| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Mucosa-associated lymphoid tissue lymphoma translocation protein 1 | Homo sapiens | Q9UDY8 | | 1200 nM|1900 nM|= 1200.0 nM|= 1900.0 nM | | | BindingDB, NPASS |
| NCI-H596 | | | | = 23000.0 nM | | | NPASS |
| NCI-H596 | Homo sapiens | | | = 27000.0 nM | | | NPASS |
| NADPH--cytochrome P450 reductase | Homo sapiens | P16435 | | 11000 nM|= 11000.0 nM | | | BindingDB, NPASS |
| NAD(P)H dehydrogenase [quinone] 1 | Homo sapiens | P15559 | | >10000 nM|3400 nM|3000 nM | | | BindingDB |
| MOLT-4 | Homo sapiens | | | = 780.0 nM | | | NPASS |
| Lysine-specific demethylase 4D-like | Homo sapiens | B2RXH2 | | = 3000.0 nM | | = 3550.0 nM | NPASS |
| MDA-MB-435 | Homo sapiens | | | = 0.06 ug.mL-1|= 250.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 4300.0 nM|= 1390.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 9960.0 nM | = 800.0 nM|= 500.0 nM|= 710.0 nM | | | NPASS |
| Lysine-specific demethylase 4E | Homo sapiens | B2RXH2 | | 3000 nM | | 3550 nM | BindingDB |
| Nuclear factor NF-kappa-B complex | Homo sapiens | Q04206 | | = 4000.0 nM | | | NPASS |
| MDCK | Canis lupus familiaris | | | = 13500.0 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 1900.0 nM | | | NPASS |
| Quinone reductase 1) | Homo sapiens | P15559 | | = 3400.0 nM|> 10000.0 nM|= 3000.0 nM | | | NPASS |
| PBMC | Homo sapiens | | | > 20600.0 nM|= 2100.0 nM|> 20630.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | = 1130.0 nM | = 1650.0 nM|= 1820.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 10000.0 nM|= 3162.28 nM|= 12589.25 nM|= 3981.07 nM|= 7943.28 nM|= 6309.57 nM|= 20500.0 nM | | | NPASS |
| Protein-glutamine gamma-glutamyltransferase 2 | Homo sapiens | P21980 | | 1.8e+3 nM | | | BindingDB |
| LoVo | Homo sapiens | | | = 300.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 4060.0 nM|= 470.0 nM | | | NPASS |
| Replicase polyprotein 1ab | 2019-nCoV | P0DTD1 | | 13330 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | = 610.0 nM | | | NPASS |
| SF-295 | Homo sapiens | | | = 0.22 ug.mL-1|= 910.0 nM|= 950.0 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 600.0 nM | | | NPASS |
| Thiosulfate sulfurtransferase | Homo sapiens | Q16762 | | 120 nM|= 120.0 nM | | | BindingDB, NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 24700.0 nM|= 391500.0 nM|< 3100.0 nM|= 61300.0 nM | | | NPASS |
| Tyrosyl-DNA phosphodiesterase 2 | Homo sapiens | O95551 | | 970 nM|= 970.0 nM | | | BindingDB, NPASS |
| OVCAR-8 | Homo sapiens | | | = 1160.0 nM | | | NPASS |
| Liver carboxylesterase 1 | Homo sapiens | P23141 | | | | 1220 nM | BindingDB |
| NON-PROTEIN TARGET | | | | = 2200.0 nM|= 2000.0 nM|= 1600.0 nM|= 950.0 nM|= 4000.0 nM|= 400.0 nM|= 600.0 nM|= 300.0 nM|< 10.0 nM|= 391500.0 nM|= 1570.0 nM|= 870.0 nM|= 1650.0 nM|= 250.0 nM|= 1160.0 nM|> 20630.0 nM|= 25310.0 nM | | | NPASS |
| Leishmania infantum | Leishmaitum | | | = 1130.0 nM|= 670.0 nM | | | NPASS |
| 1A9 | Homo sapiens | | | = 800.0 nM|> 800.0 nM | | | NPASS |
| 60 kDa chaperonin | Escherichia coli (strain K12) | P0A6F5 | | > 250000.0 nM | | | NPASS |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens | P10809 | | 2100 nM | | | BindingDB |
| A549 | Homo sapiens | | = 4210.0 nM | = 1500.0 nM|= 5700.0 nM|= 7000.0 nM|= 25000.0 nM|= 3700.0 nM|= 800.0 nM|= 3100.0 nM|= 1960.0 nM|= 3320.0 nM|= 6000.0 nM|= 29000.0 nM|= 16000.0 nM | | | NPASS |
| A549/TR | Homo sapiens | | | = 1900.0 nM|= 11000.0 nM | | | NPASS |
| Acyl coenzyme A:cholesterol acyltransferase | Homo sapiens | P23141 | | | | = 1220.0 nM | NPASS |
| CAKI-1 | Homo sapiens | | | > 5000.0 nM | | | NPASS |
| Carboxylesterase 2 | Homo sapiens | O00748 | | | | = 109.0 nM | NPASS |
| Caspase-1 | Homo sapiens | P29466 | | 1.69e+3 nM | | | BindingDB |
| Chaperonin GroEL | Escherichia coli | | | >250000 nM | | | BindingDB |
| Co-chaperonin GroES | Escherichia coli | | | 590 nM|1300 nM | | | BindingDB |
| Cocaine esterase | Homo sapiens | O00748 | | | | 109 nM | BindingDB |
| GroEL/GroES | Escherichia coli | | | = 590.0 nM|= 1300.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 870.0 nM|= 970.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 7.4 nM | | | NPASS |
| J774.A1 | Mus musculus | | | > 200.0 ug.mL-1 | | | NPASS |
| Leishmania amazonensis | Leishmaamazonensis | | | = 1390.0 nM|= 2900.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 11900.0 nM|= 4540.0 nM|= 9600.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 1200.0 nM|= 1800.0 nM|= 1000.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 1600.0 nM | | | NPASS |
| HCT-8 | Homo sapiens | | | = 0.2 ug.mL-1|= 830.0 nM | | | NPASS |
| Indoleamine 2,3-dioxygenase 1 | Homo sapiens | P14902 | | 440 nM|1000 nM | | 100 nM | BindingDB |
| Indoleamine 2,3-dioxygenase | Homo sapiens | P14902 | | = 440.0 nM|= 1000.0 nM | | = 100.0 nM | NPASS |
| Leptomonas seymouri | Leptomonas seymouri | | | = 400.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 2830.0 nM | | | NPASS |
| HaCaT | Homo sapiens | | | = 700.0 nM|= 900.0 nM | | | NPASS |
| HSP60/HSP10 | Homo sapiens | | | = 2100.0 nM | | | NPASS |
| HOS | Homo sapiens | | | = 1400.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 270.0 nM|= 0.4 ug.mL-1|= 1650.0 nM|= 1570.0 nM | | | NPASS |
| Human herpesvirus 4 | Human herpesvirus 4 | | | = 210300.0 nM | | | NPASS |