| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Plasmodium falciparum | Plasmodium falciparum | | | = 17000.0 nM | | | NPASS |
| NAD-dependent deacetylase sirtuin 2 | Homo sapiens | Q8IXJ6 | | = 9200.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 3230.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 3230.0 nM | | | NPASS |
| Neutral sphingomyelinase | Homo sapiens | O60906 | | = 46.5 ug.mL-1 | | | NPASS |
| Nuclear factor NF-kappa-B p105 subunit | Homo sapiens | P19838 | | > 20000.0 nM | | | NPASS |
| Nuclear factor NF-kappa-B p65 subunit | Homo sapiens | Q04206 | | = 15900.0 nM|> 10000.0 nM | | | NPASS |
| Phosphodiesterase 4D | Homo sapiens | Q08499 | | = 1310.0 nM | | | NPASS |
| Phosphoglycerate mutase 1 | Homo sapiens | P18669 | | = 7200.0 nM | | | NPASS |
| Plasmodium falciparum (isolate FcB1 / Columbia) | Plasmodium falciparum FcB1/Columbia | | | = 2.9 ug.mL-1 | | | NPASS |
| Stimulator of interferon genes protein | Homo sapiens | Q86WV6 | | = 137000.0 nM | = 157000.0 nM|= 137000.0 nM | | NPASS |
| SK-HEP1 | Homo sapiens | | | = 19600.0 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 2970.0 nM | | | NPASS |
| Sialidase | Clostridium perfringens | P10481 | | = 12200.0 nM | | = 5800.0 nM | NPASS |
| Solute carrier family 22 member 12 | Homo sapiens | Q96S37 | | = 58950.0 nM | | | NPASS |
| Sphingomyelin phosphodiesterase | Bos taurus | Q0VD19 | | = 14100.0 nM | | | NPASS |
| Sphingomyelin phosphodiesterase | Homo sapiens | P17405 | | = 5.15 ug.mL-1|= 24740.0 nM|= 14100.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 3040.0 nM|= 12750.0 nM | | | NPASS |
| Stimulator of interferon genes protein | Mus musculus | Q3TBT3 | | | = 137000.0 nM | | NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | = 7900.0 nM | | | | NPASS |
| WRL68 | Homo sapiens | | | = 158000.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | = 5500.0 nM | | = 3200.0 nM | NPASS |
| MCF7 | Homo sapiens | | | = 3.5 ug.mL-1|> 10000.0 nM|= 9950.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | = 8900.0 nM | | | | NPASS |
| Lysine-specific histone demethylase 1 | Homo sapiens | O60341 | | = 2810.0 nM | | | NPASS |
| 7,8-dihydro-8-oxoguanine triphosphatase | Homo sapiens | P36639 | | = 470.0 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 7200.0 nM | | | NPASS |
| ASPC1 | Homo sapiens | | | = 4020.0 nM | | | NPASS |
| Alpha glucosidase | Homo sapiens | | | = 5700.0 nM | | = 7300.0 nM | NPASS |
| Arachidonate 12-lipoxygenase | Homo sapiens | P18054 | | = 580.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase | Homo sapiens | P16050 | | = 3100.0 nM|> 50000.0 nM | | | NPASS |
| Cyclic GMP-AMP synthase | Homo sapiens | Q8N884 | | = 4.0 nM | | | NPASS |
| Cytochrome P450 19A1 | Homo sapiens | P11511 | | = 20700.0 nM | | | NPASS |
| DLD-1 | Homo sapiens | | | = 7500.0 nM | | | NPASS |
| Daoy | Homo sapiens | | | = 1900.0 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 2700.0 nM | | | NPASS |
| Fatty acid synthase | Homo sapiens | P49327 | | = 5540.0 nM | | | NPASS |
| Dengue virus 2 | Dengue virus 2 | | = 10000.0 nM | | | | NPASS |
| Leishmania infantum | Leishmaitum | | = 8000.0 nM | | | | NPASS |
| KB | Homo sapiens | | | = 14140.0 nM|> 10000.0 nM | | | NPASS |
| Isocitrate dehydrogenase [NADP] cytoplasmic | Homo sapiens | O75874 | | | | = 2850.0 nM | NPASS |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens | Q96L34 | | = 1770.0 nM | | | NPASS |
| HeLa S3 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 11950.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 200.0 nM|> 10000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 6800.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 10000.0 nM|= 8550.0 nM | | | NPASS |