| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Metabotropic glutamate receptor 8 | Mus musculus | P47743 | >100000 nM | | | | BindingDB |
| Metabotropic glutamate receptor 7 | Rattus norvegicus | P35400 | >1000000 nM | | | | BindingDB |
| Metabotropic glutamate receptor 7 | Homo sapiens | Q14831 | >1000000 nM | | | | BindingDB |
| Metabotropic glutamate receptor 3 | Homo sapiens | Q14832 | | | | 250 nM|6000 nM|>10000 nM|40000 nM | BindingDB |
| Metabotropic glutamate receptor 6 | Rattus norvegicus | P35349 | 1000000 nM | | | | BindingDB |
| Metabotropic glutamate receptor 6 | Homo sapiens | O15303 | | | | >10000 nM|1000000 nM | BindingDB |
| Metabotropic glutamate receptor 5 | Rattus norvegicus | P31424 | 300 nM|200 nM | | | >10000 nM | BindingDB |
| Metabotropic glutamate receptor 5 | Homo sapiens | P41594 | 150 nM|630 nM | | | 30 nM|29 nM|>10000 nM|55 nM | BindingDB |
| Metabotropic glutamate receptor 4 | Rattus norvegicus | P31423 | >100000 nM | | | >10000 nM | BindingDB |
| Metabotropic glutamate receptor 4 | Homo sapiens | Q14833 | >500000 nM | | | >10000 nM|1000000 nM|112000 nM | BindingDB |
| Metabotropic glutamate receptor 3 | Rattus norvegicus | P31422 | 40000 nM | | | | BindingDB |
| Metabotropic glutamate receptor 2 | Homo sapiens | Q14416 | >500000 nM|>1000000 nM | | | 420 nM|>10000 nM|178 nM|>1000000 nM|113000 nM | BindingDB |
| Glutamate metabotropic receptor 1 | Sus scrofa | | | | | 260 nM | BindingDB |
| Metabotropic glutamate receptor 1 | Homo sapiens | Q13255 | 200 nM | | | 30 nM|200 nM|10 nM|1100 nM | BindingDB |
| Metabotropic glutamate receptor 1 | Rattus norvegicus | P23385 | 750 nM|16400 nM|200 nM|2500 nM | | | 0.03 nM|>10000 nM|10 nM | BindingDB |
| Cystine/glutamate transporter | Homo sapiens | Q9UPY5 | | 5000 nM | | | BindingDB |
| Glutamate metabotropic receptor 5 | Cavia porcellus | | | | | 22 nM|47 nM | BindingDB |
| Glutamate receptor | Oryctolagus cuniculus | | | | | 16.46 nM | BindingDB |
| Glutamate receptor 3 | Rattus norvegicus | P19492 | | | | >10000 nM | BindingDB |
| Glutamate carboxypeptidase 2 [44-750] | Homo sapiens | Q04609 | | 9500 nM | | | BindingDB |
| Glutamate receptor ionotropic, kainate 1 | Rattus norvegicus | P22756 | | | | 171 nM | BindingDB |
| Glutamate receptor ionotropic, kainate 2 | Rattus norvegicus | P42260 | | | | 134 nM | BindingDB |
| Glutamate receptor ionotropic, kainate 3 | Rattus norvegicus | P42264 | | | | 1670 nM | BindingDB |
| Glutamate receptor ionotropic, kainate 4 | Homo sapiens | Q16099 | | | | 6.43 nM | BindingDB |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus | P35439 | | | | >10000 nM|260 nM | BindingDB |