IMPPAT Phytochemical information: 
Wedelolactone

Wedelolactone
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Telomere resolvase resTBorrelia burgdorferi (strain ATCC 35210 / B31 / CIP 102532 / DSM4680)O50979= 8670.0 nMNPASS
Solute carrier family 22 member 2Homo sapiensO15244= 17330.0 nMNPASS
Solute carrier family 22 member 1Homo sapiensO15245= 38400.0 nMNPASS
Rattus norvegicusRattus norvegicus= 700.0 nMNPASS
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiensP099172500 nMBindingDB
Polycomb protein EEDHomo sapiensO755302820 nM|2800 nM|= 2800.0 nM|= 2820.0 nMBindingDB, NPASS
OVCAR-3Homo sapiens= 10640.0 nMNPASS
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiensO14920>10000 nMBindingDB
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiensO15111>10000 nMBindingDB
Telomere resolvase ResTBorreliella burgdorferi (strain ATCC 35210 / DSM 4680 / CIP 102532 / B31)O509798670 nMBindingDB
Inhibitor of nuclear factor kappa B kinase alpha subunitHomo sapiensO15111> 10000.0 nMNPASS
Inhibitor of nuclear factor kappa B kinase beta subunitHomo sapiensO14920> 10000.0 nMNPASS
Arachidonate 5-lipoxygenaseHomo sapiensP09917= 2500.0 nMNPASS
Arachidonate 5-lipoxygenaseSus scrofa2500000 nMBindingDB
Arachidonate 5-lipoxygenaseSus scrofaK7GQZ4= 2500000.0 nMNPASS
Hepatitis C virusHepatitis C virus= 36100.0 nM|= 36000.0 nM|= 34000.0 nMNPASS
GABA-A receptor; anion channelRattus norvegicusQ9ES14= 2000.0 nMNPASS
Carbonyl reductase [NADPH] 1Homo sapiensP161523780 nM|= 3780.0 nM600 nM|= 600.0 nMBindingDB, NPASS
Glucose-6-phosphate 1-dehydrogenaseHomo sapiensP114135180 nM|= 5180.0 nM3640 nM|= 3640.0 nM5793 nM|1191 nM|2537 nM|9941 nM|= 5793.0 nM|= 9941.0 nM|= 2537.0 nM|= 1191.0 nMBindingDB, NPASS
Genome polyproteinHepatitis C virus genotype 1b (isolate BK)P266633.6e+4 nMBindingDB