
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| DNA gyrase | Escherichia coli K-12 | P0AES4 | > 500.0 ug.mL-1 | NPASS | |||
| DNA gyrase A/A/B/B tetramer | Escherichia coli (strain K12) | P0AES4|P0AES6 | >1750000 nM | BindingDB | |||
| H9 | Homo sapiens | = 11.5 ug.mL-1 | NPASS | ||||
| HT-29 | Homo sapiens | > 40000.0 nM | NPASS | ||||
| HepG2 | Homo sapiens | > 40000.0 nM | NPASS | ||||
| NON-PROTEIN TARGET | = 30930.0 nM | NPASS | |||||
| SW480 | Homo sapiens | = 29410.0 nM | NPASS |