IMPPAT Phytochemical information: 
Forskolin

Forskolin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Nuclear receptor subfamily 1 group I member 2Homo sapiensO7546914100 nM|7900 nM|2700 nM|700 nMBindingDB
n.a.> 67547.0 nMNPASS
Steroidogenic factor 1Homo sapiensQ13285>67547 nMBindingDB
Solute carrier family 2, facilitated glucose transporter member 1Homo sapiensP111665000 nMBindingDB
Sodium channel protein type 1/2/3 subunit alphaHomo sapiensP35498|Q99250|Q9NY4660000 nMBindingDB
Sodium channel alpha subunits; brain (Types I, II, III)Homo sapiensQ9NY46= 60000.0 nMNPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nMNPASS
SARS coronavirusSARS coronavirus= 7500.0 nMNPASS
Relaxin receptor 1Homo sapiensQ9HBX947 nM|= 47.0 nMBindingDB, NPASS
Rattus norvegicusRattus norvegicus= 240.0 nMNPASS
Pregnane X receptorHomo sapiensO75469= 700.0 nM|= 7900.0 nM|= 2700.0 nM|= 14100.0 nMNPASS
P-glycoprotein 1Homo sapiensP08183= 188200.0 nM|= 80200.0 nMNPASS
Nuclear receptor subfamily 1 group I member 2Rattus norvegicusQ9R1A77100 nM|= 7100.0 nMBindingDB, NPASS
MCF7Homo sapiens= 63300.0 nMNPASS
Adenylate cyclase type IIRattus norvegicusP26769< 2000.0 nMNPASS
Luciferin 4-monooxygenasePhotinus pyralisP08659> 112219.0 nMNPASS
ATP-dependent translocase ABCB1Homo sapiensP08183188200 nM|80200 nMBindingDB
Adenylate cyclase type 1Bos taurusP1975429 nMBindingDB
Adenylate cyclase type 1Homo sapiensQ08828500 nM41 nMBindingDB
Adenylate cyclase type 8Homo sapiensP4014594 nMBindingDB
Nuclear receptor subfamily 0 group B member 1Homo sapiensP518431729 nM|= 1729.0 nMBindingDB, NPASS
Adenylate cyclase type IBos taurusP19754= 29.0 nMNPASS
BT-474Homo sapiens> 100000.0 nMNPASS
Brain adenylate cyclase 1Homo sapiensQ08828= 500.0 nM= 41.0 nM|< 150.0 nMNPASS
Cavia porcellusCavia porcellus= 0.02 ug.mL-1NPASS
Glucose transporterHomo sapiensP11166= 5000.0 nMNPASS
Homo sapiensHomo sapiens= 240.0 nMNPASS
Adenylate cyclase type VIIIHomo sapiensP40145= 93.7 nMNPASS