| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Multidrug resistance-associated protein 4 | Homo sapiens | O15439 | | > 133000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 78000.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 1520.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| KB | Homo sapiens | | | = 0.513 ug.mL-1 | | | NPASS |
| L5178Y | Mus musculus | | | = 300.0 nM | | | NPASS |
| L929 | Mus musculus | | | = 16.1 nM | | | NPASS |
| Mitochondrial complex I; NADH oxidoreductase | Bos taurus | P52505 | | = 5.1 nM | | | NPASS |
| NADH-ubiquinone oxidoreductase chain 4 | Homo sapiens | P03905 | | 3.5 nM|= 3.5 nM | | | BindingDB, NPASS |
| HT-29 | Homo sapiens | | | = 300.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 500.0 nM | = 0.595 ug.mL-1|= 700.0 nM|= 74100.0 nM | | | NPASS |
| Pancreatic triacylglycerol lipase | Sus scrofa | P00591 | | >500000 nM|> 500000.0 nM|= 31.2 ug.mL-1 | | | BindingDB, NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | > 10000.0 nM|= 10000.0 nM|= 12589.25 nM | | | NPASS |
| Raji | Homo sapiens | | | = 1100.0 nM|= 4200.0 nM | | | NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >507000 nM | | | BindingDB |
| Serotonin 6 (5-HT6) receptor | Homo sapiens | P50406 | | = 870.0 nM | | = 404.0 nM | NPASS |
| U-937 | Homo sapiens | | | = 13000.0 nM|= 200.0 nM|= 70.0 nM | | | NPASS |
| NADH-ubiquinone oxidoreductase chain 1 | Bos taurus | P03887 | | 4.4 nM|= 4.4 nM|= 25.7 nM | | | BindingDB, NPASS |
| HCT-116 | Homo sapiens | | | = 0.045 ug | | | NPASS |
| MCF7 | Homo sapiens | | | = 0.008 ug.mL-1 | | | NPASS |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Plasmodium falciparum | | | >10000 nM | | | BindingDB |
| A549 | Homo sapiens | | | = 0.04 ug.mL-1|= 0.901 ug.mL-1 | | | NPASS |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | >133000 nM | | | BindingDB |
| Acyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial | Bos taurus | P25708|P52505 | | 5.1 nM | | | BindingDB |
| Bile salt export pump | Homo sapiens | O95342 | | 8000 nM|= 8000.0 nM | | | BindingDB, NPASS |
| Caenorhabditis elegans | Caenorhabditis elegans | | = 2000.0 nM | | | | NPASS |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens | Q92887 | | > 133000.0 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 2 | Homo sapiens | O15438 | | > 133000.0 nM | | | NPASS |
| Drosophila | Drosophila | | = 10000.0 nM | | | | NPASS |
| Cavia porcellus | Cavia porcellus | | | = 0.0155 ug.mL-1 | | | NPASS |
| Cytochrome P450 2C19 | Homo sapiens | P33261 | | = 3648.6 nM | | | NPASS |
| Cytochrome b-245 light chain | Bos taurus | O46521 | | = 0.17 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 0.465 ug.mL-1 | | | NPASS |
| Dihydroorotate dehydrogenase | Plasmodium falciparum | Q54A96 | | > 10000.0 nM | | | NPASS |
| Dihydroorotate dehydrogenase | Saccharomyces cerevisiae S288c | P28272 | | > 10000.0 nM | | | NPASS |
| Dihydroorotate dehydrogenase (fumarate) | Saccharomyces cerevisiae (strain ATCC 204508 / S288c) | P28272 | | >10000 nM | | | BindingDB |
| A2780 | Homo sapiens | | | = 0.7 ug.mL-1 | | | NPASS |
| 697 | Homo sapiens | | | = 300.0 nM | | | NPASS |