| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Tankyrase-2 | Homo sapiens | Q9H2K2 | | = 457.09 nM|= 450.0 nM | | | NPASS |
| Tankyrase-1 | Homo sapiens | O95271 | | = 562.34 nM|= 560.0 nM | | | NPASS |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens | Q9H2K2 | | 450 nM | | | BindingDB |
| Poly [ADP-ribose] polymerase-1 | Homo sapiens | P09874 | | > 100000.0 nM | | | NPASS |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens | P09874 | | >100000 nM | | | BindingDB |
| Aromatase | Homo sapiens | P11511 | | 1.00e+5 nM | | | BindingDB |
| Acetylcholinesterase | Rattus norvegicus | P37136 | | 35 nM|= 35.0 nM | | | BindingDB, NPASS |
| Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens | O95271 | | 560 nM | | | BindingDB |