CAL-54Homo sapiens= 60.59 nMNPASS
CAL-62Homo sapiens= 10.1 nMNPASS
CAL-72Homo sapiens= 647.18 nMNPASS
CAL-85-1Homo sapiens= 6079.95 nMNPASS
CAL-27Homo sapiens= 2.086 nMNPASS
Beta tubulinLeishmadonovaniQ25270= 1000.0 nMNPASS
BeckerHomo sapiens= 1.126 nMNPASS
BXPC-3Homo sapiens= 8.01 nMNPASS
B16Mus musculus= 3.6 ug.mL-1NPASS
BALL-1Homo sapiens= 313.17 nMNPASS
BB30-HNCHomo sapiens= 8.315 nMNPASS
BB49-HNCHomo sapiens= 12.56 nMNPASS
BB65-RCCHomo sapiens= 20.7 nMNPASS
BCPAPHomo sapiens= 2.33 nMNPASS
BE-13Homo sapiens= 1.416 nMNPASS
BENHomo sapiens= 81.23 nMNPASS
BFTC-905Homo sapiens= 3.773 nMNPASS
BFTC-909Homo sapiens= 7.532 nMNPASS
BHT-101Homo sapiens= 31.36 nMNPASS
BHYHomo sapiens= 15.33 nMNPASS
BPH-1Homo sapiens= 3.263 nMNPASS
BT-20Homo sapiens= 37.68 nMNPASS
BT-474Homo sapiens= 94.15 nMNPASS
BT-549Homo sapiens= 7.977 nMNPASS
BV-173Homo sapiens= 42.27 nMNPASS
Amine oxidase [flavin-containing] BBos taurusP5656077000 nMBindingDB
ES4Homo sapiens= 13.83 nMNPASS
C-33-AHomo sapiens= 12.66 nMNPASS
ES6Homo sapiens= 115.12 nMNPASS
JVM-2Homo sapiens= 5585.18 nMNPASS
JVM-3Homo sapiens= 1.705 nMNPASS
K5Homo sapiens= 4.682 nMNPASS
K562Homo sapiens= 1.0 nM= 3000.0 nM|= 0.88 nM|= 170.0 nM|= 193000.0 nM|= 0.36 nM|= 1082.28 nM|= 7.0 nM|= 2.7 nM|= 10.0 nMNPASS
KALS-1Homo sapiens= 7.787 nMNPASS
KARPAS-299Homo sapiens= 1657.4 nMNPASS
KARPAS-45Homo sapiens= 1.793 nMNPASS
JARHomo sapiens= 0.608 nMNPASS
KBHomo sapiens= 0.046 ug.mL-1|= 0.46 ug.mL-1|= 1.0 nM|= 0.8 nMNPASS
KE-37Homo sapiens= 3.993 nMNPASS
KG-1= 18.38 nMNPASS
KGNHomo sapiens= 33.33 nMNPASS
KINGS-1Homo sapiens= 9.324 nMNPASS
KLEHomo sapiens= 309.24 nMNPASS
KM-H2Homo sapiens= 5.339 nMNPASS
KM12Homo sapiens= 14.42 nMNPASS
KB 3-1Homo sapiens= 9271000.0 nMNPASS
KMOE-2Homo sapiens= 20.76 nMNPASS
J82Homo sapiens= 68.47 nMNPASS
J774Mus musculus= 2.1 nMNPASS
HuCCT-1Homo sapiens= 17.29 nMNPASS
HuO-3N1Homo sapiens= 4.827 nMNPASS
HuO9Homo sapiens= 12.64 nMNPASS
HuP-T3Homo sapiens= 17.96 nMNPASS
HuP-T4Homo sapiens= 43.18 nMNPASS
HuTu80Homo sapiens= 12.28 nMNPASS
Huh-7Homo sapiens= 87.74 nMNPASS
J774.2= 15.9 nM|= 0.8 nMNPASS
Human immunodeficiency virus type 1 reverse transcriptaseHuman immunodeficiency virus 1Q72547> 200.0 ug.mL-1NPASS
IGR-1Homo sapiens= 2.076 nMNPASS
IGROV-1Homo sapiens= 215.27 nMNPASS
IMR-90Homo sapiens> 1000.0 nMNPASS
IST-MEL1Homo sapiens= 4.526 nMNPASS
