| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| P388 | Mus musculus | | | = 36800.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 117600.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 74500.0 nM | | | NPASS |
| Matrix metalloproteinase 9 | Homo sapiens | P14780 | | = 7.95 ug.mL-1 | | | NPASS |
| Matrix metalloproteinase-9 | Homo sapiens | P14780 | | 27800 nM | | | BindingDB |
| Nuclear hormone receptor family member daf-12 | Caenorhabditis elegans | G5EFF5 | | 67574 nM | | | BindingDB |
| Oxysterols receptor LXR-beta | Homo sapiens | P55055 | | 67574 nM | | | BindingDB |
| Phosphodiesterase 5A | Homo sapiens | O76074 | | = 1230.0 nM | | | NPASS |
| Serotonin 1a (5-HT1a) receptor | Homo sapiens | P08908 | | | | > 100000.0 nM | NPASS |
| cGMP-specific 3',5'-cyclic phosphodiesterase | Homo sapiens | O76074 | | 1230 nM | | | BindingDB |
| Prostaglandin G/H synthase 1 | Homo sapiens | P23219 | | 8700 nM | | | BindingDB |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 300 nM|280 nM | | | BindingDB |
| RKO | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | = 18900.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 1 | Rattus norvegicus | O35433 | 2060 nM | | | | BindingDB |
| LXR-beta | Homo sapiens | P55055 | | > 67574.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 10000.0 nM | | | NPASS |
| LS174T | Homo sapiens | | | = 6100.0 nM | | | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 300.0 nM|= 280.0 nM | | | NPASS |
| HeLa | Homo sapiens | | = 26100.0 nM | | | | NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 731.9 nM | | | NPASS |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | | | | >100000 nM | BindingDB |
| Aorta | Rattus norvegicus | | = 1050.0 nM|= 1750.0 nM|= 1330.0 nM|= 29.7 nM|= 156.0 nM | | | | NPASS |
| CCD-18Co | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| CCD-841CoN | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Cholinesterase | Equus caballus | P81908 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| Cyclooxygenase-1 | Homo sapiens | P23219 | | = 8700.0 nM | | | NPASS |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | 260 nM|= 260.0 nM | | | BindingDB, NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | 55 nM|= 55.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | | | 107700 nM|= 107700.0 nM | BindingDB, NPASS |
| Danio rerio | Danio rerio | | | = 25490.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 31100.0 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HUVEC | Homo sapiens | | | = 16540.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 118000.0 nM | | | NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 22 nM|= 22.0 nM | | | BindingDB, NPASS |