
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | = 10000.0 nM|= 3400.0 nM | NPASS | |||
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | 15000 nM | BindingDB | |||
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | 3400 nM|10000 nM | BindingDB | |||
| GABA-A receptor; anion channel | Rattus norvegicus | O09028|P15431|P18506|P18508|P19969|P20236|P23574|P23576|P28471|P28473|P30191|P62813|P63079|P63138|Q91ZM7|Q9ES14 | = 570.0 nM | NPASS | |||
| P-glycoprotein 1 | Homo sapiens | P08183 | = 15000.0 nM | NPASS | |||
| Tankyrase-1 | Homo sapiens | O95271 | > 10000.0 nM | NPASS |