IMPPAT: Indian Medicinal Plants, Phytochemistry And Therapeutics
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IMPPAT Phytochemical information:
Febrifugine
Summary
Physicochemical
Drug-likeness
ADME
Descriptors
Bioactivity
Patents
Bioactivity information
Target name
Target organism
UniProt identifier
EC50
IC50
Kd
Ki
Source
Plasmodium falciparum (isolate K1 / Thailand)
Plasmodium falciparum K1
= 2.0 nM
NPASS
Plasmodium falciparum
Plasmodium falciparum
= 0.7 nM|= 1.2 nM|= 0.0014 ug.mL-1|= 0.00142 ug.mL-1|= 0.076 nM|= 200.0 nM
= 1.6 nM|= 1.9 nM|= 0.00076 ug.mL-1|= 2.1 nM|= 3.1 nM|= 5.4 nM
NPASS
FM3A
Mus musculus
= 170.0 nM
NPASS
Hepatocyte
= 169.0 nM
NPASS
L929
Mus musculus
= 0.167 ug.mL-1
NPASS
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