IMPPAT Phytochemical information: 
Bicuculline

Bicuculline
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Sigma non-opioid intracellular receptor 1Rattus norvegicusQ9R0C9>10000 nMBindingDB
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nMNPASS
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicusP235743800 nMBindingDB
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiensQ16445>10000 nMBindingDB
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiensP316444466.83 nMBindingDB
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiensP349032818.38 nMBindingDB
Histamine H1 receptorHomo sapiensP35367>10000 nMBindingDB
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiensP14867>10000 nM|4570.88 nMBindingDB
Gamma-aminobutyric acid (GABA) B receptor 1Rattus norvegicus6200 nMBindingDB
GABA-A receptor; anion channelHomo sapiensQ16445= 15000.0 nM|= 44000.0 nM|= 6200.0 nMNPASS
GABA receptor gamma-1 subunitRattus norvegicusP23574= 3800.0 nMNPASS
D(2) dopamine receptorRattus norvegicusP61169>10000 nMBindingDB
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiensP478691862.08 nMBindingDB