IST-MES1Homo sapiens= 67.68 nMNPASS
IST-SL1Homo sapiens= 1.187 nMNPASS
J-RT3-T3-5Homo sapiens= 0.7882 nMNPASS
IA-LMHomo sapiens= 68.58 nMNPASS
KNS-42Homo sapiens= 18.69 nMNPASS
KNS-62Homo sapiens= 5.802 nMNPASS
KNS-81-FDHomo sapiens= 20.16 nMNPASS
L1210Mus musculus= 3.15 nM|= 6.0 nM|= 0.16 nMNPASS
L929Mus musculus= 0.018 ug.mL-1NPASS
LAMA-84Homo sapiens= 7.015 nMNPASS
LAN-6Homo sapiens= 47.7 nMNPASS
LB1047-RCCHomo sapiens= 40.27 nMNPASS
LB2241-RCCHomo sapiens= 10.12 nMNPASS
LB2518-MELHomo sapiens= 145.03 nMNPASS
L-428Homo sapiens= 309.15 nMNPASS
LB373-MEL-DHomo sapiens= 64.11 nMNPASS
LB831-BLCHomo sapiens= 21.23 nMNPASS
LC-2-adHomo sapiens= 7.896 nMNPASS
LCLC-103H cell line= 1.502 nMNPASS
LCLC-97TM1Homo sapiens= 5.491 nMNPASS
LK-2Homo sapiens= 7.503 nMNPASS
LN-405Homo sapiens= 12.4 nMNPASS
ES5Homo sapiens= 3.882 nMNPASS
LB771-HNCHomo sapiens= 8.574 nMNPASS
L-363Homo sapiens= 5.997 nMNPASS
Kasumi 1= 8.059 nMNPASS
KYSE-70 cell line= 48.35 nMNPASS
KOSC-2Homo sapiens= 0.6975 nMNPASS
KP-4Homo sapiens= 2.369 nMNPASS
KP-N-YNHomo sapiens= 46.36 nMNPASS
KP-N-YSHomo sapiens= 22.91 nMNPASS
KS-1Homo sapiens= 7.987 nMNPASS
KU-19-19Homo sapiens= 43.72 nMNPASS
KU812 cell line= 16.79 nMNPASS
KURAMOCHIHomo sapiens= 233.07 nMNPASS
KY821Homo sapiens= 3.69 nMNPASS
KYSE-140Homo sapiens= 44.94 nMNPASS
KYSE-150 cell line= 46.53 nMNPASS
KYSE-180Homo sapiens= 6.385 nMNPASS
KYSE-270Homo sapiens= 9.632 nMNPASS
KYSE-410Homo sapiens= 9.297 nMNPASS
KYSE-450Homo sapiens= 9.649 nMNPASS
KYSE-510Homo sapiens= 5.875 nMNPASS
KYSE-520 cell line= 47.62 nMNPASS
Hs-578THomo sapiens= 17.31 nMNPASS
HepG2Homo sapiens= 0.07 nM|= 440.0 nM|= 5946000.0 nM|= 0.26 nM|= 4.6 ug.mL-1|= 80.7 nM|= 81.0 nMNPASS
JEG-3Homo sapiens= 12.48 nMNPASS
HUVECHomo sapiens= 49.0 nM|= 0.8 nMNPASS
GCTHomo sapiens= 4.728 nMNPASS
GI-1Homo sapiens= 4.362 nMNPASS
GI-ME-NHomo sapiens= 6.076 nMNPASS
GMS-10Homo sapiens= 11.28 nMNPASS
GOTOHomo sapiens= 8.207 nMNPASS
GP5dHomo sapiens= 4.674 nMNPASS
GR-STHomo sapiens= 7.631 nMNPASS
GCIYHomo sapiens= 49.73 nMNPASS
GT3TKBHomo sapiens= 1.92 nMNPASS
H4Homo sapiens= 5.837 nMNPASS
H9Homo sapiens= 2.248 nMNPASS
HAL-01Homo sapiens= 233.41 nMNPASS
HC-1Homo sapiens= 4.211 nMNPASS
HCC 2998Homo sapiens= 19.83 nMNPASS
HCC1143Homo sapiens= 3.8 nMNPASS
HCC1187Homo sapiens= 2.754 nMNPASS
H-EMC-SSHomo sapiens= 255.94 nMNPASS
GB-1Homo sapiens= 39.85 nMNPASS
