| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | | = 26.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 47.0 nM|< 20.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 600.0 nM|= 20.0 nM|= 25.0 nM|= 12.0 nM | | | NPASS |
| RKO | Homo sapiens | | | = 15.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 17.0 nM | | | NPASS |
| SGC-7901 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 8.0 nM | | | NPASS |
| SW1990 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 31.0 nM | | | NPASS |
| NCI-N87 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| Raji | Homo sapiens | | | = 4.0 nM | | | NPASS |
| Mus musculus | Mus musculus | | = 0.9 mg kg-1 | | | | NPASS |
| DU-145 | Homo sapiens | | | = 10.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 30.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| AGS | Homo sapiens | | | < 20.0 nM | | | NPASS |
| ASPC1 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| CFPAC-1 | Homo sapiens | | | < 20.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 0.0035 ug.mL-1|= 53.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | < 0.00046 ug.mL-1|= 8.4 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 4.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 10.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 30.0 nM | | | NPASS |
| HGC-27 | Homo sapiens | | | < 20.0 nM | | | NPASS |