| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Multidrug resistance-associated protein 1 | Homo sapiens | P33527 | | 50000 nM|= 50000.0 nM | | | BindingDB, NPASS |
| NCI-H157 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| NCI-H1792 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| M14 | Homo sapiens | | | = 380.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 1.43 ug.mL-1|= 1.69 ug.mL-1|= 28000.0 nM|> 50000.0 nM|= 10460.0 nM|= 6530.0 nM|= 390.0 nM|> 100000.0 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 16000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 73300.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | = 600.0 nM | | | | NPASS |
| NCI-H522 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| L929 | Mus musculus | | | > 100000.0 nM | | | NPASS |
| 2008 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| HOP-62 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 69720.0 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 82250.0 nM|= 57540.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 390.0 nM|= 900.0 nM|= 570.0 nM|= 540.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 46370.0 nM | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 390 nM|900 nM|570 nM|540 nM | | | BindingDB |
| HCT-15 | Homo sapiens | | | = 68110.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | = 141870.0 nM | | | NPASS |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | 16000 nM | | | BindingDB |