IMPPAT Phytochemical information: 
Digitoxin

Digitoxin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
OVCAR-8Homo sapiens= 71.5 nMNPASS
Signal transducer and activator of transcription 3 [702-738,740-752]Homo sapiensP40763700 nMBindingDB
OVCAR-5Homo sapiens= 321.0 nMNPASS
Replicase polyprotein 1ab2019-nCoVP0DTD1230 nMBindingDB
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2< 230.0 nM|> 20000.0 nM|> 19952.62 nMNPASS
SF-268Homo sapiens= 440.0 nMNPASS
SK-OV-3Homo sapiens= 440.0 nMNPASS
Signal transducer and activator of transcription 1-alpha/betaHomo sapiensP42224>55700 nM|> 55700.0 nMBindingDB, NPASS
Signal transducer and activator of transcription 3Homo sapiensP40763= 700.0 nMNPASS
Sodium/potassium-transporting ATPase subunit alpha-2/beta-3HumanP50993|P5470928.8 nMBindingDB
Sodium/potassium-transporting ATPase alpha-1 chainCanis lupus familiarisP50997= 8.0 nMNPASS
Sodium/potassium-transporting ATPase subunit alpha-1Canis lupus familiarisP509978 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1HumanP05023|P0502689.0 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1HumanP05026|P5099329.5 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-2/beta-2HumanP14415|P5099340.7 nMBindingDB
Solute carrier organic anion transporter family member 4C1Homo sapiensQ6ZQN7120 nM|= 120.0 nMBindingDB, NPASS
TK-10Homo sapiens= 3.2 nMNPASS
OVCAR-4Homo sapiens= 425.6 nMNPASS
UACC-62Homo sapiens= 33.5 nMNPASS
Sodium/potassium-transporting ATPaseHomo sapiensP54710= 8.0 nMNPASS
OVCAR-3Homo sapiens= 117.1 nM|= 120.0 nMNPASS
HCT-116Homo sapiens= 440.0 nM|= 740.0 nMNPASS
NCI/ADR-RESHomo sapiens= 440.0 nMNPASS
A549Homo sapiens= 440.0 nMNPASS
ATP-binding cassette sub-family C member 2Homo sapiensQ92887>133000 nMBindingDB
ATP-binding cassette sub-family C member 3Homo sapiensO15438>133000 nMBindingDB
ATP-binding cassette sub-family C member 4Homo sapiensO15439>133000 nMBindingDB
Bile salt export pumpHomo sapiensO95342<10000 nM|31000 nM|< 10000.0 nM|= 31000.0 nMBindingDB, NPASS
NON-PROTEIN TARGET= 440.0 nM|= 410.0 nM|= 100.0 nMNPASS
Canalicular multispecific organic anion transporter 2Homo sapiensO15438> 133000.0 nMNPASS
DU-145Homo sapiens= 440.0 nMNPASS
HT-29Homo sapiens= 4070.0 nM|= 67.6 nM|= 68.0 nMNPASS
Canalicular multispecific organic anion transporter 1Homo sapiensQ92887> 133000.0 nMNPASS
K562Homo sapiens= 6.4 nMNPASS
KURAMOCHIHomo sapiens= 5911.0 nMNPASS
MCF7Homo sapiens= 10.2 nM|= 440.0 nM|= 20.0 nMNPASS
MDA-MB-231Homo sapiens= 482.0 nM|= 480.0 nMNPASS
MDA-MB-435Homo sapiens= 43.3 nM|= 43.0 nMNPASS
Monoclonal antibody (mAb)= 0.6 nM= 0.1 nM|= 0.2 nMNPASS
Multidrug resistance-associated protein 4Homo sapiensO15439> 133000.0 nMNPASS
NCI-H460Homo sapiens= 440.0 nM|= 357.0 nMNPASS
Human herpesvirus 5Human herpesvirus 5= 23.3 nMNPASS