IMPPAT Phytochemical information: 
Coronaridine

Coronaridine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Vanilloid receptorHomo sapiensQ8NER1= 170000.0 nMNPASS
Transient receptor potential cation channel subfamily M member 8Mus musculusQ8R4D5= 16000.0 nM|= 3000.0 nMNPASS
Transient receptor potential cation channel subfamily A member 1Homo sapiensO75762= 16000.0 nMNPASS
SW480Homo sapiens= 10400.0 nMNPASS
RKOHomo sapiens> 40000.0 nMNPASS
RAW264.7Mus musculus= 25500.0 nMNPASS
NON-PROTEIN TARGET= 24400.0 nMNPASS
HeLaHomo sapiens> 40000.0 nMNPASS
HEK293Homo sapiens= 31700.0 nMNPASS
HEK-293THomo sapiens> 40000.0 nMNPASS
HCT-116Homo sapiens= 11600.0 nMNPASS
AcetylcholinesteraseElectrophorus electricusO42275= 8600.0 nMNPASS
A2780Homo sapiens= 9.9 ug.mL-1NPASS
KBHomo sapiens= 11.5 ug.mL-1|= 2.6 ug.mL-1NPASS