| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| SK-MEL-2 | Homo sapiens | | | = 1800.0 nM | | | NPASS |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens | Q9NPD5 | | | | 1430 nM|4550 nM|8290 nM|1030 nM|= 1430.0 nM|= 4550.0 nM|= 8290.0 nM|= 1030.0 nM | BindingDB, NPASS |
| SW626 | Homo sapiens | | | = 3100.0 nM | | | NPASS |
| SW1990 | Homo sapiens | | | = 500.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 810.0 nM | | | NPASS |
| P388 | Mus musculus | | | = 21900.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 3800.0 nM|> 23000.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 4560.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 22400.0 nM|= 1030.0 nM|= 879.0 nM | | | NPASS |
| Lu1 | Homo sapiens | | | = 1200.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 1700.0 nM | | | NPASS |
| KETR3 | Homo sapiens | | | = 447.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 4700.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 500.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 2000.0 nM|= 3800.0 nM | | | NPASS |
| HCT-8 | Homo sapiens | | | = 560.0 nM|= 351.0 nM|= 340.0 nM | | | NPASS |
| Col2 | Homo sapiens | | | = 2800.0 nM | | | NPASS |
| Capan-2 | Homo sapiens | | | = 50.0 nM | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 230.0 nM|= 930.0 nM|= 810.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 20700.0 nM|= 530.0 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 700.0 nM | | | NPASS |
| BGC-823 | Homo sapiens | | | = 268.0 nM|= 1080.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 4200.0 nM|= 700.0 nM|= 454.0 nM|= 810.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 4460.0 nM|= 581.0 nM|= 870.0 nM | | | NPASS |