IMPPAT Phytochemical information: 
Tetrandrine

Tetrandrine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
PC-3Homo sapiens= 7870.0 nM|= 5860.0 nMNPASS
PLC-PRF-5Homo sapiens= 18460.0 nMNPASS
Plasmodium falciparumPlasmodium falciparum= 288.0 nM|= 257.0 nMNPASS
Replicase polyprotein 1ab2019-nCoVP0DTD13000 nMBindingDB
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2= 1100.0 nM= 3000.0 nM|= 11660.0 nM|> 50100.0 nM|> 50118.72 nM|= 284.0 nMNPASS
Small conductance calcium-activated potassium channel protein 3Homo sapiensQ9UGI6= 461.0 nMNPASS
NON-PROTEIN TARGET= 1480.0 nMNPASS
U-937Homo sapiens> 50000.0 nMNPASS
Voltage-dependent L-type calcium channel subunit alpha-1SRattus norvegicusQ02485741 nMBindingDB
Voltage-gated L-type calcium channelRattus norvegicusP27732= 741.31 nMNPASS
Small conductance calcium-activated potassium channel protein 2Homo sapiensQ9H2S1= 306.0 nMNPASS
Muscarinic acetylcholine receptorRattus norvegicusP10980= 73.0 nMNPASS
AortaRattus norvegicus= 29512.09 nM|= 13489.63 nMNPASS
MCF7Homo sapiens= 8620.0 nM|= 19580.0 nMNPASS
MDA-MB-231Homo sapiens= 21970.0 nM|= 8940.0 nM|= 18450.0 nMNPASS
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptorRattus norvegicusP15823|P23944|P43140692 nMBindingDB
CCRF-CEMHomo sapiens= 15800.0 nMNPASS
ECa-109 cell lineHomo sapiens= 29.4 nM|= 29.37 nMNPASS
Adrenergic receptor alpha-1Rattus norvegicusP43140= 691.83 nMNPASS
HELHomo sapiens= 16780.0 nM|= 7450.0 nM|= 19740.0 nMNPASS
HepG2Homo sapiens= 6820.0 nMNPASS
K562Homo sapiens= 13810.0 nM|= 11760.0 nM|= 6430.0 nMNPASS
L02Homo sapiens= 44250.0 nMNPASS
Entamoeba histolyticaEoeba histolytica= 25.16 ug.mL-1|= 10.51 ug.mL-1NPASS