IMPPAT Phytochemical information: 
Cryptolepine

Cryptolepine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Plasmodium falciparumPlasmodium falciparum= 2300.0 nM|= 2000.0 nM|= 0.027 ug.mL-1|= 0.041 ug.mL-1|= 230.0 nM|= 755.0 nM|= 259.0 nM|= 222.0 nM|= 440.0 nM|= 19.65 nMNPASS
Telomerase reverse transcriptaseHomo sapiensO147469400 nM|= 9400.0 nMBindingDB, NPASS
Plasmodium falciparum (isolate K1 / Thailand)Plasmodium falciparum K1= 0.033 ug.mL-1NPASS
VeroChlorocebus aethiops= 3.2 ug.mL-1NPASS
MRC5Homo sapiens= 1500.0 nMNPASS
Trypanosoma bruceiTrypanosoma brucei= 300.0 nM= 3000.0 nMNPASS
MCF7Homo sapiens= 630.0 nMNPASS
Nucleic Acid= 65700.0 nMNPASS
Histidine-rich protein PFHRP-IIPlasmodium falciparumP052271720000000 nMBindingDB
Leishmania donovaniLeishmadonovani= 1600.0 nM= 1600.0 nMNPASS
Filobasidiella neoformansCryptococcus neoformans= 12.5 ug.mL-1|= 43251.38 nM|= 43300.0 nMNPASS
Cathepsin B-like cysteine proteaseTrypanosoma brucei64000 nMBindingDB
Candida albicansCandida albicans= 20.0 ug.mL-1|= 250.0 ug.mL-1NPASS
Calf thymus DNABos taurus= 330.0 nM|= 240.0 nMNPASS
A549Homo sapiens= 1050.0 nMNPASS