| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| DU-145 | Homo sapiens | | | = 26000.0 nM | | | NPASS |
| LIM domain kinase 1 | Homo sapiens | P53667 | | 800 nM|= 800.0 nM | | | BindingDB, NPASS |
| LIM domain kinase 2 | Homo sapiens | P53671 | | 1530 nM|= 1530.0 nM|= 1500.0 nM | | | BindingDB, NPASS |
| MCF7 | Homo sapiens | | | = 11000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 25000.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 39510.0 nM | | | NPASS |
| Tyrosine-protein kinase LCK | Homo sapiens | P06239 | | = 17.0 nM|= 620.0 nM | | | NPASS |
| Tyrosine-protein kinase Lck | Homo sapiens | P06239 | | 620 nM|17 nM | | | BindingDB |