| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| OVCAR-8 | Homo sapiens | | | = 71.5 nM | | | NPASS |
| Signal transducer and activator of transcription 3 [702-738,740-752] | Homo sapiens | P40763 | | 700 nM | | | BindingDB |
| OVCAR-5 | Homo sapiens | | | = 321.0 nM | | | NPASS |
| Replicase polyprotein 1ab | 2019-nCoV | P0DTD1 | | 230 nM | | | BindingDB |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | < 230.0 nM|> 20000.0 nM|> 19952.62 nM | | | NPASS |
| SF-268 | Homo sapiens | | | = 440.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 440.0 nM | | | NPASS |
| Signal transducer and activator of transcription 1-alpha/beta | Homo sapiens | P42224 | | >55700 nM|> 55700.0 nM | | | BindingDB, NPASS |
| Signal transducer and activator of transcription 3 | Homo sapiens | P40763 | | = 700.0 nM | | | NPASS |
| Sodium/potassium-transporting ATPase subunit alpha-2/beta-3 | Human | P50993|P54709 | | | | 28.8 nM | BindingDB |
| Sodium/potassium-transporting ATPase alpha-1 chain | Canis lupus familiaris | P50997 | | = 8.0 nM | | | NPASS |
| Sodium/potassium-transporting ATPase subunit alpha-1 | Canis lupus familiaris | P50997 | | 8 nM | | | BindingDB |
| Sodium/potassium-transporting ATPase subunit alpha-1/beta-1 | Human | P05023|P05026 | | | | 89.0 nM | BindingDB |
| Sodium/potassium-transporting ATPase subunit alpha-2/beta-1 | Human | P05026|P50993 | | | | 29.5 nM | BindingDB |
| Sodium/potassium-transporting ATPase subunit alpha-2/beta-2 | Human | P14415|P50993 | | | | 40.7 nM | BindingDB |
| Solute carrier organic anion transporter family member 4C1 | Homo sapiens | Q6ZQN7 | | 120 nM|= 120.0 nM | | | BindingDB, NPASS |
| TK-10 | Homo sapiens | | | = 3.2 nM | | | NPASS |
| OVCAR-4 | Homo sapiens | | | = 425.6 nM | | | NPASS |
| UACC-62 | Homo sapiens | | | = 33.5 nM | | | NPASS |
| Sodium/potassium-transporting ATPase | Homo sapiens | P54710 | | = 8.0 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 117.1 nM|= 120.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 440.0 nM|= 740.0 nM | | | NPASS |
| NCI/ADR-RES | Homo sapiens | | | = 440.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 440.0 nM | | | NPASS |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | >133000 nM | | | BindingDB |
| Bile salt export pump | Homo sapiens | O95342 | | <10000 nM|31000 nM|< 10000.0 nM|= 31000.0 nM | | | BindingDB, NPASS |
| NON-PROTEIN TARGET | | | | = 440.0 nM|= 410.0 nM|= 100.0 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 2 | Homo sapiens | O15438 | | > 133000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 440.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 4070.0 nM|= 67.6 nM|= 68.0 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens | Q92887 | | > 133000.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 6.4 nM | | | NPASS |
| KURAMOCHI | Homo sapiens | | | = 5911.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 10.2 nM|= 440.0 nM|= 20.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 482.0 nM|= 480.0 nM | | | NPASS |
| MDA-MB-435 | Homo sapiens | | | = 43.3 nM|= 43.0 nM | | | NPASS |
| Monoclonal antibody (mAb) | | | | | = 0.6 nM | = 0.1 nM|= 0.2 nM | NPASS |
| Multidrug resistance-associated protein 4 | Homo sapiens | O15439 | | > 133000.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 440.0 nM|= 357.0 nM | | | NPASS |
| Human herpesvirus 5 | Human herpesvirus 5 | | = 23.3 nM | | | | NPASS |