| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| K562 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | > 49019.6 nM | | | | NPASS |
| Raji | Homo sapiens | | > 22554.3 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | > 36630.0 nM|> 43478.3 nM | | | | NPASS |
| HepG2 | Homo sapiens | | > 52083.3 nM | | | | NPASS |
| Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | > 36630.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Endothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha | Homo sapiens | Q16665|Q99814 | | >50000 nM | | | BindingDB |
| BJ | Homo sapiens | | > 36630.0 nM | | | | NPASS |
| AGS | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 10000.0 nM | | | NPASS |