| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| SK-MEL-28 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 1.0 ug.mL-1 | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 1.0 ug.mL-1|>= 1.0 ug.mL-1 | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | > 12.5 ug.mL-1 | | | NPASS |
| Plasmodium falciparum (isolate K1 / Thailand) | Plasmodium falciparum K1 | | | = 7.6 ug.mL-1 | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 1.0 ug.mL-1|= 260.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | > 10000.0 nM | | | NPASS |
| MRC5 | Homo sapiens | | | = 18.11 ug.mL-1 | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | | | 11000 nM|= 11000.0 nM|= 10000.0 nM | BindingDB, NPASS |
| B16-F10 | Mus musculus | | | > 10000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 10000.0 nM | | | NPASS |