| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Telomere resolvase resT | Borrelia burgdorferi (strain ATCC 35210 / B31 / CIP 102532 / DSM4680) | O50979 | | = 8670.0 nM | | | NPASS |
| Solute carrier family 22 member 2 | Homo sapiens | O15244 | | = 17330.0 nM | | | NPASS |
| Solute carrier family 22 member 1 | Homo sapiens | O15245 | | = 38400.0 nM | | | NPASS |
| Rattus norvegicus | Rattus norvegicus | | | = 700.0 nM | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 2500 nM | | | BindingDB |
| Polycomb protein EED | Homo sapiens | O75530 | | | 2820 nM|2800 nM|= 2800.0 nM|= 2820.0 nM | | BindingDB, NPASS |
| OVCAR-3 | Homo sapiens | | = 10640.0 nM | | | | NPASS |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens | O14920 | | >10000 nM | | | BindingDB |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens | O15111 | | >10000 nM | | | BindingDB |
| Telomere resolvase ResT | Borreliella burgdorferi (strain ATCC 35210 / DSM 4680 / CIP 102532 / B31) | O50979 | | 8670 nM | | | BindingDB |
| Inhibitor of nuclear factor kappa B kinase alpha subunit | Homo sapiens | O15111 | | > 10000.0 nM | | | NPASS |
| Inhibitor of nuclear factor kappa B kinase beta subunit | Homo sapiens | O14920 | | > 10000.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 2500.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Sus scrofa | | | 2500000 nM | | | BindingDB |
| Arachidonate 5-lipoxygenase | Sus scrofa | K7GQZ4 | | = 2500000.0 nM | | | NPASS |
| Hepatitis C virus | Hepatitis C virus | | | = 36100.0 nM|= 36000.0 nM|= 34000.0 nM | | | NPASS |
| GABA-A receptor; anion channel | Rattus norvegicus | Q9ES14 | | = 2000.0 nM | | | NPASS |
| Carbonyl reductase [NADPH] 1 | Homo sapiens | P16152 | | 3780 nM|= 3780.0 nM | | 600 nM|= 600.0 nM | BindingDB, NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Homo sapiens | P11413 | | 5180 nM|= 5180.0 nM | 3640 nM|= 3640.0 nM | 5793 nM|1191 nM|2537 nM|9941 nM|= 5793.0 nM|= 9941.0 nM|= 2537.0 nM|= 1191.0 nM | BindingDB, NPASS |
| Genome polyprotein | Hepatitis C virus genotype 1b (isolate BK) | P26663 | | 3.6e+4 nM | | | BindingDB |