| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| MOLT-4 | Homo sapiens | | | = 17.0 nM | | | NPASS |
| MV4-11 | Homo sapiens | | | = 12.03 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | | = 49.0 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 15.0 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 19.0 nM|= 2.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 14.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | | = 50.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 52.0 nM|= 22.0 nM|= 28.0 nM|= 14.0 nM|= 34.0 nM|= 32.0 nM|= 8.3 nM|= 10.3 nM|= 20.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 200.0 nM|= 56.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 20.0 nM|= 43.0 nM|= 18.3 nM|= 21.0 nM|= 20.3 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | = 18.0 nM | | | NPASS |
| Proteinase-activated receptor 2 | Homo sapiens | P55085 | | 23 nM|14 nM|= 23.0 nM|= 14.0 nM | | | BindingDB, NPASS |
| RAW264.7 | Mus musculus | | | = 14.0 nM|= 23.0 nM | | | NPASS |
| SGC-7901 | Homo sapiens | | | = 15.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 9.0 nM|= 10.0 nM|= 6.0 nM|= 7.2 nM | | | NPASS |
| MKN-28 | Homo sapiens | | | = 200.0 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 163.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 50.0 nM | | | NPASS |
| THP-1 | Homo sapiens | | | = 7.04 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 49.0 nM|= 33.0 nM | | | NPASS |
| dCTP pyrophosphatase 1 | Homo sapiens | Q9H773 | | 30900 nM|= 30900.0 nM | | 1.68e+5 nM | BindingDB, NPASS |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 40 nM | | | BindingDB |
| MEF | Mus musculus | | | = 9200.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 50.0 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 10.0 nM | | | NPASS |
| MDCK | Canis lupus familiaris | | | = 1200.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 0.0013 ug.mL-1|= 59.0 nM|= 19.0 nM|= 17.5 nM|= 30.0 nM | | | NPASS |
| BGC-823 | Homo sapiens | | | = 2.0 nM | | | NPASS |
| BJ | Homo sapiens | | < 104.0 nM | | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 20.0 nM | | | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 40.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 10.0 nM|= 4.7 nM|= 3.0 nM|= 46.0 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 29.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 0.0001 ug.mL-1|= 2.1 nM|= 47.0 nM | | | NPASS |
| HUVEC | Homo sapiens | | | = 44.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 24.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 47.0 nM|= 87.0 nM|= 43.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 43.3 nM|= 14.0 nM|= 33.0 nM|= 468.0 nM | | | NPASS |
| Hepatocyte | | | | = 37.7 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 140.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 43.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 21.0 nM|= 16.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 9.7 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 19.0 nM|= 22.0 nM | | | NPASS |
| HaCaT | Homo sapiens | | | = 27.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 24.0 nM|= 51.0 nM | | | NPASS |