| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Multidrug resistance-associated protein 1 | Homo sapiens | P33527 | | 38320 nM|= 38320.0 nM | | | BindingDB, NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >306000 nM | | | BindingDB |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 25.27 nM|= 32.43 nM|= 204.61 nM|= 550.0 nM|= 2660.5 nM|= 79.31 nM|= 230.0 nM|= 187.84 nM|= 43.93 nM|= 1.59 nM|= 571.36 nM|= 118.02 nM|= 1009.5 nM|= 969.58 nM|= 100.0 nM|= 223.72 nM|= 115.02 nM|= 75.77 nM|= 2810.0 nM|= 3220.21 nM|= 280.0 nM|= 300.0 nM|= 100.25 nM|= 109.0 nM|= 25.0 nM|= 700.0 nM|= 304.03 nM|= 21.42 nM|= 1310.0 nM|= 1420.0 nM | | = 20.0 nM | NPASS |
| NON-PROTEIN TARGET | | | | = 6.99 nM|= 100.0 nM|= 4.94 nM|= 70.0 nM|= 24.53 nM|= 6.38 nM|= 0.62 nM|= 20.45 nM|= 9.29 nM|= 3.85 nM|= 6.14 nM|= 0.63 nM|= 22.75 nM|= 9.77 nM|= 110.0 nM|= 22.11 nM|= 6.02 nM|= 6.81 nM|= 1.21 nM|= 9.33 nM|= 150.0 nM|= 140.0 nM|= 120.0 nM|= 0.59 nM|= 130.0 nM|= 9.15 nM|= 5.63 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | | = 6740.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| A549 | Homo sapiens | | | = 7590.0 nM | | | NPASS |
| Hep 3B2 | Homo sapiens | | | = 6710.0 nM | | | NPASS |
| B16 | Mus musculus | | | = 5900.0 nM | | | NPASS |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | 76 nM|230 nM|571 nM|3220 nM|79 nM|304 nM|1310 nM|2661 nM|1010 nM|109 nM|25 nM|1420 nM|280 nM|32 nM|100 nM|21 nM|550 nM|224 nM|115 nM|118 nM|300 nM|700 nM|44 nM|188 nM|205 nM|1.6 nM|2810 nM|970 nM | | 20 nM | BindingDB |
| A-375 | Homo sapiens | | | = 7200.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 7420.0 nM | | | NPASS |