GAMGHomo sapiens= 19.38 nMNPASS
HeLaHomo sapiens= 10.0 nMNPASS
ES7Homo sapiens= 5.753 nMNPASS
ES8Homo sapiens= 3.24 nMNPASS
ESS-1Homo sapiens= 4.876 nMNPASS
ETK-1Homo sapiens= 5.788 nMNPASS
EW-1Homo sapiens= 3.148 nMNPASS
EW-11Homo sapiens= 7.151 nMNPASS
EW-13Homo sapiens= 36.52 nMNPASS
EW-16Homo sapiens= 7.832 nMNPASS
EW-18Homo sapiens= 510.36 nMNPASS
EW-22Homo sapiens= 29.35 nMNPASS
EW-24Homo sapiens= 18.01 nMNPASS
EW-3Homo sapiens= 37.21 nMNPASS
FTC-133Homo sapiens= 8.444 nMNPASS
FaDuHomo sapiens= 20.02 nMNPASS
G-361Homo sapiens= 4123.67 nMNPASS
G-401Homo sapiens= 8.671 nMNPASS
G-402Homo sapiens= 17.58 nMNPASS
HCC1395Homo sapiens= 29.25 nMNPASS
HCC1419Homo sapiens= 57.16 nMNPASS
GAKHomo sapiens= 219.86 nMNPASS
HCC1806Homo sapiens= 0.6303 nMNPASS
HO-1-N-1Homo sapiens= 1.756 nMNPASS
HOP-62Homo sapiens= 1406.87 nMNPASS
HOP-92Homo sapiens= 25.92 nMNPASS
HOSHomo sapiens= 6.25 nMNPASS
HPAF-IIHomo sapiens= 40.05 nMNPASS
HSC-2Homo sapiens= 20.2 nMNPASS
HSC-3Homo sapiens= 4.389 nMNPASS
HSC-4Homo sapiens= 2.355 nMNPASS
HT-1080Homo sapiens= 0.099 nM|= 4.228 nMNPASS
HT-1376Homo sapiens= 60.4 nMNPASS
HT-144Homo sapiens= 3.319 nMNPASS
HT-29Homo sapiens= 2.0 nM= 0.53 nM|= 4.0 nM|= 30.0 nM|= 45.85 nM|= 4.5 nMNPASS
HT-3Homo sapiens= 37.07 nMNPASS
HT1197Homo sapiens= 99.76 nMNPASS
HT55Homo sapiens= 391.6 nMNPASS
HCC1569Homo sapiens= 92.26 nMNPASS
HTC-C3Homo sapiens= 10.38 nMNPASS
HNHomo sapiens= 4.15 nMNPASS
HMV-2 cell line= 3.905 nMNPASS
HTHomo sapiens= 15.64 nMNPASS
HL-60Homo sapiens= 1.0 nM|= 1.6 nM|= 1.11 nM|= 4.371 nMNPASS
HCC1954Homo sapiens= 121.72 nMNPASS
HLEHomo sapiens= 4.235 nMNPASS
HCC1937Homo sapiens= 2049.18 nMNPASS
HCC2218Homo sapiens= 79.26 nMNPASS
HCC38Homo sapiens= 58.38 nMNPASS
HCC70Homo sapiens= 20.8 nM|= 3.5 nMNPASS
HCE-THomo sapiens= 20.01 nMNPASS
HCT-116Homo sapiens= 44.0 nM|= 36.0 nM= 8.7 nM|= 4.0 nM|= 0.7 nM|= 3.0 nM|= 135.0 nM|= 1.8 nM|= 1.1 nM|= 1.3 nM|= 6.8 nM|= 600.0 nM|= 27.0 nM|= 1.42 nM|= 3.626 nM|= 3.5 nMNPASS
HCT-116/VM46Homo sapiens= 600.0 nM|> 110.0 nMNPASS
HCE-4Homo sapiens= 18.09 nMNPASS
HCT-15Homo sapiens= 43.0 nM|= 79.4 nM|= 10.0 nM|= 28.5 nM|= 24.0 nM|= 78.58 nMNPASS
HD-MY-ZHomo sapiens= 3.33 nMNPASS
HDLM-2Homo sapiens= 642.79 nMNPASS
HEC-1Homo sapiens= 11.35 nMNPASS
HELHomo sapiens= 32.84 nMNPASS
HGC-27Homo sapiens= 1.012 nMNPASS
HHHomo sapiens= 6.367 nMNPASS