
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Histamine H1 receptor | Homo sapiens | P35367 | 1 nM|1.53 nM|1.11 nM|1.6 nM | BindingDB | |||
| Histamine H1 receptor | Rattus norvegicus | P31390 | 5.6 nM | BindingDB | |||
| Bile salt export pump | Homo sapiens | O95342 | 290800 nM | BindingDB | |||
| Histamine H1 receptor | Cavia porcellus | P31389 | 0.31 nM|0.93 nM|0.69 nM | BindingDB |