IMPPAT Phytochemical information: 
Makisterone A

Makisterone A
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Ultraspiracle isoform BLeptinotarsa decemlia1738 nMBindingDB
Protein ultraspiracleDrosophila melanogasterP201531380 nMBindingDB
Ecdysone receptor/Ultraspiracle proteinSpodoptera frugiperda389 nMBindingDB
Ecdysone receptor/UltraspiracleNezara viridula1380 nMBindingDB
Ecdysone receptorSpodoptera frugiperdaQ8MWR1= 389.05 nMNPASS
Ecdysone receptorDrosophila melanogasterP34021112.2 nM|= 112.2 nMBindingDB, NPASS
Ecdysone receptorLeptinotarsa decemliaQ4W6C8= 1737.8 nMNPASS
Ecdysone receptorDrosophila melanogasterP20153= 1380.38 nMNPASS
Cytochrome P450 3A4Homo sapiensP08684>100000 nM|> 100000.0 nMBindingDB, NPASS
Ecdysone receptorNezara viridulaE5L6Y0= 1380.38 nMNPASS