IMPPAT Phytochemical information: 
Retusin

Retusin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Multidrug resistance-associated protein 1Homo sapiensP3352750000 nM|= 50000.0 nMBindingDB, NPASS
NCI-H157Homo sapiens> 50000.0 nMNPASS
MCF7Homo sapiens> 100000.0 nMNPASS
NCI-H1792Homo sapiens> 50000.0 nMNPASS
M14Homo sapiens= 380.0 nMNPASS
NON-PROTEIN TARGET= 1.43 ug.mL-1|= 1.69 ug.mL-1|= 28000.0 nM|> 50000.0 nM|= 10460.0 nM|= 6530.0 nM|= 390.0 nM|> 100000.0 nMNPASS
P-glycoprotein 1Homo sapiensP08183= 16000.0 nMNPASS
Plasmodium falciparumPlasmodium falciparum= 73300.0 nMNPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2= 600.0 nMNPASS
NCI-H522Homo sapiens> 50000.0 nMNPASS
L929Mus musculus> 100000.0 nMNPASS
2008Homo sapiens> 100000.0 nMNPASS
HOP-62Homo sapiens> 50000.0 nMNPASS
A-375Homo sapiens= 69720.0 nMNPASS
A-431Homo sapiens= 82250.0 nM|= 57540.0 nMNPASS
A549Homo sapiens> 50000.0 nMNPASS
ATP-binding cassette sub-family G member 2Homo sapiensQ9UNQ0= 390.0 nM|= 900.0 nM|= 570.0 nM|= 540.0 nMNPASS
HeLaHomo sapiens= 46370.0 nMNPASS
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiensQ9UNQ0390 nM|900 nM|570 nM|540 nMBindingDB
HCT-15Homo sapiens= 68110.0 nMNPASS
HEK293Homo sapiens= 141870.0 nMNPASS
ATP-dependent translocase ABCB1Homo sapiensP0818316000 nMBindingDB