| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Peroxisome proliferator-activated receptor delta | Homo sapiens | Q03181 | > 100000.0 nM | > 100000.0 nM | | | NPASS |
| Vitamin D receptor | Homo sapiens | P11473 | > 100000.0 nM | = 2000.0 nM | | | NPASS |
| Thyroid hormone receptor | Homo sapiens | P10828 | > 100000.0 nM | > 100000.0 nM | | | NPASS |
| Retinoid X receptor alpha | Homo sapiens | P19793 | > 100000.0 nM | = 33000.0 nM | | | NPASS |
| Retinoic acid receptor | Homo sapiens | | > 100000.0 nM | > 100000.0 nM | | | NPASS |
| Progesterone receptor | Homo sapiens | P06401 | = 1900.0 nM | = 1200.0 nM|> 100000.0 nM | | = 201.0 nM | NPASS |
| Pregnane X receptor | Homo sapiens | O75469 | = 2500.0 nM | = 2.4 nM|> 100000.0 nM | | | NPASS |
| Peroxisome proliferator-activated receptor gamma | Homo sapiens | P37231 | > 100000.0 nM | = 27000.0 nM | | | NPASS |
| Peroxisome proliferator-activated receptor alpha | Homo sapiens | Q07869 | > 100000.0 nM | = 20000.0 nM | | | NPASS |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | > 100000.0 nM|= 220.0 nM|= 310.0 nM|= 420.0 nM|= 130.0 nM|= 400.0 nM|= 380.0 nM | = 100000.0 nM|= 4100.0 nM|= 44000.0 nM|= 41000.0 nM|= 25000.0 nM|= 13000.0 nM|= 6000.0 nM|= 10000.0 nM|= 4200.0 nM | | > 5000.0 nM | NPASS |
| Mineralocorticoid receptor | Homo sapiens | P08235 | > 100000.0 nM | = 1000.0 nM|= 320.0 nM | | = 39.0 nM | NPASS |
| LXR-beta | Homo sapiens | P55055 | = 3600.0 nM | > 100000.0 nM | | | NPASS |
| LXR-alpha | Homo sapiens | Q13133 | > 100000.0 nM | > 100000.0 nM | | | NPASS |
| Glucocorticoid receptor | Homo sapiens | P04150 | > 100000.0 nM | = 1740.0 nM|> 100000.0 nM | | = 224.0 nM | NPASS |
| Estrogen receptor alpha | Homo sapiens | P03372 | > 100000.0 nM | = 62000.0 nM | | | NPASS |
| Estrogen receptor | Homo sapiens | P03372 | | > 5000.0 nM | | > 5000.0 nM | NPASS |
| Androgen Receptor | Homo sapiens | P10275 | | = 220.0 nM | | = 240.0 nM | NPASS |
| PANC-1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |