| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Vitamin D3 receptor | Homo sapiens | P11473 | >150000 nM | >50000 nM|>150000 nM | | | BindingDB |
| Vitamin D receptor | Homo sapiens | P11473 | > 150000.0 nM | > 150000.0 nM|> 50000.0 nM | | | NPASS |
| Steroid Delta-isomerase | Pseudomonas putida | P07445 | | | 16000 nM|= 16000.0 nM | | BindingDB, NPASS |
| Solute carrier organic anion transporter family member [3-691] | Zebrafish | | | | | 9.94e+3 nM | BindingDB |
| Plasmodium falciparum 3D7 | Plasmodium falciparum 3D7 | | | = 93600.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | > 80000.0 nM | | | NPASS |
| KB 3-1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Ileal bile acid transporter | Homo sapiens | Q12908 | | | | = 6300.0 nM | NPASS |
| HuTu80 | Homo sapiens | | | = 82900.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | 1250 nM|= 1250.0 nM | | | | BindingDB, NPASS |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | = 50000.0 nM|= 45000.0 nM | | | | NPASS |
| Bile acid receptor | Homo sapiens | Q96RI1 | 45000 nM | | | | BindingDB |
| Ileal sodium/bile acid cotransporter | Homo sapiens | Q12908 | | | | 6300 nM | BindingDB |