| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Liver carboxylesterase 1 | Oryctolagus cuniculus | P12337 | | | | >100000 nM | BindingDB |
| MDA-MB-231 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| MRC5 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Meloidogyne incognita | Meloidogyne incognita | | > 250.0 ug.mL-1 | | | | NPASS |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 40000.0 nM|= 56234.13 nM|= 31800.0 nM|= 22540.0 nM|> 500000.0 nM|= 8430.0 nM | | = 15000.0 nM|= 8380.0 nM|= 16000.0 nM|= 5940.0 nM|= 16.0 10^3nM | NPASS |
| Monoamine oxidase B | Homo sapiens | P27338 | | = 18750.0 nM|= 18754.0 nM|= 7943.28 nM|= 12400.0 nM|= 21070.0 nM|= 34390.0 nM|= 12070.0 nM|= 368400.0 nM|= 3900.0 nM | | = 3000.0 nM|= 5340.0 nM|= 33.0 nM|= 2000.0 nM|= 5200.0 nM|= 4.0 10^3nM | NPASS |
| NON-PROTEIN TARGET | | | | > 50000.0 nM | | | NPASS |
| Protein-glutamine gamma-glutamyltransferase 2 | Homo sapiens | P21980 | | >250000 nM | | | BindingDB |
| Protein-glutamine gamma-glutamyltransferase | Homo sapiens | P21980 | | > 250000.0 nM | | | NPASS |
| SK-N-SH | Homo sapiens | | | = 9840.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 565000.0 nM|= 562341.33 nM | | | NPASS |
| Secreted chorismate mutase | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) | P9WIB9 | | 1.08e+3 nM | | | BindingDB |
| Transthyretin | Homo sapiens | P02766 | | >50000 nM|> 50000.0 nM | | | BindingDB, NPASS |
| Liver carboxylesterase 1 | Homo sapiens | P23141 | | | | >100000 nM | BindingDB |
| Plasmodium falciparum | Plasmodium falciparum | | | > 100000.0 nM | | | NPASS |
| K562 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | | | >100000 nM|> 100000.0 nM | BindingDB, NPASS |
| HepG2 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 13500.0 nM | | | NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | > 1000000.0 nM | | | NPASS |
| Acyl coenzyme A:cholesterol acyltransferase | Homo sapiens | P23141 | | | | > 100000.0 nM | NPASS |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | 56234 nM|40000 nM|31800 nM|>500000 nM | | 15000 nM|8380 nM|16000 nM | BindingDB |
| Jurkat | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Amine oxidase [flavin-containing] B | Homo sapiens | P27338 | | 7943 nM|18750 nM|34390 nM|12400 nM|18754 nM|21070 nM|368400 nM | | 3000 nM|5340 nM|33 nM|2000 nM|4000 nM | BindingDB |
| Amine oxidase [flavin-containing] B [I199F] | Homo sapiens | P27338 | | | | 500 nM | BindingDB |
| Amine oxidase [flavin-containing] B | Bos taurus | P56560 | | | | 6000 nM | BindingDB |
| Caspase-3 | Homo sapiens | P42574 | | > 100000.0 nM | | | NPASS |
| Cholinesterase | Equus caballus | P81908 | | > 1000000.0 nM | | | NPASS |
| Cholinesterase | Homo sapiens | P06276 | | | | >100000 nM | BindingDB |
| Coagulation factor XII | Homo sapiens | P00748 | | | | >100000 nM | BindingDB |
| Cruzipain | Trypanosoma cruzi | P25779 | | >> 10000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Butyrylcholinesterase | Homo sapiens | P06276 | | | | > 100000.0 nM | NPASS |